null
SMILES Nc1nc2CC[C@@H](Cc2s1)NC(=O)c1cc(Br)c[nH]1
InChI Key InChIKey=RCJXOQVSWUVVKP-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50095288
Affinity DataIC50: 5.20E+5nMAssay Description:Inhibition of Escherichia coli DNA gyrase using relaxed pNO1 plasmid and biotinylated oligonucelotide incubated for 30 mins by fluorescence based DNA...More data for this Ligand-Target Pair
TargetSodium channel protein type 3 subunit alpha(Homo sapiens (Human))
University of Ljubljana
Curated by ChEMBL
University of Ljubljana
Curated by ChEMBL
Affinity DataIC50: 2.60E+4nMAssay Description:Modulation of human Nav1.3 by automated patch clamp electrophysiology assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha(Homo sapiens (Human))
University of Ljubljana
Curated by ChEMBL
University of Ljubljana
Curated by ChEMBL
Affinity DataIC50: 1.80E+4nMAssay Description:Modulation of human Nav1.7 by automated patch clamp electrophysiology assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 5 subunit alpha(Homo sapiens (Human))
University of Ljubljana
Curated by ChEMBL
University of Ljubljana
Curated by ChEMBL
Affinity DataIC50: 2.10E+4nMAssay Description:Modulation of human Nav1.5 by automated patch clamp electrophysiology assayMore data for this Ligand-Target Pair
TargetSodium channel protein type 4 subunit alpha(Homo sapiens (Human))
University of Ljubljana
Curated by ChEMBL
University of Ljubljana
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Modulation of human Nav1.4 by automated patch clamp electrophysiology assayMore data for this Ligand-Target Pair