3D structures from the PDB for "Breakpoint cluster region protein/Tyrosine-protein kinase ABL1" AND "BDBM13530"
(Proteins have >= 85% sequence identity and ligands are exact matches)
| Seq Identity | Jmol Display | PDB Title |
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6NPE | 100% | | C-ABL KINASE DOMAIN WITH THE ACTIVATOR(CMPD6), 2-CYANO-N-(4-(3,4- DICHLOROPHENYL)THIAZOL-2-YL)ACETAMIDE 10.1021/ACS.JMEDCHEM.8B01872 |
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6NPV | 100% | | C-ABL KINASE DOMAIN WITH THE ACTIVATOR(CMPD51), N-(1-(3,4- DICHLOROPHENYL)-4-(2-HYDROXYETHYL)-4,5-DIHYDRO-1H-PYRAZOL-3-YL) ISONICOTINAMIDE 10.1021/ACS.JMEDCHEM.8B01872 |
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6NPU | 100% | | C-ABL KINASE DOMAIN WITH THE ACTIVATOR(CMPD29), N-(1-(3,4- DICHLOROPHENYL)-4,5-DIHYDRO-1H-PYRAZOL-3-YL)ACETAMIDE 10.1021/ACS.JMEDCHEM.8B01872 |
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2HYY | 100% | | HUMAN ABL KINASE DOMAIN IN COMPLEX WITH IMATINIB (STI571, GLIVEC) 10.1107/S0907444906047287 |
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7N9G | 100% | | CRYSTAL STRUCTURE OF THE ABL 1B KINASE DOMAIN IN COMPLEX WITH DASATINIB AND IMATINIB 10.1016/J.JMB.2021.167349 |
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3PYY | 100% | | DISCOVERY AND CHARACTERIZATION OF A CELL-PERMEABLE, SMALL-MOLECULE C- ABL KINASE ACTIVATOR THAT BINDS TO THE MYRISTOYL BINDING SITE 10.1016/J.CHEMBIOL.2010.12.013 |
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6HD6 | >99% | | ABL1 IN COMPLEX WITH COMPOUND6 AND IMATINIB (STI-571) 10.1021/ACS.JMEDCHEM.8B01040 |
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6HD4 | >99% | | ABL1 IN COMPLEX WITH COMPOUND 7 AND IMATINIB (STI-571) 10.1021/ACS.JMEDCHEM.8B01040 |
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3MS9 | >99% | | ABL KINASE IN COMPLEX WITH IMATINIB AND A FRAGMENT (FRAG1) IN THE MYRISTATE POCKET 10.1021/JA101837N |
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1IEP | >99% | | CRYSTAL STRUCTURE OF THE C-ABL KINASE DOMAIN IN COMPLEX WITH STI-571. No DOI |
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1OPJ | >99% | | STRUCTURAL BASIS FOR THE AUTO-INHIBITION OF C-ABL TYROSINE KINASE 10.1016/S0092-8674(03)00194-6 |
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3GVU | 85% | | THE CRYSTAL STRUCTURE OF HUMAN ABL2 IN COMPLEX WITH GLEEVEC No DOI |
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