null
SMILES COc1cc2c(NC3CCN(C)CC3)cc(nc2cc1OCCCN1CCCC1)C1CCC(C)O1
InChI Key InChIKey=BZJGYMRAKCPWJV-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50281366
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias
Curated by ChEMBL
Universidad de Oviedo-Principado de Asturias
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of human G9a using biotinylated-H3K9 peptide as substrate after 1 hr in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
Universidad de Oviedo-Principado de Asturias
Curated by ChEMBL
Universidad de Oviedo-Principado de Asturias
Curated by ChEMBL
Affinity DataIC50: 1.37E+3nMAssay Description:Inhibition of human DNMT1 using polydeoxyinosine polydeoxycytosine DNA as substrate after 15 mins in presence of SAM by TR-FRET assayMore data for this Ligand-Target Pair