Compile Data Set for Download or QSAR
Found 127 with Last Name = 'bommi-reddy' and Initial = 'a'
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Constellation Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50542060(CHEMBL4641354 | US11274090, Example 33 Isomer 2)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Binding affinity to recombinant full length EP300 (unknown origin) incubated for 30 mins followed by H3(1 to 21) addition and measured after 1 hr by ...More data for this Ligand-Target Pair
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Constellation Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50542055(CHEMBL4636118 | US11274090, Example 22 Isomer 2)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Binding affinity to recombinant full length EP300 (unknown origin) incubated for 30 mins followed by H3(1 to 21) addition and measured after 1 hr by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Constellation Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50542046(CHEMBL4633516 | US11414384, Example 84 Isomer 2)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Binding affinity to recombinant full length EP300 (unknown origin) incubated for 30 mins followed by H3(1 to 21) addition and measured after 1 hr by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9NT5PubMed
TargetCREB-binding protein(Homo sapiens (Human))
Constellation Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50542060(CHEMBL4641354 | US11274090, Example 33 Isomer 2)copy SMILEScopy InChI
Affinity DataIC50: 2.90nMAssay Description:Binding affinity to recombinant full length CBP (unknown origin) incubated for 30 mins followed by H3(1 to 21) addition and measured after 1 hr by sc...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9NT5PubMed
TargetCREB-binding protein(Homo sapiens (Human))
Constellation Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50542046(CHEMBL4633516 | US11414384, Example 84 Isomer 2)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:Binding affinity to recombinant full length CBP (unknown origin) incubated for 30 mins followed by H3(1 to 21) addition and measured after 1 hr by sc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9NT5PubMed
TargetCREB-binding protein(Homo sapiens (Human))
Constellation Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50542055(CHEMBL4636118 | US11274090, Example 22 Isomer 2)copy SMILEScopy InChI
Affinity DataIC50: 6.70nMAssay Description:Binding affinity to recombinant full length CBP (unknown origin) incubated for 30 mins followed by H3(1 to 21) addition and measured after 1 hr by sc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9NT5PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Constellation Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50542060(CHEMBL4641354 | US11274090, Example 33 Isomer 2)copy SMILEScopy InChI
Affinity DataIC50: 8.10nMAssay Description:Binding affinity to recombinant N-terminal His-tagged EP300 HAT domain (unknown origin) (1287 to 1666 residues) expressed in Escherichia coli incubat...More data for this Ligand-Target Pair
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269687(CHEMBL4073178)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Constellation Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50542051(CHEMBL4648384 | US11414384, Example 79 Isomer 1)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Binding affinity to recombinant N-terminal His-tagged EP300 HAT domain (unknown origin) (1287 to 1666 residues) expressed in Escherichia coli incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9NT5PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Constellation Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50542055(CHEMBL4636118 | US11274090, Example 22 Isomer 2)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Binding affinity to recombinant N-terminal His-tagged EP300 HAT domain (unknown origin) (1287 to 1666 residues) expressed in Escherichia coli incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Constellation Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50542052(CHEMBL4643833 | US11274090, Example 152 Isomer 2)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Binding affinity to recombinant N-terminal His-tagged EP300 HAT domain (unknown origin) (1287 to 1666 residues) expressed in Escherichia coli incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9NT5PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Constellation Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50542047(CHEMBL4640553 | US11414384, Example 94 Isomer 2)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Binding affinity to recombinant N-terminal His-tagged EP300 HAT domain (unknown origin) (1287 to 1666 residues) expressed in Escherichia coli incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9NT5PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Constellation Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50542046(CHEMBL4633516 | US11414384, Example 84 Isomer 2)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Binding affinity to recombinant N-terminal His-tagged EP300 HAT domain (unknown origin) (1287 to 1666 residues) expressed in Escherichia coli incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9NT5PubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269689(CHEMBL4075584)copy SMILEScopy InChI
Affinity DataIC50: 44nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269688(CHEMBL4077439)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269691(CHEMBL4076944)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269690(CHEMBL4104121)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269694(CHEMBL4088221)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269697(CHEMBL4062038)copy SMILEScopy InChI
Affinity DataIC50: 55nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269693(CHEMBL4062597)copy SMILEScopy InChI
Affinity DataIC50: 59nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269696(CHEMBL4081975)copy SMILEScopy InChI
Affinity DataIC50: 71nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269698(CHEMBL4093696)copy SMILEScopy InChI
Affinity DataIC50: 83nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269695(CHEMBL4076384)copy SMILEScopy InChI
Affinity DataIC50: 93nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Constellation Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50542049(CHEMBL4639768 | US11414384, Example 100 Isomer 2)copy SMILEScopy InChI
Affinity DataIC50: 97nMAssay Description:Binding affinity to recombinant N-terminal His-tagged EP300 HAT domain (unknown origin) (1287 to 1666 residues) expressed in Escherichia coli incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9NT5PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Constellation Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50542054(CHEMBL4636245 | US11274090, Example 1 Isomer 2)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Binding affinity to recombinant N-terminal His-tagged EP300 HAT domain (unknown origin) (1287 to 1666 residues) expressed in Escherichia coli incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9NT5PubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269705(CHEMBL4102588)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged TAF1 bromodomain 2 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269699(CHEMBL4076381)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269685(CHEMBL4077529)copy SMILEScopy InChI
Affinity DataIC50: 190nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269700(CHEMBL4068293)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269701(CHEMBL4078864)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269686(CHEMBL4077036)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269704(CHEMBL4061800)copy SMILEScopy InChI
Affinity DataIC50: 330nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Constellation Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50542057(CHEMBL4639561 | US11274090, Example 56 Isomer 2)copy SMILEScopy InChI
Affinity DataIC50: 460nMAssay Description:Binding affinity to recombinant N-terminal His-tagged EP300 HAT domain (unknown origin) (1287 to 1666 residues) expressed in Escherichia coli incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9NT5PubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269703(CHEMBL4089866)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269702(CHEMBL4061901)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Constellation Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50542050(CHEMBL4636484 | US11414384, Example 93 Isomer 2)copy SMILEScopy InChI
Affinity DataIC50: 520nMAssay Description:Binding affinity to recombinant N-terminal His-tagged EP300 HAT domain (unknown origin) (1287 to 1666 residues) expressed in Escherichia coli incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9NT5PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Constellation Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50542048(CHEMBL4648100 | US11414384, Example 77)copy SMILEScopy InChI
Affinity DataIC50: 570nMAssay Description:Binding affinity to recombinant N-terminal His-tagged EP300 HAT domain (unknown origin) (1287 to 1666 residues) expressed in Escherichia coli incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9NT5PubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Constellation Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50542058(CHEMBL4642909 | US11274090, Example 57 Isomer 2)copy SMILEScopy InChI
Affinity DataIC50: 770nMAssay Description:Binding affinity to recombinant N-terminal His-tagged EP300 HAT domain (unknown origin) (1287 to 1666 residues) expressed in Escherichia coli incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9NT5PubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269706(CHEMBL4088418)copy SMILEScopy InChI
Affinity DataIC50: 780nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetChromatin remodeling regulator CECR2(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269705(CHEMBL4102588)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged CECR2 expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269687(CHEMBL4073178)copy SMILEScopy InChI
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged TAF1 bromodomain 2 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269689(CHEMBL4075584)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged BRD9 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269687(CHEMBL4073178)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged BRD9 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269690(CHEMBL4104121)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged BRD9 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269698(CHEMBL4093696)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged TAF1 bromodomain 2 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetCytochrome P450 2C8(Homo sapiens (Human))
Constellation Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50542060(CHEMBL4641354 | US11274090, Example 33 Isomer 2)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of CYP2C8 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NV9NT5PubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269686(CHEMBL4077036)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged TAF1 bromodomain 2 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269690(CHEMBL4104121)copy SMILEScopy InChI
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged TAF1 bromodomain 2 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetBromodomain-containing protein 9(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269705(CHEMBL4102588)copy SMILEScopy InChI
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged BRD9 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins by TR-FRET as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
TargetTranscription initiation factor TFIID subunit 1(Homo sapiens (Human))
Genentech Inc., 1 DNA Way, South San Francisco, California 94080, United States.

Curated by ChEMBL
LigandPNGBDBM50269691(CHEMBL4076944)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of recombinant human N-terminal His6-FLAG-tagged TAF1 bromodomain 2 (unknown origin) expressed in Rosetta2 (DE3) pLysS cells after 60 mins...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JXNPubMed
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