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3D structures from the PDB for "Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform" AND "BDBM50436459"
(Proteins have >= 85% sequence identity and ligands are exact matches)


Seq IdentityJmol DisplayPDB Title
8GUB 0%JmolCRYO-EM STRUCTURE OF CANCER-SPECIFIC PI3KALPHA MUTANT H1047R IN COMPLEX WITH BYL-719 10.1073/PNAS.2215621119
8GUA 0%JmolCRYO-EM STRUCTURE OF CANCER-SPECIFIC PI3KALPHA MUTANT E542K IN COMPLEX WITH BYL-719 10.1073/PNAS.2215621119
8GUD 0%JmolCRYO-EM STRUCTURE OF CANCER-SPECIFIC PI3KALPHA MUTANT E545K IN COMPLEX WITH BYL-719 10.1073/PNAS.2215621119
4JPS 0%JmolCO-CRYSTAL STRUCTURES OF THE LIPID KINASE PI3K ALPHA WITH PAN AND ISOFORM SELECTIVE INHIBITORS 10.1016/J.BMCL.2013.05.007
7MYO 0%JmolCRYO-EM STRUCTURE OF P110ALPHA IN COMPLEX WITH P85ALPHA INHIBITED BY BYL-719 10.1073/PNAS.2109327118
7PG6 0%JmolCRYSTAL STRUCTURE OF PI3KALPHA IN COMPLEX WITH THE INHIBITOR NVP- BYL719 No DOI