null
SMILES OC(=O)C(F)(F)F.OC(=O)C(F)(F)F.OC(=O)C(F)(F)F.OC(=O)C(F)(F)F.[H][C@@]1(N)Cc2ccc(NC(=O)CCN3CCN(CC3)CCC(=O)Nc3ccc(C[C@]([H])(NC1=O)C(=O)NCc1ccc(cc1)C(N)=N)cc3)cc2
InChI Key InChIKey=SXCYORRQBGIHCT-NTNLIPOVSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 10 hits for monomerid = 50532395
Affinity DataKi: 13nMAssay Description:Inhibition of human plasmin using Mes-DSer(Bzl)-Phe-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition of human plasmin using Mes-DSer(Bzl)-Phe-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.45E+4nMAssay Description:Inhibition of human plasma kallikrein using Mes-DArg-Pro-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.45E+4nMAssay Description:Inhibition of human plasma kallikrein using Mes-DArg-Pro-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 6.08E+4nMAssay Description:Inhibition of bovine thrombin using Tos-Gly-Pro-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 6.08E+4nMAssay Description:Inhibition of bovine thrombin using Tos-Gly-Pro-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
TargetVitamin K-dependent protein C(Homo sapiens (Human))
Philipps University Marburg
Curated by ChEMBL
Philipps University Marburg
Curated by ChEMBL
Affinity DataKi: 1.06E+5nMAssay Description:Inhibition of human activated Protein C using Mes-DArg-Pro-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
TargetVitamin K-dependent protein C(Homo sapiens (Human))
Philipps University Marburg
Curated by ChEMBL
Philipps University Marburg
Curated by ChEMBL
Affinity DataKi: 1.06E+5nMAssay Description:Inhibition of human activated Protein C using Mes-DArg-Pro-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 4.05E+5nMAssay Description:Inhibition of human f10a using Mes-DArg-Pro-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 4.05E+5nMAssay Description:Inhibition of human f10a using Mes-DArg-Pro-Arg-AMC as substrate by Dixon plot analysisMore data for this Ligand-Target Pair