null
SMILES Clc1ccccc1N1CCN(CC1)C(=O)[C@H](CCCCNC(=O)C=C)NC(=O)OCc1ccccc1
InChI Key InChIKey=KYVYJVRZPFRADU-QHCPKHFHSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50400625
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
University of Ottawa
Curated by ChEMBL
University of Ottawa
Curated by ChEMBL
Affinity DataKi: 1.74E+4nMAssay Description:Irreversible inhibition of human TG2 using AL5 as substrate by colorimetric assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.70E+4nMAssay Description:Inhibition of coagulation factor 13aMore data for this Ligand-Target Pair
Affinity DataIC50: 1.29E+4nMAssay Description:Inhibition of transglutaminase 1More data for this Ligand-Target Pair
TargetProtein-glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
University of Ottawa
Curated by ChEMBL
University of Ottawa
Curated by ChEMBL
Affinity DataIC50: 62nMAssay Description:Irreversible inhibition of transglutaminase 2More data for this Ligand-Target Pair
Affinity DataIC50: 6.90E+4nMAssay Description:Inhibition of transglutaminase 6More data for this Ligand-Target Pair
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of transglutaminase 3More data for this Ligand-Target Pair