null
SMILES Cc1cc(NCCN2CCC(COc3ccc4c(NCCCc5ccccc5)ncnc4c3)CC2)c2ccccc2n1
InChI Key InChIKey=LSTZHFHBQKLOBB-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50239285
TargetDNA (cytosine-5)-methyltransferase 1(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388
Curated by ChEMBL
CNRS-Pierre Fabre USR3388
Curated by ChEMBL
Affinity DataEC50: 2.40E+4nMAssay Description:Inhibition of full length His-tagged human DNMT1 using SAM/[methyl-3H]SAM assessed as reduction of methylation in biotinylated hemimethylated DNA dup...More data for this Ligand-Target Pair
TargetDNA (cytosine-5)-methyltransferase 3A(Homo sapiens (Human))
CNRS-Pierre Fabre USR3388
Curated by ChEMBL
CNRS-Pierre Fabre USR3388
Curated by ChEMBL
Affinity DataEC50: 2.10E+3nMAssay Description:Inhibition of human DNMT3A catalytic domain using AdoMet assessed as reduction of methylation in 5'-biotin/3' 6-carboxyfluorescein labeled DNA duplex...More data for this Ligand-Target Pair