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Target
Sequence
Name
&
Ki
IC50
Kd
EC50
Rate constants
ΔG°
ΔH°
-TΔS°
pH (Enzymatic Assay)
pH (ITC)
Substrate or Competitor
Compound Mol. Wt.
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Target Names &
Ki
IC50
Kd
EC50
ΔG°
ΔH°
-TΔS°
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Deposition
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rcsb
for
BDBM79403
3KWA
7QI6
7QI5
7QI4
1DNS
4FAU
2D47
6YWV
6YWS
6YWX
6YWY
6YWE
7P2E
4P5J
2B2B
7QIZ
7QIW
8AZW
1YB9
7K00
1VRO
198D
6E1X
1EI4
8AKN
8EMM
8G6X
2PL8
2PLB
7NQL
7NQH
7D5D
7D5E
7OP3
7OP1
1RFI
1RFF
4FB0
1Y8L
1Y84
2DCG
8IER
8IEN
8IEO
8IEM
4E8T
4E8Q
4E8P
4E8M
4E8N
4E8K
7FJQ
355D
1TN1
1TN2
1RGT
1RGU
1RG1
1RG2
1WOE
2RF3
1Z7I
258D
6E8S
6GAW
1EVV
6RSK
6RSJ
8OIP
8OIN
6T3R
6T3K
8AUV
4FAR
8BTK
6XXL
326D
3P4J
4R4A
6HIW
6HIV
6HIY
1ICK
2GUN
5OB3
4FAQ
4FAW
1J8G
1I2Y
8OE8
1FQ2
8ONO
3VKG
6CHR
1DPL
8OEB
8SZF
8SZH
7OAX
4R87
8OEX
1XPQ
8OEC
8OE9
7XIG
7YWZ
7YWS
6VFN
3TZO
7NE4
7NE5
7NE7
8SKW
3EUI
8P2K
324D
7EDT
1S2R
428D
7O7Z
7O7Y
1Z5T
131D
206D
6GAZ
2GWA
1PWF
1N7A
1N7B
1XPF
5VJ9
5VJB
2O3Y
7OAW
1D10
1D12
1D15
8AM9
1EDR
1RH0
5DE9
1OFX
2WLK
2WLJ
3C6M
8FV0
3BJ8
1I1P
7VPL
6S7D
3B7P
3LP9
3QJ7
2TRA
6GB2
7YX7
7N72
4MJ8
8ANY
8ANA
6YDP
8EIU
1I0T
4R0D
410D
248D
6YEC
6AF2
2F8W
1FUF
8G2N
5XJZ
7VPK
6RSL
8FV1
8B2L
8A3D
323D
1M69
1DCR
210D
6YDW
8IFB
6GDA
7OB1
4MI4
1D48
100D
7ZJZ
2B8J
5V1L
320D
211D
8SZG
321D
1F6C
8IFC
6RW5
6RW4
7N78
1XL6
7NSJ
7NSH
7NSI
6XT7
4HQI
6UEJ
2C12
4NFO
7L0Z