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SMILES Fc1ccc2c(Cc3nnc(Cc4ccccc4)n3CCCc3c[nH]cn3)c[nH]c2c1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 9 hits for monomerid = 523758   

TargetSomatostatin receptor type 4(Homo sapiens (Human))TBA
LigandPNGBDBM523758(US11136312, Compound MM-I-89)copy SMILES
Affinity DataKi:  2.97nMAssay Description:Competitive radioligand binding experiments were performed using MEMBRANE TARGET Systems (Perkin-Elmer, Boston, Mass.) for human somatostatin recepto...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DB851BUS Patent
TargetSomatostatin receptor type 4(Homo sapiens (Human))TBA
LigandPNGBDBM523758(US11136312, Compound MM-I-89)copy SMILES
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21X0PubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))TBA
LigandPNGBDBM523758(US11136312, Compound MM-I-89)copy SMILES
Affinity DataKi:  1.83E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21X0PubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))TBA
LigandPNGBDBM523758(US11136312, Compound MM-I-89)copy SMILES
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21X0PubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))TBA
LigandPNGBDBM523758(US11136312, Compound MM-I-89)copy SMILES
Affinity DataKi: >1.00E+4nMAssay Description:Competitive radioligand binding experiments were performed using MEMBRANE TARGET Systems (Perkin-Elmer, Boston, Mass.) for human somatostatin recepto...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DB851BUS Patent
TargetSomatostatin receptor type 2(Homo sapiens (Human))TBA
LigandPNGBDBM523758(US11136312, Compound MM-I-89)copy SMILES
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21X0PubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))TBA
LigandPNGBDBM523758(US11136312, Compound MM-I-89)copy SMILES
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21X0PubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))TBA
LigandPNGBDBM523758(US11136312, Compound MM-I-89)copy SMILES
Affinity DataEC50:  2.80nMAssay Description:Measurement of forskolin stimulated inhibition of cAMP was performed via time-resolved fluorescence resonance energy transfer (TR-FRET) LANCE assay (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DB851BUS Patent
TargetSomatostatin receptor type 4(Homo sapiens (Human))TBA
LigandPNGBDBM523758(US11136312, Compound MM-I-89)copy SMILES
Affinity DataEC50:  2.80nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21X0PubMed