null
SMILES CC(C)C[C@H](NC(=O)[C@H](Cc1ccc(OP(O)(O)=O)cc1)NC(=O)c1ccc(cc1)C#N)C(=O)Nc1cc(cc(c1)-c1ccc(cc1)C(N)=O)C(=O)NCc1ccccc1
InChI Key InChIKey=PEXNGCNKHRPGFE-YDAXCOIMSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50337198
TargetSignal transducer and activator of transcription 3(Mus musculus (mouse))
University of Toronto
Curated by ChEMBL
University of Toronto
Curated by ChEMBL
Affinity DataKi: 9.00E+3nMAssay Description:Displacement of 5-carboxyfluorescein-GpYLPQTV-NH2 from mouse recombinant His-tagged STAT3-SH2 domain expressed in Escherichia coli BL21 (DE3) by fluo...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 1(Mus musculus)
University of Toronto
Curated by ChEMBL
University of Toronto
Curated by ChEMBL
Affinity DataKi: 1.65E+4nMAssay Description:Displacement of 5-carboxyfluorescein-GpYDKPHVL-NH2 from mouse recombinant His-tagged STAT1-SH2 domain expressed in Escherichia coli BL21 (DE3) by flu...More data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Mus musculus (mouse))
University of Toronto
Curated by ChEMBL
University of Toronto
Curated by ChEMBL
Affinity DataKd: 205nMAssay Description:Inhibition of mouse recombinant SH2 domain of His-tagged full-length STAT3 by surface plasmon resonance assayMore data for this Ligand-Target Pair
TargetSignal transducer and activator of transcription 3(Mus musculus (mouse))
University of Toronto
Curated by ChEMBL
University of Toronto
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of STAT3 dimerization in mouse NIH3T3 cells expressing v-Src assessed as disruption of STAT3-STAT3: DNA complexation in nucleus after 30 m...More data for this Ligand-Target Pair