null
SMILES OC(=O)CN1C(=S)S\C(=C/c2ccco2)C1=O
InChI Key InChIKey=DFCZJGAFQKNSEX-DAXSKMNVSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 8436
Affinity DataIC50: 1.40E+5nMAssay Description:Fluorescence peptide cleavage assay was performed in a 96-well plate. Each reaction contained MAPKKide, LF, and the small-molecule inhibitor. The C-t...More data for this Ligand-Target Pair
In DepthDetails
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
NAS of Ukraine
Curated by ChEMBL
NAS of Ukraine
Curated by ChEMBL
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of human ASK1 using MBP as substrate incubated for 10 mins prior to ATP addition measured after 20 mins by liquid scintillation counting a...More data for this Ligand-Target Pair