null
SMILES CC(C)n1nc(Cc2cccc(NS(=O)(=O)C=C)c2)c2c(N)ncnc12
InChI Key InChIKey=AAFALAKLPXVLIO-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50403061
TargetProto-oncogene tyrosine-protein kinase Src [251-533](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 5.00E+3nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533,T338C](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 150nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))
Covalution Pharma BV
Curated by ChEMBL
Covalution Pharma BV
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of chicken c-Src using IYGEFKKK peptide as a substrate and [32P]ATP by fluorescence analysisMore data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533,V323S,T338C](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 424nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase Src [251-533,V323A,T338C](Gallus gallus (Chicken))
The Regents of the University of California
US Patent
The Regents of the University of California
US Patent
Affinity DataIC50: 207nMpH: 8.0Assay Description:In vitro kinase assays for c-Src variants were performed in 50 mM Tris (pH 8.0), 10 mM MgCl2 and 1 mg/mL BSA. When obtaining kinetic parameters (kcat...More data for this Ligand-Target Pair