null
SMILES Cc1cc(C)cc(c1)-c1nc(NC(=O)c2cccnc2)sc1-c1ccncc1
InChI Key InChIKey=YDXZLBYHXZOWOC-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 22 hits for monomerid = 50397728
Affinity DataKi: 0.360nMAssay Description:Displacement of [125I]I-AB-MECA from human recombinant adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counterMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [125I]I-AB-MECA from human rat adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counterMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor expressed in HEK293 cells incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.5nMAssay Description:Displacement of [125I]I-AB-MECA from rat adenosine A3 receptor expressed in HEK293 cells incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 9.60nMAssay Description:Displacement of [125I]I-AB-MECA from mouse adenosine A3 receptor expressed in HEK293 cells incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 121nMAssay Description:Displacement of [3H] ZM241385 from human adenosine A2A receptor expressed in HEK293 cells incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 162nMAssay Description:Displacement of [3H] DPCPX from human adenosine A1 receptor expressed in HEK293 cells incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 163nMAssay Description:Displacement of [3H] DPCPX from rat adenosine A2B receptor expressed in HEK293 cells incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 189nMAssay Description:Displacement of [3H] DPCPX from mouse adenosine A2B receptor expressed in HEK293 cells incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:Displacement of [3H] DPCPX from human adenosine A2B receptor expressed in HEK293 cells incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 333nMAssay Description:Displacement of [3H] DPCPX from rat adenosine A1 receptor expressed in HEK293 cells incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 411nMAssay Description:Displacement of [3H] DPCPX from mouse adenosine A1 receptor expressed in HEK293 cells incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: >666nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cells after 60 mins by gamma counterMore data for this Ligand-Target Pair
Affinity DataKi: 790nMAssay Description:Binding affinity to human 5-HT2C receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: >826nMAssay Description:Displacement of [3H]CGS21680 from human recombinant adenosine A2A receptor expressed in CHO cells after 60 mins by gamma counterMore data for this Ligand-Target Pair
Affinity DataKi: 830nMAssay Description:Displacement of [3H] ZM241385 from mouse adenosine A2A receptor expressed in HEK293 cells incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 960nMAssay Description:Binding affinity to human 5-HT2A receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.15E+3nMAssay Description:Displacement of [3H] ZM241385 from rat adenosine A2A receptor expressed in HEK293 cells incubated for 60 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.70E+3nMAssay Description:Binding affinity to human M5 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.550nMAssay Description:Binding affinity to human adenosine A3 receptor expressed in HEK293 cells measured by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKd: 3.70nMAssay Description:Binding affinity to mouse adenosine A3 receptor expressed in HEK293 cells measured by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKd: 2.80nMAssay Description:Binding affinity to rat adenosine A3 receptor expressed in HEK293 cells measured by radioligand binding assayMore data for this Ligand-Target Pair