TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataKi: 160nMAssay Description:Competitive inhibition of CPT2More data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries S.p.A.
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries S.p.A.
Curated by ChEMBL
Affinity DataKi: 360nMAssay Description:Inhibition of rat liver carnitine palmitoyltransferase IMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataKi: 2.80E+3nMAssay Description:Competitive inhibition of CPT2 in heart mitochondria using carnitineMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataKi: 4.20E+3nMAssay Description:Competitive inhibition of CPT2 in liver mitochondria using carnitineMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of human CPT1AMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of human CPT1AMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of human CPT1AMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of human CPT1AMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of rat CPT1B expressed in intact Saccharomyces cerevisiae using [methyl-3H]carnitine by radiometric assayMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 65nMAssay Description:Inhibition of human CPT1AMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of human CPT2More data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of human CPT1AMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of human CPT2More data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of human CPT1AMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Rattus norvegicus)
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 380nMAssay Description:Inhibition of rat CPT2More data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries S.p.A.
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries S.p.A.
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries S.p.A.
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries S.p.A.
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries S.p.A.
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries S.p.A.
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of rat CPT1A expressed in intact Saccharomyces cerevisiae using [methyl-3H]carnitine by radiometric assayMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 740nMAssay Description:Inhibition of human CPT2More data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries S.p.A.
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries S.p.A.
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries S.p.A.
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries S.p.A.
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Rattus norvegicus)
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Inhibition of CPT2 in 24 hrs fasted rat liver mitochondria assessed as palmitoylcarnitine oxidation by radiometryMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of human CPT1AMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries S.p.A.
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries S.p.A.
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of CPT1A in rat myocardiumMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 1.45E+3nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries S.p.A.
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries S.p.A.
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human CPT1AMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries S.p.A.
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries S.p.A.
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries S.p.A.
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries S.p.A.
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of rat liver mitochondrial carnitine palmitoyltransferase 1 using [14C]-palmitoyl-CoA radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]-palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human CPT1AMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 2.67E+3nMAssay Description:Inhibition of human CPT1AMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of human CPT2More data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 2, mitochondrial(Rattus norvegicus)
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of rat CPT2More data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, liver isoform(Rattus norvegicus)
Sigma Tau Pharmaceutical Industries S.p.A.
Curated by ChEMBL
Sigma Tau Pharmaceutical Industries S.p.A.
Curated by ChEMBL
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I from rat liver mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 3.40E+3nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]-palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
F. Hoffmann-La Roche Ltd.
Curated by ChEMBL
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]-palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair