null
SMILES CC(C)c1ccc2c(c1)oc1nc(N)c(cc1c2=O)C(O)=O
InChI Key InChIKey=ILCMMGSPXXYUSR-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 357909
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
THE REGENTS OF THE UNIVERSITY OF MICHIGAN
US Patent
THE REGENTS OF THE UNIVERSITY OF MICHIGAN
US Patent
Affinity DataIC50: 410nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
THE REGENTS OF THE UNIVERSITY OF MICHIGAN
US Patent
THE REGENTS OF THE UNIVERSITY OF MICHIGAN
US Patent
Affinity DataIC50: 302nMAssay Description:Inhibition of human TBK1 (1 to 657 residues) expressed in Baculovirus infected SF9 insect cells using myelin basic protein as substrate in presence o...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
THE REGENTS OF THE UNIVERSITY OF MICHIGAN
US Patent
THE REGENTS OF THE UNIVERSITY OF MICHIGAN
US Patent
Affinity DataIC50: 300nMAssay Description:Inhibition of human TBK1 (1 to 657 residues) expressed in Baculovirus infected SF9 insect cells using myelin basic protein as substrate in presence o...More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataIC50: 4.68E+3nMAssay Description:Inhibition of human IKKepsilon (1 to 655 residues) expressed in Baculovirus infected SF9 insect cells using myelin basic protein as substrate in pres...More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
University of Michigan
Curated by ChEMBL
University of Michigan
Curated by ChEMBL
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of human IKKepsilon (1 to 655 residues) expressed in Baculovirus infected SF9 insect cells using myelin basic protein as substrate in pres...More data for this Ligand-Target Pair