null
SMILES COc1ccc(Cn2c(nnc2[C@@H](Cc2ccccc2)NC(C)=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)C2=CCCCO2)cc1
InChI Key InChIKey=SFFGKVUDXGNQIY-ROJLCIKYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50165590
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier
Curated by ChEMBL
Universit£ de Montpellier
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Displacement of [125I]-His9-ghrelin from human GHS-R1a transfected in pig LLC PK-1 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier
Curated by ChEMBL
Universit£ de Montpellier
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Antagonist activity at human GHS-R1a transfected in mouse LTK cells after 6 hrs by CRE/luciferase reporter gene assay in presence of ghrelin and roli...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Universit£ de Montpellier
Curated by ChEMBL
Universit£ de Montpellier
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human GHS-R1a transfected in CHO cells assessed as inhibition of ghrelin-induced intracellular calcium mobilization measured o...More data for this Ligand-Target Pair