null
SMILES COc1cc(cc(OC)c1OC)-c1cncc(c1C)-c1ccc(cc1)C1=CCN(C)CC1
InChI Key InChIKey=XIKOWUNWIVBZIV-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50544415
TargetActivin receptor type-1(Homo sapiens (Human))
Ontario Institute for Cancer Research
Curated by ChEMBL
Ontario Institute for Cancer Research
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of human ALK2 using casein as substrate in presence of [gamma-33P]-ATP by radiometric hotspot assayMore data for this Ligand-Target Pair
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Ontario Institute for Cancer Research
Curated by ChEMBL
Ontario Institute for Cancer Research
Curated by ChEMBL
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibition of recombinant human ALK5 expressed in HEK293 cells transfected with CAGA-luciferase and Renilla luciferase reporter after 24 hrs by dual ...More data for this Ligand-Target Pair
TargetActivin receptor type-1(Homo sapiens (Human))
Ontario Institute for Cancer Research
Curated by ChEMBL
Ontario Institute for Cancer Research
Curated by ChEMBL
Affinity DataIC50: 102nMAssay Description:Competitive displacement of PBI-6908 from nanoluciferase-fused ALK2 (unknown origin) expressed in HEK293 cells incubated for 2 hrs by NanoBRET NanoGl...More data for this Ligand-Target Pair
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Ontario Institute for Cancer Research
Curated by ChEMBL
Ontario Institute for Cancer Research
Curated by ChEMBL
Affinity DataIC50: 2.52E+3nMAssay Description:Inhibition of human ALK5 using casein as substrate in presence of [gamma-33P]-ATP by radiometric hotspot assayMore data for this Ligand-Target Pair