Compile Data Set for Download or QSAR
Found 216 with Last Name = 'bhalerao' and Initial = 'a'
TargetCannabinoid receptor 2(Homo sapiens (Human))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402859(CHEMBL2205591)copy SMILEScopy InChI
Affinity DataKi:  81.5nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402858(CHEMBL2205592)copy SMILEScopy InChI
Affinity DataKi:  240nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402864(CHEMBL2205615)copy SMILEScopy InChI
Affinity DataKi:  241nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402863(CHEMBL2205616)copy SMILEScopy InChI
Affinity DataKi:  347nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402857(CHEMBL2205593)copy SMILEScopy InChI
Affinity DataKi:  444nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402859(CHEMBL2205591)copy SMILEScopy InChI
Affinity DataKi:  594nMAssay Description:Displacement of [3H]-CP55,940 from rat CB2 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402857(CHEMBL2205593)copy SMILEScopy InChI
Affinity DataKi:  630nMAssay Description:Displacement of [3H]-CP55,940 from rat CB2 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402860(CHEMBL2205588)copy SMILEScopy InChI
Affinity DataKi:  899nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402861(CHEMBL2205584)copy SMILEScopy InChI
Affinity DataKi:  904nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402862(CHEMBL2205620)copy SMILEScopy InChI
Affinity DataKi:  999nMAssay Description:Displacement of [3H]-CP55,940 from human CB2 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402864(CHEMBL2205615)copy SMILEScopy InChI
Affinity DataKi:  1.61E+3nMAssay Description:Displacement of [3H]-CP55,940 from rat CB2 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402861(CHEMBL2205584)copy SMILEScopy InChI
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]-CP55,940 from rat CB2 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402863(CHEMBL2205616)copy SMILEScopy InChI
Affinity DataKi:  2.13E+3nMAssay Description:Displacement of [3H]-CP55,940 from rat CB2 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402862(CHEMBL2205620)copy SMILEScopy InChI
Affinity DataKi:  2.54E+3nMAssay Description:Displacement of [3H]-CP55,940 from rat CB2 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402860(CHEMBL2205588)copy SMILEScopy InChI
Affinity DataKi:  3.11E+3nMAssay Description:Displacement of [3H]-CP55,940 from rat CB2 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402858(CHEMBL2205592)copy SMILEScopy InChI
Affinity DataKi:  4.62E+3nMAssay Description:Displacement of [3H]-CP55,940 from rat CB2 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402859(CHEMBL2205591)copy SMILEScopy InChI
Affinity DataKi:  7.19E+3nMAssay Description:Displacement of [3H]-CP55,940 from human CB1 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402857(CHEMBL2205593)copy SMILEScopy InChI
Affinity DataKi:  1.11E+4nMAssay Description:Displacement of [3H]-CP55,940 from human CB1 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402864(CHEMBL2205615)copy SMILEScopy InChI
Affinity DataKi:  1.17E+4nMAssay Description:Displacement of [3H]-CP55,940 from human CB1 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402857(CHEMBL2205593)copy SMILEScopy InChI
Affinity DataKi:  1.35E+4nMAssay Description:Displacement of [3H]-CP55,940 from rat CB1 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402864(CHEMBL2205615)copy SMILEScopy InChI
Affinity DataKi:  1.51E+4nMAssay Description:Displacement of [3H]-CP55,940 from rat CB1 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402863(CHEMBL2205616)copy SMILEScopy InChI
Affinity DataKi:  1.94E+4nMAssay Description:Displacement of [3H]-CP55,940 from human CB1 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402863(CHEMBL2205616)copy SMILEScopy InChI
Affinity DataKi:  2.26E+4nMAssay Description:Displacement of [3H]-CP55,940 from rat CB1 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402862(CHEMBL2205620)copy SMILEScopy InChI
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-CP55,940 from human CB1 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402861(CHEMBL2205584)copy SMILEScopy InChI
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-CP55,940 from human CB1 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402860(CHEMBL2205588)copy SMILEScopy InChI
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-CP55,940 from human CB1 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402858(CHEMBL2205592)copy SMILEScopy InChI
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-CP55,940 from human CB1 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402862(CHEMBL2205620)copy SMILEScopy InChI
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-CP55,940 from rat CB1 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402861(CHEMBL2205584)copy SMILEScopy InChI
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-CP55,940 from rat CB1 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402860(CHEMBL2205588)copy SMILEScopy InChI
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-CP55,940 from rat CB1 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402859(CHEMBL2205591)copy SMILEScopy InChI
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-CP55,940 from rat CB1 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Nycomed Pharma Pvt. Ltd

Curated by ChEMBL
LigandPNGBDBM50402858(CHEMBL2205592)copy SMILEScopy InChI
Affinity DataKi: >3.00E+4nMAssay Description:Displacement of [3H]-CP55,940 from rat CB1 receptor after 60 mins by microscintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4Z9VPubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Advinus Therapeutics Ltd

Curated by ChEMBL
LigandPNGBDBM202199(US9233983, P-14)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human full length BTK preincubated for 10 mins followed by Tk-biotin peptide substrate addition after 90 mins by TR-FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35X74PubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Advinus Therapeutics Ltd

Curated by ChEMBL
LigandPNGBDBM202131(US9233983, I-2)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human full length BTK preincubated for 10 mins followed by Tk-biotin peptide substrate addition after 90 mins by TR-FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35X74PubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Advinus Therapeutics Ltd

Curated by ChEMBL
LigandPNGBDBM202200(US9233983, P-15)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of recombinant human full length BTK preincubated for 10 mins followed by Tk-biotin peptide substrate addition after 90 mins by TR-FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35X74PubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Advinus Therapeutics Ltd

Curated by ChEMBL
LigandPNGBDBM50450836(CHEMBL4216939)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of recombinant human full length BTK preincubated for 10 mins followed by Tk-biotin peptide substrate addition after 90 mins by TR-FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35X74PubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Advinus Therapeutics Ltd

Curated by ChEMBL
LigandPNGBDBM202208(US9233983, P-23)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Inhibition of recombinant human full length BTK preincubated for 10 mins followed by Tk-biotin peptide substrate addition after 90 mins by TR-FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35X74PubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Advinus Therapeutics Ltd

Curated by ChEMBL
LigandPNGBDBM202122(US9233983, D-14)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Inhibition of recombinant human full length BTK preincubated for 10 mins followed by Tk-biotin peptide substrate addition after 90 mins by TR-FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35X74PubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Advinus Therapeutics Ltd

Curated by ChEMBL
LigandPNGBDBM202141(US9233983, I-12)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:Inhibition of recombinant human full length BTK preincubated for 10 mins followed by Tk-biotin peptide substrate addition after 90 mins by TR-FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35X74PubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Advinus Therapeutics Ltd

Curated by ChEMBL
LigandPNGBDBM202127(US9233983, G-1)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:Inhibition of recombinant human full length BTK preincubated for 10 mins followed by Tk-biotin peptide substrate addition after 90 mins by TR-FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35X74PubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Advinus Therapeutics Ltd

Curated by ChEMBL
LigandPNGBDBM202197(US9233983, P-12)copy SMILEScopy InChI
Affinity DataIC50: 3.10nMAssay Description:Inhibition of recombinant human full length BTK preincubated for 10 mins followed by Tk-biotin peptide substrate addition after 90 mins by TR-FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35X74PubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Advinus Therapeutics Ltd

Curated by ChEMBL
LigandPNGBDBM202128(US9233983, G-2)copy SMILEScopy InChI
Affinity DataIC50: 5.10nMAssay Description:Inhibition of recombinant human full length BTK preincubated for 10 mins followed by Tk-biotin peptide substrate addition after 90 mins by TR-FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35X74PubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Advinus Therapeutics Ltd

Curated by ChEMBL
LigandPNGBDBM202130(US9233983, I-1)copy SMILEScopy InChI
Affinity DataIC50: 5.40nMAssay Description:Inhibition of recombinant human full length BTK preincubated for 10 mins followed by Tk-biotin peptide substrate addition after 90 mins by TR-FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35X74PubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Advinus Therapeutics Ltd

Curated by ChEMBL
LigandPNGBDBM202196(US9233983, P-11)copy SMILEScopy InChI
Affinity DataIC50: 5.5nMAssay Description:Inhibition of recombinant human full length BTK preincubated for 10 mins followed by Tk-biotin peptide substrate addition after 90 mins by TR-FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35X74PubMed
TargetTyrosine-protein kinase BTK(Mus musculus)
Advinus Therapeutics Ltd

Curated by ChEMBL
LigandPNGBDBM202131(US9233983, I-2)copy SMILEScopy InChI
Affinity DataIC50: 5.5nMAssay Description:Inhibition of C57BL/6J mouse BTK assessed as decrease in anti-mouse IgM antibody stimulated BCR mediated CD69 upregulation preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35X74PubMed
TargetTyrosine-protein kinase BTK(Mus musculus)
Advinus Therapeutics Ltd

Curated by ChEMBL
LigandPNGBDBM202199(US9233983, P-14)copy SMILEScopy InChI
Affinity DataIC50: 5.80nMAssay Description:Inhibition of C57BL/6J mouse BTK assessed as decrease in anti-mouse IgM antibody stimulated BCR mediated CD69 upregulation preincubated for 30 mins f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35X74PubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Advinus Therapeutics Ltd

Curated by ChEMBL
LigandPNGBDBM202109(US9233983, D-1)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant human full length BTK preincubated for 10 mins followed by Tk-biotin peptide substrate addition after 90 mins by TR-FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35X74PubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Advinus Therapeutics Ltd

Curated by ChEMBL
LigandPNGBDBM202082(US9233983, B-1)copy SMILEScopy InChI
Affinity DataIC50: 6.5nMAssay Description:Inhibition of recombinant human full length BTK preincubated for 10 mins followed by Tk-biotin peptide substrate addition after 90 mins by TR-FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35X74PubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Advinus Therapeutics Ltd

Curated by ChEMBL
LigandPNGBDBM202087(US9233983, B-6)copy SMILEScopy InChI
Affinity DataIC50: 6.80nMAssay Description:Inhibition of recombinant human full length BTK preincubated for 10 mins followed by Tk-biotin peptide substrate addition after 90 mins by TR-FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35X74PubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Advinus Therapeutics Ltd

Curated by ChEMBL
LigandPNGBDBM202086(US9233983, B-5)copy SMILEScopy InChI
Affinity DataIC50: 8.30nMAssay Description:Inhibition of recombinant human full length BTK preincubated for 10 mins followed by Tk-biotin peptide substrate addition after 90 mins by TR-FRET as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K35X74PubMed
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