null
SMILES Cc1nnn2CCN(Cc3cccc(Br)c3)c3ccccc3-c12
InChI Key InChIKey=UYRUHHLEYUGTMC-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50285938
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research
Curated by ChEMBL
Walter and Eliza Hall Institute of Medical Research
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 3(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research
Curated by ChEMBL
Walter and Eliza Hall Institute of Medical Research
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of human His-tagged Brd3 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research
Curated by ChEMBL
Walter and Eliza Hall Institute of Medical Research
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 2 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research
Curated by ChEMBL
Walter and Eliza Hall Institute of Medical Research
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Inhibition of human His-tagged Brd4 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 2(Homo sapiens (Human))
Walter and Eliza Hall Institute of Medical Research
Curated by ChEMBL
Walter and Eliza Hall Institute of Medical Research
Curated by ChEMBL
Affinity DataIC50: 129nMAssay Description:Inhibition of human His-tagged Brd2 bromodomain 1 expressed in Escherichia coli BL21 (DE3) preincubated for 30 mins followed by addition of biotinyla...More data for this Ligand-Target Pair