null
SMILES CN(CC#N)C(=O)c1ccc(cc1)-c1cn(C)c(=O)c2[nH]ccc12
InChI Key InChIKey=CFDRMWOIMXZRDV-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 310891
TargetBromodomain-containing protein 4 [42-168](Homo sapiens (Human))
Genentech, Inc.; Constellation Pharmaceuticals Inc.
US Patent
Genentech, Inc.; Constellation Pharmaceuticals Inc.
US Patent
Affinity DataIC50: 200nMAssay Description:His/Flag epitope tagged BRD4 BD142-168 was cloned, expressed, and purified to. BRD4 binding and inhibition was assessed by monitoring the engagement ...More data for this Ligand-Target Pair