BindingDB

null

SMILES COc1cc(ccc1-c1cn(C\C=C\C)c(=O)c2[nH]ccc12)C(C)(C)O

InChI Key

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 47 hits for monomerid = 50615275

Bromodomain-containing protein 9(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

IC50: 48nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
GoogleScholar

Platelet-derived growth factor receptor alpha/beta(Mus musculus (mouse))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

IC50: 4.00E+3nMMore data for this Ligand-Target Pair

MMDB KEGG
UniProtKB/SwissProt
DrugBank GoogleScholar

Bromodomain-containing protein 4(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

IC50: 2.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Chromatin remodeling regulator CECR2(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

IC50: 2.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
GoogleScholar

Transcription initiation factor TFIID subunit 1(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

IC50: 2.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
GoogleScholar

Bromodomain-containing protein 9(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

EC50: 190nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
GoogleScholar

Stromelysin-3(Mus musculus)TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

IC50: 1.02E+4nMMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank GoogleScholar

ATPase family AAA domain-containing protein 2(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: >1.00E+4nMMore data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

ATPase family AAA domain-containing protein 2B(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: >1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
GoogleScholar

Bromodomain adjacent to zinc finger domain protein 2A(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: >1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
GoogleScholar

Bromodomain adjacent to zinc finger domain protein 2B(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: >1.00E+4nMMore data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Bromodomain-containing protein 1(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: >1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
GoogleScholar

Bromodomain-containing protein 2(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: 2.70E+3nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

Bromodomain-containing protein 2(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: 2.80E+3nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

Bromodomain-containing protein 2(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: 3.30E+3nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
B.MOAD GoogleScholar

Bromodomain-containing protein 3(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: 3.20E+3nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Bromodomain-containing protein 3(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: 5.50E+3nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Bromodomain-containing protein 3(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: 4.00E+3nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Bromodomain-containing protein 4(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: 1.60E+3nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Bromodomain-containing protein 4(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: 1.70E+3nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Bromodomain-containing protein 4(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: 3.70E+3nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Bromodomain-containing protein 4(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: 580nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Bromodomain-containing protein 7(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: 340nMMore data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Bromodomain-containing protein 8(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: >1.00E+4nMMore data for this Ligand-Target Pair

UniProtKB/SwissProt
GoogleScholar

Bromodomain-containing protein 8(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: >1.00E+4nMMore data for this Ligand-Target Pair

UniProtKB/SwissProt
GoogleScholar

Bromodomain-containing protein 9(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: 25nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
GoogleScholar

Bromodomain testis-specific protein(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: 830nMMore data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Bromodomain testis-specific protein(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: 1.20E+3nMMore data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Bromodomain testis-specific protein(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: 2.60E+3nMMore data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Peregrin(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: >1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
GoogleScholar

Bromodomain and PHD finger-containing protein 3(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: >1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
GoogleScholar

Chromatin remodeling regulator CECR2(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: >1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
GoogleScholar

CREB-binding protein(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: 3.50E+3nMMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Histone acetyltransferase p300(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: 4.50E+3nMMore data for this Ligand-Target Pair

PDB MMDB
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Nucleosome-remodeling factor subunit BPTF(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: >1.00E+4nMMore data for this Ligand-Target Pair

PDB MMDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Histone acetyltransferase KAT2A(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: 410nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Protein polybromo-1(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: 7.60E+3nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
GoogleScholar

Protein polybromo-1(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: >1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
GoogleScholar

Histone acetyltransferase KAT2B(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: >1.00E+4nMMore data for this Ligand-Target Pair

PDB MMDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank GoogleScholar

Probable global transcription activator SNF2L2(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: >1.00E+4nMMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Transcription activator BRG1(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: >1.00E+4nMMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Transcription initiation factor TFIID subunit 1(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: >1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
GoogleScholar

Transcription initiation factor TFIID subunit 1-like(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: >1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
GoogleScholar

Transcription intermediary factor 1-alpha(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: >1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
GoogleScholar

E3 ubiquitin-protein ligase TRIM33(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: >1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
GoogleScholar

Bromodomain and WD repeat-containing protein 1(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

Kd: >1.00E+4nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
GoogleScholar

Bromodomain-containing protein 4(Homo sapiens (Human))TBA

PNG

BDBM50615275(CHEMBL5282240)copy SMILES

IC50: 5.10E+3nMMore data for this Ligand-Target Pair

PDB KEGG
UniProtKB/SwissProt
B.MOAD antibodypedia GoogleScholar

Targets 30 ▿
- Bromodomain-containing protein 4 6
- Bromodomain-containing protein 3 3
- Bromodomain-containing protein 2 3
- Bromodomain testis-specific protein 3
- Bromodomain-containing protein 9 3
- Protein polybromo-1 2
- Transcription initiation factor TFIID subunit 1 2
- Bromodomain-containing protein 8 2
- Chromatin remodeling regulator CECR2 2
- ATPase family AAA domain-containing protein 2B 1
- Transcription initiation factor TFIID subunit 1-like 1
- Bromodomain and WD repeat-containing protein 1 1
- Bromodomain adjacent to zinc finger domain protein 2A 1
- Platelet-derived growth factor receptor alpha/beta 1
- Peregrin 1
- Bromodomain adjacent to zinc finger domain protein 2B 1
- Nucleosome-remodeling factor subunit BPTF 1
- Bromodomain and PHD finger-containing protein 3 1
- Bromodomain-containing protein 1 1
- E3 ubiquitin-protein ligase TRIM33 1
- Histone acetyltransferase p300 1
- Transcription activator BRG1 1
- ATPase family AAA domain-containing protein 2 1
- CREB-binding protein 1
- Histone acetyltransferase KAT2B 1
- Histone acetyltransferase KAT2A 1
- Bromodomain-containing protein 7 1
- Transcription intermediary factor 1-alpha 1
- Probable global transcription activator SNF2L2 1
- Stromelysin-3 1
Publications 0 ▿
Institutions 0 ▿
Affinity: 25 to 2.0E+4 nM▿
- IC50 7
- Kd 39
- EC50 1
- Affinity ≤ nM
Xtal structures: 0
Docked structures: 0
Catalog Cmpds: 0