null
SMILES Nc1nccc(n1)-c1c[nH]c2c(Br)cccc12
InChI Key InChIKey=VHKRTWNLRWRPSB-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50347796
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Inhibition of human recombinant GST-tagged CLK1 using GRSRSRSRSRSR as substrateMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 68nMAssay Description:Inhibition of rat recombinant GST-tagged DYRK1A using myelin protein as substrate and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6...More data for this Ligand-Target Pair
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 2.25E+4nMAssay Description:Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Clermont Universite£
Curated by ChEMBL
Clermont Universite£
Curated by ChEMBL
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of human recombinant CDK5/p25 using Histone H1 and [gamma32]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair