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3D structures from the PDB for "Tyrosine-protein kinase ABL1 [201-500,Q252H]" AND "BDBM13534"
(Proteins have >= 85% sequence identity and ligands are exact matches)


Seq IdentityJmol DisplayPDB Title
4ZOG 0%JmolVX-680/MK-0457 BINDS TO HUMAN ABL1 ALSO IN INACTIVE DFG CONFORMATIONS. No DOI
2F4J 0%JmolSTRUCTURE OF THE KINASE DOMAIN OF AN IMATINIB-RESISTANT ABL MUTANT IN COMPLEX WITH THE AURORA KINASE INHIBITOR VX-680 10.1158/0008-5472.CAN-05-2788