Compile Data Set for Download or QSAR
Found 67 Enz. Inhib. hit(s) with Target = 'NAD kinase'
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50070942((-)-Epigallocatechin gallate | (-)-Epigallocatechi...)copy SMILEScopy InChI
Affinity DataKi:  3.28E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M049F8PubMed
TargetNAD kinase(Staphylococcus aureus)
Institut Pasteur; Institut Curie

US Patent
LigandPNGBDBM141970(US8927520, 19)copy SMILEScopy InChI
Affinity DataKi:  5.00E+3nMAssay Description:For inhibitor assays, IC50 was determined, in the presence of 1 mM NAD and 4 mM ATP (for LmNADK1) or 2 mM ATP (for SaNADK). Dixon plots were used to ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZG6QX6US Patent
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50295365(CHEMBL562056 | Di(8-bromoadenosine-5'-yl)disulfide)copy SMILEScopy InChI
Affinity DataKi:  6.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M049F8PubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50295364((8-Bromoadenosine-5'-yl)(adenosine-5'-yl)disulfide...)copy SMILEScopy InChI
Affinity DataKi:  6.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M049F8PubMed
TargetNAD kinase 1(Listeria monocytogenes)
Institut Pasteur; Institut Curie

US Patent
LigandPNGBDBM141970(US8927520, 19)copy SMILEScopy InChI
Affinity DataKi:  1.00E+4nMAssay Description:For inhibitor assays, IC50 was determined, in the presence of 1 mM NAD and 4 mM ATP (for LmNADK1) or 2 mM ATP (for SaNADK). Dixon plots were used to ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZG6QX6US Patent
TargetNAD kinase(Staphylococcus aureus)
Institut Pasteur; Institut Curie

US Patent
LigandPNGBDBM141971(US8927520, 22)copy SMILEScopy InChI
Affinity DataKi:  1.50E+4nMAssay Description:For inhibitor assays, IC50 was determined, in the presence of 1 mM NAD and 4 mM ATP (for LmNADK1) or 2 mM ATP (for SaNADK). Dixon plots were used to ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZG6QX6US Patent
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208878(CHEMBL3883415)copy SMILEScopy InChI
Affinity DataKi:  2.00E+4nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase 1(Listeria monocytogenes)
Institut Pasteur; Institut Curie

US Patent
LigandPNGBDBM141971(US8927520, 22)copy SMILEScopy InChI
Affinity DataKi:  2.00E+4nMAssay Description:For inhibitor assays, IC50 was determined, in the presence of 1 mM NAD and 4 mM ATP (for LmNADK1) or 2 mM ATP (for SaNADK). Dixon plots were used to ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZG6QX6US Patent
TargetNAD kinase 1(Listeria monocytogenes serovar 1/2a (strain ATCC B...)
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50514423(CHEMBL4552749)copy SMILEScopy InChI
Affinity DataKi:  2.50E+4nMAssay Description:Inhibition of Listeria monocytogenes NAD kinase assessed as suppression of reduced NADP formation by yeast glucose-6-phosphate dehydrogenase coupled ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ8C0RPubMed
TargetNAD kinase 1(Listeria monocytogenes)
Institut Pasteur; Institut Curie

US Patent
LigandPNGBDBM141969(US8927520, 17)copy SMILEScopy InChI
Affinity DataKi:  3.00E+4nMAssay Description:For inhibitor assays, IC50 was determined, in the presence of 1 mM NAD and 4 mM ATP (for LmNADK1) or 2 mM ATP (for SaNADK). Dixon plots were used to ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZG6QX6US Patent
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50295362((2S,3S,4R,5R,2'S,3'S,4'R,5'R)-2,2'-[DITHIOBIS(METH...)copy SMILEScopy InChI
Affinity DataKi:  4.50E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M049F8PubMed
TargetNAD kinase(Staphylococcus aureus)
Institut Pasteur; Institut Curie

US Patent
LigandPNGBDBM141969(US8927520, 17)copy SMILEScopy InChI
Affinity DataKi:  5.00E+4nMAssay Description:For inhibitor assays, IC50 was determined, in the presence of 1 mM NAD and 4 mM ATP (for LmNADK1) or 2 mM ATP (for SaNADK). Dixon plots were used to ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZG6QX6US Patent
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208780(CHEMBL3884180)copy SMILEScopy InChI
Affinity DataKi:  5.50E+4nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208778(CHEMBL3885397)copy SMILEScopy InChI
Affinity DataKi:  6.50E+4nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208739(CHEMBL3885207)copy SMILEScopy InChI
Affinity DataKi:  8.00E+4nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208802(CHEMBL3885465)copy SMILEScopy InChI
Affinity DataKi:  8.00E+4nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50203628(Benzamide adenine dinucleotide | CHEMBL233434 | be...)copy SMILEScopy InChI
Affinity DataKi:  9.00E+4nMAssay Description:Inhibition of human NAD kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X066PQPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50593321(CHEMBL5178304)copy SMILES
Affinity DataKi:  9.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M049F8PubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208741(CHEMBL3883614)copy SMILEScopy InChI
Affinity DataKi:  1.30E+5nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208736(CHEMBL3883373)copy SMILEScopy InChI
Affinity DataKi:  1.30E+5nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208740(CHEMBL3885345)copy SMILEScopy InChI
Affinity DataKi:  1.40E+5nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208745(CHEMBL3884239)copy SMILEScopy InChI
Affinity DataKi:  1.40E+5nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208805(CHEMBL3883397)copy SMILEScopy InChI
Affinity DataKi:  1.40E+5nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208904(CHEMBL3884876)copy SMILEScopy InChI
Affinity DataKi:  1.40E+5nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208743(CHEMBL3884081)copy SMILEScopy InChI
Affinity DataKi:  1.50E+5nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208779(CHEMBL3884775)copy SMILEScopy InChI
Affinity DataKi:  1.60E+5nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208737(CHEMBL3884746)copy SMILEScopy InChI
Affinity DataKi:  1.60E+5nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208795(CHEMBL3885356)copy SMILEScopy InChI
Affinity DataKi:  1.80E+5nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208735(CHEMBL3884857)copy SMILEScopy InChI
Affinity DataKi:  2.00E+5nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208774(CHEMBL3885310)copy SMILEScopy InChI
Affinity DataKi:  2.10E+5nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208874(CHEMBL3883624)copy SMILEScopy InChI
Affinity DataKi:  2.20E+5nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208781(CHEMBL3883763)copy SMILEScopy InChI
Affinity DataKi:  2.30E+5nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208773(CHEMBL3884901)copy SMILEScopy InChI
Affinity DataKi:  2.50E+5nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208775(CHEMBL3884119)copy SMILEScopy InChI
Affinity DataKi:  3.00E+5nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208742(CHEMBL3884982)copy SMILEScopy InChI
Affinity DataKi:  3.30E+5nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208734(CHEMBL3883980)copy SMILEScopy InChI
Affinity DataKi:  3.35E+5nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208744(CHEMBL3885137)copy SMILEScopy InChI
Affinity DataKi:  3.50E+5nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208738(CHEMBL3885227)copy SMILEScopy InChI
Affinity DataKi:  3.50E+5nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208776(CHEMBL3883970)copy SMILEScopy InChI
Affinity DataKi:  4.25E+5nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208777(CHEMBL3883775)copy SMILEScopy InChI
Affinity DataKi:  5.25E+5nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50208905(CHEMBL3884652)copy SMILEScopy InChI
Affinity DataKi:  7.75E+5nMAssay Description:Inhibition of human NADK expressed in Escherichia coli BL21(DE3) assessed as reduction in NADP production using NAD as substrate by glucose-6-phospha...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WH2S1KPubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50070942((-)-Epigallocatechin gallate | (-)-Epigallocatechi...)copy SMILEScopy InChI
Affinity DataIC50: 960nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M049F8PubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50295364((8-Bromoadenosine-5'-yl)(adenosine-5'-yl)disulfide...)copy SMILEScopy InChI
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human NAD kinase by modified HPLC based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T153N2PubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50295365(CHEMBL562056 | Di(8-bromoadenosine-5'-yl)disulfide)copy SMILEScopy InChI
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human NAD kinase by modified HPLC based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T153N2PubMed
TargetNAD kinase(Mycobacterium tuberculosis)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50295364((8-Bromoadenosine-5'-yl)(adenosine-5'-yl)disulfide...)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis NAD kinase by modified HPLC based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T153N2PubMed
TargetNAD kinase(Mycobacterium tuberculosis)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50295365(CHEMBL562056 | Di(8-bromoadenosine-5'-yl)disulfide)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis NAD kinase by modified HPLC based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T153N2PubMed
TargetNAD kinase(Mycobacterium tuberculosis)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50295362((2S,3S,4R,5R,2'S,3'S,4'R,5'R)-2,2'-[DITHIOBIS(METH...)copy SMILEScopy InChI
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis NAD kinase by modified HPLC based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T153N2PubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50295367(CHEMBL538665 | Di(8-Phenyladenosine-5'-yl)disulfid...)copy SMILEScopy InChI
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of human NAD kinase by modified HPLC based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T153N2PubMed
TargetNAD kinase(Mycobacterium tuberculosis)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50295363((tiazofurin-5'-yl)(adenosin-5'-yl)disulfide | CHEM...)copy SMILEScopy InChI
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis NAD kinase by modified HPLC based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T153N2PubMed
TargetNAD kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50295362((2S,3S,4R,5R,2'S,3'S,4'R,5'R)-2,2'-[DITHIOBIS(METH...)copy SMILEScopy InChI
Affinity DataIC50: 8.70E+4nMAssay Description:Inhibition of human NAD kinase by modified HPLC based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T153N2PubMed
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