Compile Data Set for Download or QSAR
Found 208 with Last Name = 'cheltsov' and Initial = 'a'
TargetAndrogen receptor(Rattus norvegicus (Rat))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM82475(ACETOPHENAZINE | CAS_5714-00-1 | NSC_17676 | med.2...)copy SMILEScopy InChI
Affinity DataKi:  800nMAssay Description:Displacement of [3H]mibolerone from rat androgen receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP544FPubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM78433(2-[4-[3-[2-(trifluoromethyl)-10-phenothiazinyl]pro...)copy SMILEScopy InChI
Affinity DataKi:  800nMAssay Description:Displacement of [3H]mibolerone from rat androgen receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP544FPubMed
TargetAndrogen receptor(Rattus norvegicus (Rat))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50346422(10-(3-(4-hydroxypiperidin-1-yl)propyl)-10H-phenoth...)copy SMILEScopy InChI
Affinity DataKi:  3.00E+3nMAssay Description:Displacement of [3H]mibolerone from rat androgen receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP544FPubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447413(CHEMBL3115157)copy SMILEScopy InChI
Affinity DataKi:  3.20E+3nMAssay Description:Competitive inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells using p-nitrophenyl phosphate as subst...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7RB8PubMed
TargetAndrogen receptor(Homo sapiens (Human))
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50376214(CHEMBL263660)copy SMILEScopy InChI
Affinity DataIC50: 250nMAssay Description:Inhibition of wild type androgen receptor expressed in CV1 cells assessed as dihydrotestosterone-stimulated transactivation by CAT reporter gene assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP544FPubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM76214(CHEMBL1322977 | MLS001096094 | N-(2,5-dimethylphen...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7RB8PubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447450(CHEMBL3115119)copy SMILEScopy InChI
Affinity DataIC50: 530nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7RB8PubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447413(CHEMBL3115157)copy SMILEScopy InChI
Affinity DataIC50: 540nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7RB8PubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50316625(4-benzhydrylnaphthalene-1,2-diol | CHEMBL1094496)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence polariza...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50316625(4-benzhydrylnaphthalene-1,2-diol | CHEMBL1094496)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from 0.5 uM Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447458(CHEMBL3115158)copy SMILEScopy InChI
Affinity DataIC50: 730nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7RB8PubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50316629(1,2,3-trimethoxy-7-(3,4,5-trimethoxyphenyl)naphtha...)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from 0.5 uM Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM34138(4,5-dibenzylbenzene-1,2-diol, 9)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence polariza...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM34138(4,5-dibenzylbenzene-1,2-diol, 9)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from 0.5 uM Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50316629(1,2,3-trimethoxy-7-(3,4,5-trimethoxyphenyl)naphtha...)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence polariza...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50316627(4,4'-(1,2-phenylenebis(azan-1-yl-1-ylidene))bis(me...)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence polariza...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50316627(4,4'-(1,2-phenylenebis(azan-1-yl-1-ylidene))bis(me...)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from 0.5 uM Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50316627(4,4'-(1,2-phenylenebis(azan-1-yl-1-ylidene))bis(me...)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from 1 uM Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence pol...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50316626(2'-methoxy-1,1'-binaphthyl-2-ol | CHEMBL1094828)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence polariza...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50316626(2'-methoxy-1,1'-binaphthyl-2-ol | CHEMBL1094828)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from 0.5 uM Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447426(CHEMBL3115137)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7RB8PubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447415(CHEMBL3115148)copy SMILEScopy InChI
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7RB8PubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50316629(1,2,3-trimethoxy-7-(3,4,5-trimethoxyphenyl)naphtha...)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from 1 uM Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence pol...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50316628(CHEMBL1098663 | N-((4-methoxyphenyl)(phenyl)methyl...)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from 1 uM Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence pol...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50316628(CHEMBL1098663 | N-((4-methoxyphenyl)(phenyl)methyl...)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence polariza...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50316624(4-benzhydryl-2-methoxynaphthalen-1-ol | CHEMBL1098...)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from 0.5 uM Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM34138(4,5-dibenzylbenzene-1,2-diol, 9)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from 1 uM Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence pol...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50316624(4-benzhydryl-2-methoxynaphthalen-1-ol | CHEMBL1098...)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+3nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence polariza...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM76215(CHEMBL1349252 | MLS001096095 | N-(3-cyanophenyl)-3...)copy SMILEScopy InChI
Affinity DataIC50: 1.82E+3nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7RB8PubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50316625(4-benzhydrylnaphthalene-1,2-diol | CHEMBL1094496)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from 1 uM Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence pol...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50316624(4-benzhydryl-2-methoxynaphthalen-1-ol | CHEMBL1098...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from 1 uM Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence pol...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447425(CHEMBL3115138)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7RB8PubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447449(CHEMBL3115120)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7RB8PubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447457(CHEMBL3115159)copy SMILEScopy InChI
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7RB8PubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447448(CHEMBL3115121)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7RB8PubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50316623((N,N)-N,N'-(1,2-bis(3,4,5-trimethoxyphenyl)ethane-...)copy SMILEScopy InChI
Affinity DataIC50: 2.40E+3nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence polariza...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50316623((N,N)-N,N'-(1,2-bis(3,4,5-trimethoxyphenyl)ethane-...)copy SMILEScopy InChI
Affinity DataIC50: 2.40E+3nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from 0.5 uM Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447447(CHEMBL3115122)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7RB8PubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50316623((N,N)-N,N'-(1,2-bis(3,4,5-trimethoxyphenyl)ethane-...)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+3nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from 1 uM Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence pol...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50316626(2'-methoxy-1,1'-binaphthyl-2-ol | CHEMBL1094828)copy SMILEScopy InChI
Affinity DataIC50: 3.60E+3nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from 1 uM Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence pol...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447413(CHEMBL3115157)copy SMILEScopy InChI
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells using p-nitrophenyl phosphate as substrate after 3...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7RB8PubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447424(CHEMBL3115139)copy SMILEScopy InChI
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7RB8PubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447456(CHEMBL3115160)copy SMILEScopy InChI
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7RB8PubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM34138(4,5-dibenzylbenzene-1,2-diol, 9)copy SMILEScopy InChI
Affinity DataIC50: 4.70E+3nMAssay Description:Displacement of FITC-conjugated BH3-Bim peptide from human recombinant Bcl-2 expressed in Escherichia coli BL21 (DE3) by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50316632(2,6-dimethoxy-4-(4-methoxyphenethyl)phenol | CHEMB...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence polariza...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50316632(2,6-dimethoxy-4-(4-methoxyphenethyl)phenol | CHEMB...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from 0.5 uM Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50316631(1,2,3-trimethoxy-5-(1-(4-methoxyphenyl)ethyl)benze...)copy SMILEScopy InChI
Affinity DataIC50: 5.60E+3nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence polariza...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50316631(1,2,3-trimethoxy-5-(1-(4-methoxyphenyl)ethyl)benze...)copy SMILEScopy InChI
Affinity DataIC50: 5.60E+3nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from 0.5 uM Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
TargetIntestinal-type alkaline phosphatase(Mus musculus)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50447422(CHEMBL3115141)copy SMILEScopy InChI
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of mouse duodenal-specific FLAG-tagged IAP expressed in African green monkey COS1 cells after 30 mins by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ST7RB8PubMed
TargetVirokine/NFkB inhibitor(Vaccinia virus)
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50316631(1,2,3-trimethoxy-5-(1-(4-methoxyphenyl)ethyl)benze...)copy SMILEScopy InChI
Affinity DataIC50: 6.60E+3nMAssay Description:Displacement of FITC-conjugated BH3-Bak peptide from 1 uM Vaccinia virus recombinant N1L expressed in Escherichia coli BL21 (DE3) by fluorescence pol...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NZ87SDPubMed
Displayed 1 to 50 (of 208 total ) | Next | Last >>
Jump to: