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SMILES [Na;v0+].[H][C@@]12[#6]-[#8]P([#8-])(=O)[#8][C@@]1([H])[#6@@H](-[#8])-[#6@@H](-[#8]2)-n1c(Br)cc2c(-[#7])ncnc12
InChI Key InChIKey=VQQUWDVOCJKUMP-YCSZXMBFSA-M
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50526580
TargetRap guanine nucleotide exchange factor 4(Mus musculus)
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 300nMAssay Description:Inhibition of 8Fluo-cAMP binding to DEP domain deficient mouse EPAC2 (280 to 988 residues) measured after 5 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetCyclic nucleotide-gated olfactory channel(Rattus norvegicus)
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 630nMAssay Description:Activation of recombinant rat CNGA2/CNGA4/CNGB1b heterotetramer expressed in Xenopus laevis oocyte assessed as increase in current amplitude by patch...More data for this Ligand-Target Pair
TargetCyclic nucleotide-gated olfactory channel(Rattus norvegicus)
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 6.40E+3nMAssay Description:Activation of recombinant rat CNGA2 expressed in Xenopus laevis oocyte assessed as increase in current amplitude by patch-clamp electrophysiology met...More data for this Ligand-Target Pair
TargetRap guanine nucleotide exchange factor 3(Homo sapiens (Human))
University Hospital Jena
Curated by ChEMBL
University Hospital Jena
Curated by ChEMBL
Affinity DataEC50: 530nMAssay Description:Inhibition of 8Fluo-cAMP binding to recombinant human His-tagged EPAC1 (157 to 881 residues) expressed in Escherichia coli measured after 5 mins by f...More data for this Ligand-Target Pair