Compile Data Set for Download or QSAR
Found 164 with Last Name = 'cronin' and Initial = 'a'
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50599238(CHEMBL5181303 | US11884671, Example 29)copy SMILES
Affinity DataIC50: 0.100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP57BCPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50599239(CHEMBL5184141 | US11884671, Example 32)copy SMILES
Affinity DataIC50: 0.100nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP57BCPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50599237(CHEMBL5180090 | US11884671, Example 30)copy SMILES
Affinity DataIC50: 0.120nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP57BCPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50599240(CHEMBL5194436 | US11884671, Example 31)copy SMILES
Affinity DataIC50: 0.130nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP57BCPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50599247(CHEMBL5197250)copy SMILES
Affinity DataIC50: 0.370nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP57BCPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50599234(CHEMBL5170489 | US11884671, Example 52)copy SMILES
Affinity DataIC50: 0.510nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP57BCPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM413450(7-methyl-2-((7-methyl-[1,2,4]triazolo[1,5-a]pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMMore data for this Ligand-Target Pair
Ligand InfoPurchaseMCE
PDB
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50599248(CHEMBL5179972)copy SMILES
Affinity DataIC50: 0.640nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP57BCPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50599243(CHEMBL5192430 | US11884671, Example 37)copy SMILES
Affinity DataIC50: 0.690nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP57BCPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50599242(CHEMBL5196848 | US11884671, Example 45)copy SMILES
Affinity DataIC50: 0.690nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP57BCPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50599245(CHEMBL5191577)copy SMILES
Affinity DataIC50: 0.75nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP57BCPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50599251(CHEMBL5198414 | US11884671, Example 42)copy SMILES
Affinity DataIC50: 1.40nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP57BCPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50599250(CHEMBL5178837)copy SMILES
Affinity DataIC50: 1.70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP57BCPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50599246(CHEMBL5204870)copy SMILES
Affinity DataIC50: 1.70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP57BCPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50599244(CHEMBL5182028 | US11884671, Example 41)copy SMILES
Affinity DataIC50: 2.60nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP57BCPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50599249(CHEMBL5182752)copy SMILES
Affinity DataIC50: 2.70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP57BCPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50599236(CHEMBL5186637 | US11884671, Example 44)copy SMILES
Affinity DataIC50: 2.90nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP57BCPubMed
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50427322(CHEMBL2325703)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of ATR-mediated CHK1 phosphorylation at serine 345 in human HT29 cells after 1 hr in presence of 4-nitroquinoline 1-oxideMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5Q5CPubMed
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50427320(CHEMBL2325705)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of ATR-mediated CHK1 phosphorylation at serine 345 in human HT29 cells after 1 hr in presence of 4-nitroquinoline 1-oxideMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5Q5CPubMed
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50427326(CHEMBL2325697)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of ATR in human HeLa cell nuclear extracts using glutathione S-transferase-p53N66 and ATP as substrate incubated for 10 mins prior to ATP ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5Q5CPubMed
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50427314(CHEMBL2325711)copy SMILEScopy InChI
Affinity DataIC50: 5nMAssay Description:Inhibition of ATR-mediated CHK1 phosphorylation at serine 345 in human HT29 cells after 1 hr in presence of 4-nitroquinoline 1-oxideMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5Q5CPubMed
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50427327(CHEMBL2325699)copy SMILEScopy InChI
Affinity DataIC50: 7nMAssay Description:Inhibition of ATR-mediated CHK1 phosphorylation at serine 345 in human HT29 cells after 1 hr in presence of 4-nitroquinoline 1-oxideMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5Q5CPubMed
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50427321(CHEMBL2325704)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of ATR-mediated CHK1 phosphorylation at serine 345 in human HT29 cells after 1 hr in presence of 4-nitroquinoline 1-oxideMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5Q5CPubMed
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50427305(CHEMBL2325720)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Inhibition of ATR in human HeLa cell nuclear extracts using glutathione S-transferase-p53N66 and ATP as substrate incubated for 10 mins prior to ATP ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5Q5CPubMed
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50427319(CHEMBL2325706)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of ATR-mediated CHK1 phosphorylation at serine 345 in human HT29 cells after 1 hr in presence of 4-nitroquinoline 1-oxideMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5Q5CPubMed
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50427317(CHEMBL2325708)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of ATR-mediated CHK1 phosphorylation at serine 345 in human HT29 cells after 1 hr in presence of 4-nitroquinoline 1-oxideMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5Q5CPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50599237(CHEMBL5180090 | US11884671, Example 30)copy SMILES
Affinity DataIC50: 13nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP57BCPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50599235(CHEMBL5171684)copy SMILES
Affinity DataIC50: 14nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP57BCPubMed
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50427297(CHEMBL2325439)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of ATR-mediated CHK1 phosphorylation at serine 345 in human HT29 cells after 1 hr in presence of 4-nitroquinoline 1-oxideMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5Q5CPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50599241(CHEMBL5198162 | US11884671, Example 43)copy SMILES
Affinity DataIC50: 15nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP57BCPubMed
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50427296(CHEMBL2325440)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of ATR-mediated CHK1 phosphorylation at serine 345 in human HT29 cells after 1 hr in presence of 4-nitroquinoline 1-oxideMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5Q5CPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50599239(CHEMBL5184141 | US11884671, Example 32)copy SMILES
Affinity DataIC50: 21nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP57BCPubMed
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50427295(CHEMBL2325695)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Inhibition of ATR in human HeLa cell nuclear extracts using glutathione S-transferase-p53N66 and ATP as substrate incubated for 10 mins prior to ATP ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5Q5CPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50599240(CHEMBL5194436 | US11884671, Example 31)copy SMILES
Affinity DataIC50: 24nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP57BCPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50599238(CHEMBL5181303 | US11884671, Example 29)copy SMILES
Affinity DataIC50: 24nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP57BCPubMed
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50427307(CHEMBL2325718)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Inhibition of ATR-mediated CHK1 phosphorylation at serine 345 in human HT29 cells after 1 hr in presence of 4-nitroquinoline 1-oxideMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5Q5CPubMed
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50384254(CHEMBL2030442)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of ATR-mediated CHK1 phosphorylation at serine 345 in human HT29 cells after 1 hr in presence of 4-nitroquinoline 1-oxideMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5Q5CPubMed
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50427313(CHEMBL2325712)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Inhibition of ATR-mediated CHK1 phosphorylation at serine 345 in human HT29 cells after 1 hr in presence of 4-nitroquinoline 1-oxideMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5Q5CPubMed
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50427316(CHEMBL2325709)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Inhibition of ATR-mediated CHK1 phosphorylation at serine 345 in human HT29 cells after 1 hr in presence of 4-nitroquinoline 1-oxideMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5Q5CPubMed
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50427329(CHEMBL2325696)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Inhibition of ATR in human HeLa cell nuclear extracts using glutathione S-transferase-p53N66 and ATP as substrate incubated for 10 mins prior to ATP ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5Q5CPubMed
TargetSerine/threonine-protein kinase mTOR(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50427326(CHEMBL2325697)copy SMILEScopy InChI
Affinity DataIC50: 38nMAssay Description:Inhibition of mTOR-mediated AKT phosphorylation at serine 473 in human MDA-MB-468 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5Q5CPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50599247(CHEMBL5197250)copy SMILES
Affinity DataIC50: 39nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP57BCPubMed
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50427298(CHEMBL2325438)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Inhibition of ATR-mediated CHK1 phosphorylation at serine 345 in human HT29 cells after 1 hr in presence of 4-nitroquinoline 1-oxideMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5Q5CPubMed
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50427315(CHEMBL2325710)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Inhibition of ATR-mediated CHK1 phosphorylation at serine 345 in human HT29 cells after 1 hr in presence of 4-nitroquinoline 1-oxideMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5Q5CPubMed
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50427326(CHEMBL2325697)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of ATR-mediated CHK1 phosphorylation at serine 345 in human HT29 cells after 1 hr in presence of 4-nitroquinoline 1-oxideMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5Q5CPubMed
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50427318(CHEMBL2325707)copy SMILEScopy InChI
Affinity DataIC50: 61nMAssay Description:Inhibition of ATR-mediated CHK1 phosphorylation at serine 345 in human HT29 cells after 1 hr in presence of 4-nitroquinoline 1-oxideMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5Q5CPubMed
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50427301(CHEMBL2325724)copy SMILEScopy InChI
Affinity DataIC50: 66nMAssay Description:Inhibition of ATR in human HeLa cell nuclear extracts using glutathione S-transferase-p53N66 and ATP as substrate incubated for 10 mins prior to ATP ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5Q5CPubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM413450(7-methyl-2-((7-methyl-[1,2,4]triazolo[1,5-a]pyridi...)copy SMILEScopy InChI
Affinity DataIC50: 92nMMore data for this Ligand-Target Pair
Ligand InfoPurchaseMCE
PDB
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))TBA
LigandPNGBDBM50599242(CHEMBL5196848 | US11884671, Example 45)copy SMILES
Affinity DataIC50: 107nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MP57BCPubMed
TargetSerine/threonine-protein kinase ATR(Homo sapiens (Human))
AstraZeneca

Curated by ChEMBL
LigandPNGBDBM50427310(CHEMBL2325715)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of ATR-mediated CHK1 phosphorylation at serine 345 in human HT29 cells after 1 hr in presence of 4-nitroquinoline 1-oxideMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5Q5CPubMed
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