null
SMILES FC(F)(F)COc1ccc(cn1)C(=O)N[C@@H]1COc2cccc(-c3cccnc3)c2C1
InChI Key InChIKey=AQNRVBHBIZRPCK-INIZCTEOSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50390096
Affinity DataIC50: 3.16E+3nMAssay Description:Inhibition of human NaV1.5 expressed in CHO cells by IonWorks assayMore data for this Ligand-Target Pair
Affinity DataIC50: 79.4nMAssay Description:Inhibition of human NaV1.7 expressed in HEK293 cells by whole-cell voltage clamp assayMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
AstraZeneca
Curated by ChEMBL
AstraZeneca
Curated by ChEMBL
Affinity DataIC50: 2.51E+4nMAssay Description:Inhibition of human ERG expressed in CHO cells by IonWorks HT assayMore data for this Ligand-Target Pair