Compile Data Set for Download or QSAR
Found 22 Enz. Inhib. hit(s) with Target = 'Lysine-specific demethylase 7A'
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273472(CHEMBL4126235)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD-JmjC) (unknown origin) preincubated for 15 mins followed...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50395076(CHEMBL2164243)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human KDM7A catalytic domain expressed in Escherichia coli by MALDI assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3N9SPubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273469(CHEMBL4126406)copy SMILEScopy InChI
Affinity DataIC50: 5.60E+3nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD-JmjC) (unknown origin) preincubated for 15 mins followed...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273469(CHEMBL4126406)copy SMILEScopy InChI
Affinity DataIC50: 5.60E+3nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD-JmjC) (unknown origin) preincubated for 15 mins followed...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM92788(WAG-005)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD) (unknown origin) preincubated for 15 mins followed by p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM92788(WAG-005)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD-JmjC) (unknown origin) preincubated for 15 mins followed...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273477(CHEMBL4129830)copy SMILEScopy InChI
Affinity DataIC50: 6.80E+4nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD) (unknown origin) preincubated for 15 mins followed by p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273474(CHEMBL4129980)copy SMILEScopy InChI
Affinity DataIC50: 7.60E+4nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD-JmjC) (unknown origin) preincubated for 15 mins followed...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273478(CHEMBL4130224)copy SMILEScopy InChI
Affinity DataIC50: 8.60E+4nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD) (unknown origin) preincubated for 15 mins followed by p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273478(CHEMBL4130224)copy SMILEScopy InChI
Affinity DataIC50: 8.60E+4nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD-JmjC) (unknown origin) preincubated for 15 mins followed...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273476(CHEMBL4128152)copy SMILEScopy InChI
Affinity DataIC50: 9.80E+4nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD-JmjC) (unknown origin) preincubated for 15 mins followed...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273476(CHEMBL4128152)copy SMILEScopy InChI
Affinity DataIC50: 9.80E+4nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD) (unknown origin) preincubated for 15 mins followed by p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50270479(CHEMBL4127094)copy SMILEScopy InChI
Affinity DataIC50: 1.02E+5nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD) (unknown origin) preincubated for 15 mins followed by p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273473(CHEMBL4127792)copy SMILEScopy InChI
Affinity DataIC50: 1.04E+5nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD-JmjC) (unknown origin) preincubated for 15 mins followed...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273471(CHEMBL4127515)copy SMILEScopy InChI
Affinity DataIC50: 1.51E+5nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD) (unknown origin) preincubated for 15 mins followed by p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM18957((2-{4-[(2-butyl-1-benzofuran-3-yl)carbonyl]-2,6-di...)copy SMILEScopy InChI
Affinity DataIC50: 1.56E+5nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD-JmjC) (unknown origin) preincubated for 15 mins followed...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM18957((2-{4-[(2-butyl-1-benzofuran-3-yl)carbonyl]-2,6-di...)copy SMILEScopy InChI
Affinity DataIC50: 1.56E+5nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD) (unknown origin) preincubated for 15 mins followed by p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273475(CHEMBL4126951)copy SMILEScopy InChI
Affinity DataIC50: 2.95E+5nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD-JmjC) (unknown origin) preincubated for 15 mins followed...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273470(CHEMBL4128613)copy SMILEScopy InChI
Affinity DataIC50: 3.26E+5nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD) (unknown origin) preincubated for 15 mins followed by p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50273475(CHEMBL4126951)copy SMILEScopy InChI
Affinity DataIC50: 3.33E+5nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD-JmjC) (unknown origin) preincubated for 15 mins followed...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM50270475(CHEMBL4126135)copy SMILEScopy InChI
Affinity DataIC50: 5.34E+5nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD) (unknown origin) preincubated for 15 mins followed by p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University of Oxford

Curated by ChEMBL
LigandPNGBDBM92787(WAG-003)copy SMILEScopy InChI
Affinity DataIC50: 2.23E+6nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD-JmjC) (unknown origin) preincubated for 15 mins followed...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01912PubMed