null
SMILES Clc1ccc(CCNC(=O)Nc2ccc3[nH]ncc3c2)cc1
InChI Key InChIKey=OMZOSZCBUJIGIG-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50382689
TargetRho-associated protein kinase 1 [1-535](Homo sapiens (Human))
H. Lee Moffin Cancer Center and Research Institute, Inc.
US Patent
H. Lee Moffin Cancer Center and Research Institute, Inc.
US Patent
Affinity DataIC50: 2.20E+3nMpH: 7.5 T: 2°CAssay Description:A robust FRET-based, enzyme-coupled assay format, Z-Lyte® Kinase Assay Ser/Thr 13 Peptide Kit (Invitrogen, cat. PV3793), was employed in this stu...More data for this Ligand-Target Pair
TargetRho-associated protein kinase 1(Homo sapiens (Human))
H. Lee Moffitt Cancer Center and Research Institute
Curated by ChEMBL
H. Lee Moffitt Cancer Center and Research Institute
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human His-puritin-tagged ROCK1 expressed in Sf9 cells after 1 hr by FRET-based enzyme-coupled assayMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center and Research Institute
Curated by ChEMBL
H. Lee Moffitt Cancer Center and Research Institute
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of ROCK2 after 1 hr by FRET-based enzyme-coupled assayMore data for this Ligand-Target Pair
TargetRho-associated protein kinase 2 [1-552](Homo sapiens (Human))
H. Lee Moffin Cancer Center and Research Institute, Inc.
US Patent
H. Lee Moffin Cancer Center and Research Institute, Inc.
US Patent
Affinity DataIC50: 1.10E+3nMpH: 7.5 T: 2°CAssay Description:A robust FRET-based, enzyme-coupled assay format, Z-Lyte® Kinase Assay Ser/Thr 13 Peptide Kit (Invitrogen, cat. PV3793), was employed in this stu...More data for this Ligand-Target Pair