null

SMILES N[C@@H](Cc1ccc(O)cc1)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc1ccccc1)C(N)=O

InChI Key InChIKey=XIJHWXXXIMEHKW-LJWNLINESA-N

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 125 hits for monomerid = 50139013   

TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  0.00950nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain after 45 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2XBNPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  0.490nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain homogenates by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22809FJPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  0.690nMAssay Description:Binding affinity to mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474BPWPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  0.690nMAssay Description:Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W095DJPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  0.690nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B931SPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC038RPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  1.30nMAssay Description:Binding affinity to mu opioid receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z96DBPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]endomorphin-2 from mu opioid receptor in Wistar rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC038RPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  1.33nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosome membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B0264PubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  1.33nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain P2 synaptosomeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348K1FPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  1.35nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0MX9PubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52QR5PubMed
TargetMu-type opioid receptor(GUINEA PIG)
Clinical Research Institute of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  2.06nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23X856NPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  2.06nMAssay Description:Binding affinity towards mu receptor in rat brain using [3H]DAMGOMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2BC408MPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Displacement of [3H]DAMGO from rat cortex mu opioid receptor after 30 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B90RZPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Displacement of [3H]DAMGO from human recombinant MOR expressed in CHO cell membranes incubated for 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2697704PubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]DAMGO from FLAG-tagged mu opioid receptor expressed in HEK293 cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154S8PubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain membranes by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2D79FCGPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  3.70nMAssay Description:Inhibition of [3H]-naloxone binding to rat brain homogenate Opioid receptor muMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057FF6PubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-endomorphin-2 from Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J965TSPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor (unknown origin) expressed in CHO cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20G3P2RPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  6.10nMAssay Description:Displacement of [3H]DAMGO from MOR in Wistar rat brain membranes measured after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2988BVJPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  8.23nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane after 3 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9C0QPubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Vrije Universiteit Brussels

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  8.23nMAssay Description:Binding affinity to human mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23N23GCPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  8.23nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR1Z1FPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  8.23nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445M2GPubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  8.70nMAssay Description:Displacement of [3H]SP1-7 from NK1 receptor in Sprague-Dawley rat spinal cord membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542NQKPubMed
TargetSubstance-P receptor(Rattus norvegicus (rat))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  8.70nMAssay Description:Displacement of [3H]SP1-7 from NK1 receptor in Sprague-Dawley rat spinal cord membranes after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QF8WCBPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  9.5nMAssay Description:Inhibition of DAMGO (Tyr-[D-Ala]-Gly-[NMe-Phe]-Gly-ol) binding to rat brain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P601QPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  9.53nMAssay Description:Displacement of [3H]-DAMGO from Opioid receptor mu 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J965TSPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  9.56nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZS2WJXPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  9.60nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4PTKPubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  10.6nMAssay Description:Displacement of [3H]-Dynorphin A from Opioid receptor kappa 1 of rat brain membranes (DAMGO/DADLE quenching of mu/delta receptor binding)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J965TSPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Biological Research Center of the Hungarian Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-DAMGO from Wistar rat mu opioid receptor incubated for 1 hr by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F47SQMPubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£ di Chieti-Pescara G. d'Annunzio

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi: >500nMAssay Description:Displacement of [3H]U69593 from human kappa opioid receptor expressed in CHO cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP25JDPubMed
TargetOpioid receptor delta 1(Bos taurus)
Universit£ di Chieti-Pescara G. d'Annunzio

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi: >500nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in calf frontal cortex after 1 hr by gamma counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NP25JDPubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£ di Chieti-Pescara G. d'Annunzio

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  1.14E+3nMAssay Description:Displacement of [3H]U-69593 from human recombinant KOR expressed in CHO cell membranes incubated for 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2697704PubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  2.30E+3nMAssay Description:Inhibition of [3H]-naloxone binding to rat brain homogenate Opioid receptor deltaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057FF6PubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  2.65E+3nMAssay Description:Displacement of [3H]Ile5,6-deltorphin II from opioid receptor delta 1 of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J965TSPubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  2.71E+3nMAssay Description:Displacement of [3H]U69,593 from guinea pig cortex/cerebella kappa opioid receptor after 2 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B90RZPubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universit£ degli Studi di Milano

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  3.39E+3nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor (unknown origin) expressed in CHO cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20G3P2RPubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  3.94E+3nMAssay Description:Binding affinity towards delta receptor in rat brain using [3H]DSLETMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2BC408MPubMed
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute of Montreal

Curated by PDSP Ki Database
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  3.94E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23X856NPubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi: >4.00E+3nMAssay Description:Displacement of [3H]U69,593 from kappa opioid receptor in Hartley guinea pig cerebellum P2 synaptosome membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B0264PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Universit£ di Chieti-Pescara G. d'Annunzio

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  5.24E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22B931SPubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  5.65E+3nMAssay Description:Displacement of [3H]Ile5,6deltorphin-2 from delta opioid receptor in Wistar rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC038RPubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  6.08E+3nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in rat brain P2 synaptosomeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2348K1FPubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University of Catania

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  6.09E+3nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosome membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B0264PubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universit£ degli Studi di Milano

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  6.09E+3nMAssay Description:Binding affinity to delta opioid receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z96DBPubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Universit£ degli Studi di Milano

Curated by ChEMBL
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)copy SMILEScopy InChI
Affinity DataKi:  6.42E+3nMAssay Description:Displacement of [3H]DPDPE from Myc-tagged delta opioid receptor expressed in HEK293 cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T154S8PubMed
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