null
SMILES Cc1ccc2nc(NC(=O)CSc3nc4CCSc4c(=O)n3Cc3ccccc3)sc2c1
InChI Key InChIKey=VBUSMYOJWTVVPF-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50455468
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital
Curated by ChEMBL
Ulm University Hospital
Curated by ChEMBL
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of full-length rat GST-tagged CK1delta using alpha-casein as substrate after 30 mins in presence of [gamma-32P]-ATP by Cherenkov counting ...More data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital
Curated by ChEMBL
Ulm University Hospital
Curated by ChEMBL
Affinity DataIC50: 420nMAssay Description:Inhibition of rat recombinant CK1delta kinase domain using alpha-casein as substrate after 30 mins in presence of [gamma-32P]-ATP by Cherenkov counti...More data for this Ligand-Target Pair
Affinity DataIC50: 7.34E+3nMAssay Description:Inhibition of human recombinant CK1epsilon using alpha-casein as substrate after 30 mins in presence of [gamma-32P]-ATP by Cherenkov counting methodMore data for this Ligand-Target Pair
TargetCasein kinase I isoform delta(Rattus norvegicus (rat))
Ulm University Hospital
Curated by ChEMBL
Ulm University Hospital
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of rat GST-tagged CK1delta M82F mutant at 10 uM using alpha-casein as substrate after 30 mins in presence of [gamma-32P]-ATP by Cherenkov ...More data for this Ligand-Target Pair