null
SMILES Oc1nc(nc2sc3CCCCc3c12)-c1ccccc1
InChI Key InChIKey=CDFWRIZOSNAGCV-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50250991
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center of Biotherapy
Curated by ChEMBL
Sichuan University and Collaborative Innovation Center of Biotherapy
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GST-tagged BRD4 bromodomain (unknown origin) using biotinylated histone H4KAc peptide (1 to 21 residues) as substrate by HTRF assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Sichuan University and Collaborative Innovation Center of Biotherapy
Curated by ChEMBL
Sichuan University and Collaborative Innovation Center of Biotherapy
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of His/thioredoxin-tagged human recombinant BRD4 bromodomain-1 (43 to 166 residues) expressed in Escherichia coli BL21 Star (DE3) pre-incu...More data for this Ligand-Target Pair