null
SMILES Cn1cc(cn1)-c1cc2CC[C@]3(NC(=O)N(CC(=O)N4Cc5cc(F)ccc5OC[C@H]4C(F)(F)F)C3=O)c2cn1
InChI Key InChIKey=WPGMGBWETYWLPU-OFVILXPXSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 50506378
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Chinese Academy of Sciences
Curated by ChEMBL
Chinese Academy of Sciences
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of p300 (unknown origin) using histone H3 (1 to 21 residues) as substrate preincubated for 15 mins followed by substrate and [3H]acetyl-Co...More data for this Ligand-Target Pair