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Found 150 with Last Name = 'bancet' and Initial = 'a'
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))TBA
LigandPNGBDBM50162774(ABT-199 | US11420968, Example ABT-199 | Venetoclax)copy SMILEScopy InChI
Affinity DataKi: <0.0100nMAssay Description:Inhibition of BCL2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22HBPubMed
TargetCaspase-3(Homo sapiens (Human))TBA
LigandPNGBDBM50546262(CHEMBL4751195)copy SMILES
Affinity DataKi:  0.0800nMAssay Description:Inhibition of caspase-3 (unknown origin) using Ac-DEVD-AMCA as substrate incubated for 5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22HBPubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))TBA
LigandPNGBDBM50270877((R)-4-(4-((2-(4-chlorophenyl)-5,5-dimethylcyclohex...)copy SMILEScopy InChI
Affinity DataKi: <0.5nMAssay Description:Inhibition of BCL2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22HBPubMed
LigandPNGBDBM13954(3-({5-[(2S)-3-{4-[(2-carboxyphenyl)amidoformic aci...)copy SMILEScopy InChI
Affinity DataKi:  22nMAssay Description:Inhibition of PTP1B (unknown origin) using pNPP as substrate measured every 30 secs for 15 mins by Michaelis-Menten plot analysisMore data for this Ligand-Target Pair
TargetCaspase-3(Homo sapiens (Human))TBA
LigandPNGBDBM50546260(CHEMBL4782926)copy SMILES
Affinity DataKi:  25nMAssay Description:Inhibition of caspase-3 (unknown origin) using Ac-DEVD-AMCA as substrate incubated for 5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22HBPubMed
TargetCoagulation factor X(Homo sapiens (Human))TBA
LigandPNGBDBM50462575(CHEMBL4238121)copy SMILEScopy InChI
Affinity DataKi:  29nMAssay Description:Inhibition of human factor 10a using Boc-Leu-Gly-Arg-AMC as fluorogenic substrate measured after 10 mins by spectrofluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCaspase-3(Homo sapiens (Human))TBA
LigandPNGBDBM220(5-{[(4-{[(2S)-1-carboxy-3-oxopropan-2-yl]carbamoyl...)copy SMILEScopy InChI
Affinity DataKi:  200nMAssay Description:Inhibition of recombinant human caspase 3 using Ac-Asp-Glu-Val-Asp-AFC as substrate preincubated for 30 mins followed by substrate addition and measu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22HBPubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))TBA
LigandPNGBDBM50546250(CHEMBL4754689)copy SMILES
Affinity DataKi:  1.90E+3nMAssay Description:Displacement of biotin-labelled geldanamycin from human HSP90 (D9 to E236 residues) incubated for 3 hrs by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22HBPubMed
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))TBA
LigandPNGBDBM50546251(CHEMBL4783360)copy SMILES
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of human HSP90 (D9 to E236 residues) by fluorescence spectroscopyMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22HBPubMed
LigandPNGBDBM13990(5-{2-fluoro-5-[(1E)-3-[3-hydroxy-2-(methoxycarbony...)copy SMILEScopy InChI
Affinity DataKi:  7.00E+3nMAssay Description:Inhibition of PTP1B (unknown origin) using pNPP as substrate measured every 30 secs for 15 mins by Michaelis-Menten plot analysisMore data for this Ligand-Target Pair
TargetCaspase-3(Homo sapiens (Human))TBA
LigandPNGBDBM50546261(CHEMBL234378)copy SMILES
Affinity DataKi:  1.20E+5nMAssay Description:Inhibition of caspase-3 (unknown origin) using Ac-DEVD-AMCA as substrate incubated for 5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22HBPubMed
TargetCoagulation factor X(Homo sapiens (Human))TBA
LigandPNGBDBM50232690(4-Aminomethyl-Benzamidine | CHEMBL187301)copy SMILEScopy InChI
Affinity DataKi:  6.80E+5nMAssay Description:Inhibition of human factor 10a using Boc-Leu-Gly-Arg-AMC as fluorogenic substrate measured after 10 mins by spectrofluorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22HBPubMed
TargetCoagulation factor X(Homo sapiens (Human))TBA
LigandPNGBDBM50514418(CHEMBL4572188)copy SMILEScopy InChI
Affinity DataKi:  5.50E+6nMAssay Description:Inhibition of human factor 10a using Boc-Leu-Gly-Arg-AMC as fluorogenic substrate measured after 10 mins by spectrofluorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22HBPubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))TBA
LigandPNGBDBM9047(Bis-THA inhibitor 5 | CHEMBL73800 | Hexylene-Linke...)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Inhibition of rat brain Acetylcholinesterase using acetylthiocholine as substrate in presence of BChE inhibitor ethopropazineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22HBPubMed
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50520331(CHEMBL4445137)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of human NMT1 by fluorescence methodMore data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616483(US20230278983, Code AB1455)copy SMILES
Affinity DataIC50: 5.10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616482(US20230278983, Code AB1454)copy SMILES
Affinity DataIC50: 11nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetStromelysin-1(Homo sapiens (Human))TBA
LigandPNGBDBM50149219(3-(3'-Cyanomethyl-biphenyl-4-yloxy)-N-hydroxy-prop...)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of MMP3 (unknown origin) using Ac-Pro-Leu-Gly-[2-mercapto-4-methyl-pentanoyl]-Leu-Gly-OEt as substrate incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22HBPubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616454(US20230278983, Code AB1206)copy SMILES
Affinity DataIC50: 16nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616473(US20230278983, Code AB1381)copy SMILES
Affinity DataIC50: 17nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616446(US20230278983, Code AB1073)copy SMILES
Affinity DataIC50: 18nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetChitinase B(Serratia marcescens)TBA
LigandPNGBDBM50462584(CHEMBL4245260)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of Serratia marcescens chitinase BMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616474(US20230278983, Code AB1394)copy SMILES
Affinity DataIC50: 23nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616451(US20230278983, Code AB1133)copy SMILES
Affinity DataIC50: 26nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50504620(GW280670X)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of CDK2/Cyclin A (unknown origin) using histone H1 as substrate by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22HBPubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616466(US20230278983, Code AB1303)copy SMILES
Affinity DataIC50: 33nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616423(US20230278983, Code AB668)copy SMILES
Affinity DataIC50: 41nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616455(US20230278983, Code AB1208)copy SMILES
Affinity DataIC50: 45nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616481(US20230278983, Code AB1451)copy SMILES
Affinity DataIC50: 45nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616476(US20230278983, Code AB1402)copy SMILES
Affinity DataIC50: 45nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616449(US20230278983, Code AB1076)copy SMILES
Affinity DataIC50: 46nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616452(US20230278983, Code AB1135)copy SMILES
Affinity DataIC50: 48nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616463(US20230278983, Code AB1287)copy SMILES
Affinity DataIC50: 49nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616437(US20230278983, Code AB935 | isobutyl 5-fluoro-3-(1...)copy SMILES
Affinity DataIC50: 49nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616480(US20230278983, Code AB1450)copy SMILES
Affinity DataIC50: 49nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616450(US20230278983, Code AB1130)copy SMILES
Affinity DataIC50: 49nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616477(US20230278983, Code AB1415)copy SMILES
Affinity DataIC50: 50nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616436(US20230278983, Code AB934)copy SMILES
Affinity DataIC50: 52nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetEndothiapepsin(Cryphonectria parasitica)TBA
LigandPNGBDBM50546276(CHEMBL4743297)copy SMILES
Affinity DataIC50: 54nMAssay Description:Inhibition of Endothia parasitica endothiapepsin using Abz-Thr-Ile-Nle-p-nitro-Phe-Gln-Arg-NH2 as substrate by fluorescence methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22HBPubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616440(US20230278983, Code AB1030)copy SMILES
Affinity DataIC50: 54nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616432(US20230278983, Code AB929)copy SMILES
Affinity DataIC50: 58nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616435(US20230278983, Code AB933)copy SMILES
Affinity DataIC50: 62nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))TBA
LigandPNGBDBM50546256(CHEMBL4793660)copy SMILES
Affinity DataIC50: 64nMAssay Description:Inhibition of c-Src (unknown origin) using biotin-KVEKIGEGTYGVVYK as substrate by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22HBPubMed
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616444(US20230278983, Code AB1071)copy SMILES
Affinity DataIC50: 65nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616447(US20230278983, Code AB1074)copy SMILES
Affinity DataIC50: 69nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616456(US20230278983, Code AB1209)copy SMILES
Affinity DataIC50: 70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616429(US20230278983, Code AB914)copy SMILES
Affinity DataIC50: 71nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616434(US20230278983, Code AB932)copy SMILES
Affinity DataIC50: 75nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616464(US20230278983, Code AB1288)copy SMILES
Affinity DataIC50: 78nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
TargetCasein kinase II subunit alpha(Homo sapiens (Human))TBA
LigandPNGBDBM616448(US20230278983, Code AB1075)copy SMILES
Affinity DataIC50: 79nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2WH2V4R
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