Compile Data Set for Download or QSAR
Found 14 Enz. Inhib. hit(s) with Target = 'NEDD8-activating enzyme E1 regulatory subunit'
TargetNEDD8-activating enzyme E1 regulatory subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50594972(CHEMBL5177755)copy SMILES
Affinity DataIC50: 0.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21WJPubMed
TargetNEDD8-activating enzyme E1 regulatory subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50427034(CHEMBL2322194)copy SMILEScopy InChI
Affinity DataIC50: 4.70nMAssay Description:Inhibition of NAE (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32ZTPubMed
TargetNEDD8-activating enzyme E1 regulatory subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50427035(CHEMBL2017005)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of NAE (unknown origin) in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32ZTPubMed
TargetNEDD8-activating enzyme E1 regulatory subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50285607(MLN-4924 | MLN-4924003 | Pevonedistat)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:Inhibition of NAE (unknown origin)-mediated neddylation assessed as suppression of cullin1-Nedd8 adduct formation preincubated for 10 mins followed b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN99CFPubMed
TargetNEDD8-activating enzyme E1 regulatory subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50574026(CHEMBL4282603)copy SMILES
Affinity DataIC50: 260nMAssay Description:Inhibition of NAE1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2280CFCPubMed
TargetNEDD8-activating enzyme E1 regulatory subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50427031(CHEMBL2322197)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Inhibition of NAE (unknown origin)-catalyzed NEDD8-Ubcl2 intermediate formation by densitometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32ZTPubMed
TargetNEDD8-activating enzyme E1 regulatory subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50427032(6,6''-Biapigenin | CHEMBL2322196)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of NAE (unknown origin) assessed as decrease in NEDD8-Ubcl2 formationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32ZTPubMed
TargetNEDD8-activating enzyme E1 regulatory subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50562350(CHEMBL4788522)copy SMILES
Affinity DataIC50: 5.51E+3nMAssay Description:Inhibition of NAE (unknown origin)-mediated neddylation assessed as suppression of cullin1-Nedd8 adduct formation preincubated for 10 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN99CFPubMed
TargetNEDD8-activating enzyme E1 regulatory subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50562351(CHEMBL4746177)copy SMILES
Affinity DataIC50: 6.67E+3nMAssay Description:Inhibition of NAE (unknown origin)-mediated neddylation assessed as suppression of cullin1-Nedd8 adduct formation preincubated for 10 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN99CFPubMed
TargetNEDD8-activating enzyme E1 regulatory subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50562352(CHEMBL4744561)copy SMILES
Affinity DataIC50: 9.94E+3nMAssay Description:Inhibition of NAE (unknown origin)-mediated neddylation assessed as suppression of cullin1-Nedd8 adduct formation preincubated for 10 mins followed b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN99CFPubMed
TargetNEDD8-activating enzyme E1 regulatory subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50318907(2-Ethoxy-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)copy SMILEScopy InChI
Affinity DataIC50: 1.64E+4nMAssay Description:Inhibition of NAE (unknown origin)-mediated neddylation assessed as suppression of cullin1-Nedd8 adduct formation preincubated for 10 mins followed b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PN99CFPubMed
TargetNEDD8-activating enzyme E1 regulatory subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50427032(6,6''-Biapigenin | CHEMBL2322196)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of NAE (unknown origin)-catalyzed transthiolation of NEDD8 from NAE to Ubc12More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P32ZTPubMed
TargetNEDD8-activating enzyme E1 regulatory subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50537681(CHEMBL4640167)copy SMILEScopy InChI
Affinity DataEC50:  3.56E+3nMAssay Description:Inhibition of Protein kinase C delta expressed in Sf-9 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0KPRPubMed
TargetNEDD8-activating enzyme E1 regulatory subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50537681(CHEMBL4640167)copy SMILEScopy InChI
Affinity DataEC50:  3.56E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21WJPubMed