null
SMILES CN1C(=O)CCc2c(CCN3CCN(CC3)c3cccc4nc(C)ccc34)c(C)ccc12
InChI Key InChIKey=PDLXDQOODGXTSQ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50417421
Affinity DataKi: 0.631nMAssay Description:Antagonist activity at human 5-HT1A receptor expressed in HEK293 cells assessed as inhibition of GTPgammaS binding by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Antagonist activity at human 5-HT1D receptor expressed in CHO cells assessed as inhibition of GTPgammaS binding by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 25.1nMAssay Description:Displacement of [3H]-citalopram in human SERT expressed in LLCPK cells by filtration assayMore data for this Ligand-Target Pair
Affinity DataKi: 794nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
Affinity DataEC50: 398nMAssay Description:Agonist activity at human 5-HT1B receptor expressed in CHO cells assessed as stimulation of GTPgammaS binding by scintillation proximity assayMore data for this Ligand-Target Pair