null
SMILES Cc1ccc(cc1)-c1c(\C=C(/C#N)C(=O)NC(C)(C)C)n(CCCO)c2ncnc(N)c12
InChI Key InChIKey=SVXJIKFFHBDTNV-SFQUDFHCSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50403059
TargetRibosomal protein S6 kinase alpha-3(Homo sapiens (Human))
Covalution Pharma BV
Curated by ChEMBL
Covalution Pharma BV
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of RSK2 transfected in HEK293 cellsMore data for this Ligand-Target Pair
TargetRibosomal protein S6 kinase alpha-3 [399-740](Homo sapiens (Human))
THE REGENTS OF THE UNIVERSITY OF CALIFORNIA
US Patent
THE REGENTS OF THE UNIVERSITY OF CALIFORNIA
US Patent
Affinity DataIC50: 4.5nMpH: 8.0 T: 2°CAssay Description:RSK2 CTD and His6-ERK2 were expressed and purified as described (Cohen et al., Science, 308: 1318). The C436V mutant of RSK2 CTD was generated by Qui...More data for this Ligand-Target Pair