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SMILES Cc1cccc(Nc2ncc(cn2)-c2cncc(NC3CN(C3)C(=O)C=C)n2)n1

InChI Key

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 588169   

TargetEpidermal growth factor receptor(Homo sapiens (Human))TBA
LigandPNGBDBM588169(1-[3-[[6-[2-[(6- methyl-2- pyridyl)amino] pyrimidi...)copy SMILES
Affinity DataIC50: 54.9nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREENŽ Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2J38XD6US Patent
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))TBA
LigandPNGBDBM588169(1-[3-[[6-[2-[(6- methyl-2- pyridyl)amino] pyrimidi...)copy SMILES
Affinity DataIC50: 5.58nMAssay Description:The BTK and EGFR biochemical assays utilize LANTHASCREENŽ Eu Kinase Binding Assays from Thermo Fisher Scientific, measuring the binding of the kinase...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2J38XD6US Patent