Compile Data Set for Download or QSAR
Found 73 Enz. Inhib. hit(s) with Target = 'Vasoactive intestinal polypeptide receptor 1'
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50435130(CHEMBL1893324)copy SMILEScopy InChI
Affinity DataKi:  0.0670nMAssay Description:Binding affinity to human VPAC1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NKCPubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM81828(CAS_37221-79-7 | VIP(4-28) | Vasoactive intestinal...)copy SMILEScopy InChI
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78CSRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM81828(CAS_37221-79-7 | VIP(4-28) | Vasoactive intestinal...)copy SMILEScopy InChI
Affinity DataKi:  1.60nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78CSRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM86051(CAS_0 | NSC_0 | [Lys15, Arg16, Leu27]VIP(1-7)GRF(8...)copy SMILEScopy InChI
Affinity DataKi:  1.70nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78CSRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM81828(CAS_37221-79-7 | VIP(4-28) | Vasoactive intestinal...)copy SMILEScopy InChI
Affinity DataKi:  1.70nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78CSRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM86051(CAS_0 | NSC_0 | [Lys15, Arg16, Leu27]VIP(1-7)GRF(8...)copy SMILEScopy InChI
Affinity DataKi:  7.70nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78CSRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM86051(CAS_0 | NSC_0 | [Lys15, Arg16, Leu27]VIP(1-7)GRF(8...)copy SMILEScopy InChI
Affinity DataKi:  8.90nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78CSRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM86050(Ac-L-His-L-Ser-L-Asp-L-Ala-L-Val-L-Phe-L-Thr-L-Glu...)copy SMILEScopy InChI
Affinity DataKi:  1.02E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78CSRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM86050(Ac-L-His-L-Ser-L-Asp-L-Ala-L-Val-L-Phe-L-Thr-L-Glu...)copy SMILEScopy InChI
Affinity DataKi:  1.20E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78CSRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM86694(N'-(3-Chloro-4-morpholinophenyl)-N-hydroxyform...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MW2FQQPubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50122872(4-Amino-5-chloro-2,3-dihydro-benzofuran-7-carboxyl...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9FSXPubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50250019(CHEMBL524658 | PACAP | PACAP(1-38) | PACAP-38 | PA...)copy SMILEScopy InChI
Affinity DataIC50: 0.0400nMAssay Description:Displacement of [125I]PACAP1-27 from human recombinant PAC1 receptor expressed in CHO cells measured after 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9S3SPubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50250019(CHEMBL524658 | PACAP | PACAP(1-38) | PACAP-38 | PA...)copy SMILEScopy InChI
Affinity DataIC50: 0.0500nMAssay Description:Binding affinity to human VPAC1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N87C5QPubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50435130(CHEMBL1893324)copy SMILEScopy InChI
Affinity DataIC50: 0.110nMAssay Description:Displacement of [125I]VIP from human recombinant VIP1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67JS7PubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50208990(CHEMBL3884667)copy SMILEScopy InChI
Affinity DataIC50: 0.110nMAssay Description:Displacement of [125I]VIP from human recombinant VPAC1 receptor expressed in CHO cells measured after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9S3SPubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50435130(CHEMBL1893324)copy SMILEScopy InChI
Affinity DataIC50: 0.120nMAssay Description:Binding affinity to human VPAC1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JH3NKCPubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50435130(CHEMBL1893324)copy SMILEScopy InChI
Affinity DataIC50: 0.120nMAssay Description:Binding affinity to human VPAC1 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N87C5QPubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM392076(US10301272, Example 7/9)copy SMILEScopy InChI
Affinity DataIC50: 0.470nMAssay Description:Displacement of [125I]VIP from human recombinant VPAC1 receptor after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6FPCPubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50250018(CHEMBL524852 | PACAP27)copy SMILEScopy InChI
Affinity DataIC50: 5.90nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human VPAC1 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HH6P1FPubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50498951(CHEMBL3736134)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human VPAC1 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HH6P1FPubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50498951(CHEMBL3736134)copy SMILEScopy InChI
Affinity DataIC50: 9.30nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human VPAC1 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HH6P1FPubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50498950(CHEMBL3736230)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human VPAC1 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HH6P1FPubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50498950(CHEMBL3736230)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human VPAC1 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HH6P1FPubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50200209(CHEMBL219499)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]PACAP27 from human VPAC1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD708RPubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50250074(CHEMBL507480 | [Bip6]PACAP27)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Displacement of Ac-[125I]-PACAP27 from recombinant human VPAC1 expressed in CHO cells after 90 mins by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HH6P1FPubMed
TargetVasoactive intestinal polypeptide receptor 1(Rattus norvegicus)
Bristol-Myers Squibb Co.

Curated by ChEMBL
LigandPNGBDBM50365986(CHEMBL1956427)copy SMILEScopy InChI
Affinity DataIC50: 81nMAssay Description:Antagonist activity at vasoactive intestinal peptide receptor 1 in rat RKE cells assessed as inhibition of VIP-induced intracellular cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q240QRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Rattus norvegicus)
Bristol-Myers Squibb Co.

Curated by ChEMBL
LigandPNGBDBM50365985(CHEMBL1956426)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Antagonist activity at vasoactive intestinal peptide receptor 1 in rat RKE cells assessed as inhibition of VIP-induced intracellular cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q240QRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Homo sapiens (Human))
Universit£ degli Studi di Siena

Curated by ChEMBL
LigandPNGBDBM50606528(CHEMBL5219662)copy SMILES
Affinity DataIC50: 118nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9H5MPubMed
TargetVasoactive intestinal polypeptide receptor 1(Rattus norvegicus)
Bristol-Myers Squibb Co.

Curated by ChEMBL
LigandPNGBDBM50366026(CHEMBL1956425)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Antagonist activity at vasoactive intestinal peptide receptor 1 in rat RKE cells assessed as inhibition of VIP-induced intracellular cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q240QRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Rattus norvegicus)
Bristol-Myers Squibb Co.

Curated by ChEMBL
LigandPNGBDBM50366024(CHEMBL1956413)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:Antagonist activity at vasoactive intestinal peptide receptor 1 in rat RKE cells assessed as inhibition of VIP-induced intracellular cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q240QRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Rattus norvegicus)
Bristol-Myers Squibb Co.

Curated by ChEMBL
LigandPNGBDBM50366025(CHEMBL1956424)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:Antagonist activity at vasoactive intestinal peptide receptor 1 in rat RKE cells assessed as inhibition of VIP-induced intracellular cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q240QRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Rattus norvegicus)
Bristol-Myers Squibb Co.

Curated by ChEMBL
LigandPNGBDBM50366023(CHEMBL1956412)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Antagonist activity at vasoactive intestinal peptide receptor 1 in rat RKE cells assessed as inhibition of VIP-induced intracellular cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q240QRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Rattus norvegicus)
Bristol-Myers Squibb Co.

Curated by ChEMBL
LigandPNGBDBM50366022(CHEMBL1956423)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:Antagonist activity at vasoactive intestinal peptide receptor 1 in rat RKE cells assessed as inhibition of VIP-induced intracellular cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q240QRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Rattus norvegicus)
Bristol-Myers Squibb Co.

Curated by ChEMBL
LigandPNGBDBM50366021(CHEMBL1956422)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Antagonist activity at vasoactive intestinal peptide receptor 1 in rat RKE cells assessed as inhibition of VIP-induced intracellular cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q240QRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Rattus norvegicus)
Bristol-Myers Squibb Co.

Curated by ChEMBL
LigandPNGBDBM50366020(CHEMBL1956421)copy SMILEScopy InChI
Affinity DataIC50: 290nMAssay Description:Antagonist activity at vasoactive intestinal peptide receptor 1 in rat RKE cells assessed as inhibition of VIP-induced intracellular cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q240QRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Rattus norvegicus)
Bristol-Myers Squibb Co.

Curated by ChEMBL
LigandPNGBDBM50365996(CHEMBL1956433)copy SMILEScopy InChI
Affinity DataIC50: 290nMAssay Description:Antagonist activity at vasoactive intestinal peptide receptor 1 in rat RKE cells assessed as inhibition of VIP-induced intracellular cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q240QRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Rattus norvegicus)
Bristol-Myers Squibb Co.

Curated by ChEMBL
LigandPNGBDBM50366019(CHEMBL1956420)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Antagonist activity at vasoactive intestinal peptide receptor 1 in rat RKE cells assessed as inhibition of VIP-induced intracellular cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q240QRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Rattus norvegicus)
Bristol-Myers Squibb Co.

Curated by ChEMBL
LigandPNGBDBM50366018(CHEMBL1956419)copy SMILEScopy InChI
Affinity DataIC50: 310nMAssay Description:Antagonist activity at vasoactive intestinal peptide receptor 1 in rat RKE cells assessed as inhibition of VIP-induced intracellular cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q240QRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Rattus norvegicus)
Bristol-Myers Squibb Co.

Curated by ChEMBL
LigandPNGBDBM50366017(CHEMBL1956418)copy SMILEScopy InChI
Affinity DataIC50: 390nMAssay Description:Antagonist activity at vasoactive intestinal peptide receptor 1 in rat RKE cells assessed as inhibition of VIP-induced intracellular cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q240QRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Rattus norvegicus)
Bristol-Myers Squibb Co.

Curated by ChEMBL
LigandPNGBDBM50366001(CHEMBL1956438)copy SMILEScopy InChI
Affinity DataIC50: 410nMAssay Description:Antagonist activity at vasoactive intestinal peptide receptor 1 in rat RKE cells assessed as inhibition of VIP-induced intracellular cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q240QRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Rattus norvegicus)
Bristol-Myers Squibb Co.

Curated by ChEMBL
LigandPNGBDBM50365993(CHEMBL1956432)copy SMILEScopy InChI
Affinity DataIC50: 470nMAssay Description:Antagonist activity at vasoactive intestinal peptide receptor 1 in rat RKE cells assessed as inhibition of VIP-induced intracellular cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q240QRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Rattus norvegicus)
Bristol-Myers Squibb Co.

Curated by ChEMBL
LigandPNGBDBM50365994(CHEMBL396627)copy SMILEScopy InChI
Affinity DataIC50: 470nMAssay Description:Antagonist activity at vasoactive intestinal peptide receptor 1 in rat RKE cells assessed as inhibition of VIP-induced intracellular cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q240QRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Rattus norvegicus)
Bristol-Myers Squibb Co.

Curated by ChEMBL
LigandPNGBDBM50365999(CHEMBL1956436)copy SMILEScopy InChI
Affinity DataIC50: 480nMAssay Description:Antagonist activity at vasoactive intestinal peptide receptor 1 in rat RKE cells assessed as inhibition of VIP-induced intracellular cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q240QRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Rattus norvegicus)
Bristol-Myers Squibb Co.

Curated by ChEMBL
LigandPNGBDBM50366000(CHEMBL1956437)copy SMILEScopy InChI
Affinity DataIC50: 610nMAssay Description:Antagonist activity at vasoactive intestinal peptide receptor 1 in rat RKE cells assessed as inhibition of VIP-induced intracellular cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q240QRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Rattus norvegicus)
Bristol-Myers Squibb Co.

Curated by ChEMBL
LigandPNGBDBM50366016(CHEMBL1956417)copy SMILEScopy InChI
Affinity DataIC50: 680nMAssay Description:Antagonist activity at vasoactive intestinal peptide receptor 1 in rat RKE cells assessed as inhibition of VIP-induced intracellular cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q240QRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Rattus norvegicus)
Bristol-Myers Squibb Co.

Curated by ChEMBL
LigandPNGBDBM50366015(CHEMBL1956416)copy SMILEScopy InChI
Affinity DataIC50: 740nMAssay Description:Antagonist activity at vasoactive intestinal peptide receptor 1 in rat RKE cells assessed as inhibition of VIP-induced intracellular cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q240QRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Rattus norvegicus)
Bristol-Myers Squibb Co.

Curated by ChEMBL
LigandPNGBDBM50365998(CHEMBL1956435)copy SMILEScopy InChI
Affinity DataIC50: 750nMAssay Description:Antagonist activity at vasoactive intestinal peptide receptor 1 in rat RKE cells assessed as inhibition of VIP-induced intracellular cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q240QRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Rattus norvegicus)
Bristol-Myers Squibb Co.

Curated by ChEMBL
LigandPNGBDBM50366014(CHEMBL1956415)copy SMILEScopy InChI
Affinity DataIC50: 820nMAssay Description:Antagonist activity at vasoactive intestinal peptide receptor 1 in rat RKE cells assessed as inhibition of VIP-induced intracellular cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q240QRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Rattus norvegicus)
Bristol-Myers Squibb Co.

Curated by ChEMBL
LigandPNGBDBM50366002(CHEMBL1956439)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Antagonist activity at vasoactive intestinal peptide receptor 1 in rat RKE cells assessed as inhibition of VIP-induced intracellular cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q240QRPubMed
TargetVasoactive intestinal polypeptide receptor 1(Rattus norvegicus)
Bristol-Myers Squibb Co.

Curated by ChEMBL
LigandPNGBDBM50366013(CHEMBL1956414)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Antagonist activity at vasoactive intestinal peptide receptor 1 in rat RKE cells assessed as inhibition of VIP-induced intracellular cAMP accumulatio...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q240QRPubMed
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