Compile Data Set for Download or QSAR
Found 70 with Last Name = 'dunne' and Initial = 'a'
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173167((S)-(2-(4-fluorophenyl)-3-(2-(propylamino)pyrimidi...)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:Inhibitory activity against c-Jun N-terminal kinase 3 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8K8KPubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173169(CHEMBL383799 | [(R)-2-(4-Fluoro-phenyl)-3-(2-propy...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against c-Jun N-terminal kinase 3 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8K8KPubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173173(CHEMBL383348 | {4-[(S)-2-(4-Fluoro-phenyl)-5-(4-me...)copy SMILEScopy InChI
Affinity DataIC50: 10.9nMAssay Description:Inhibitory activity against c-Jun N-terminal kinase 3 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8K8KPubMed
TargetFibroblast growth factor 2(Homo sapiens (Human))
University College Dublin

Curated by ChEMBL
LigandPNGBDBM50000130(CHEMBL320550)copy SMILEScopy InChI
Affinity DataIC50: 25.2nMAssay Description:24% inhibition of FGF-2 binding to heparin-albumin by ELISAMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZP45G2PubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173167((S)-(2-(4-fluorophenyl)-3-(2-(propylamino)pyrimidi...)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Inhibitory activity against p38 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8K8KPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173169(CHEMBL383799 | [(R)-2-(4-Fluoro-phenyl)-3-(2-propy...)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Inhibitory activity against p38 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8K8KPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173166(CHEMBL371720 | N-{3-[4-(3-Azido-phenyl)-5-pyridin-...)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Inhibitory concentration against p38 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8K8KPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173173(CHEMBL383348 | {4-[(S)-2-(4-Fluoro-phenyl)-5-(4-me...)copy SMILEScopy InChI
Affinity DataIC50: 54nMAssay Description:Inhibitory activity against p38 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8K8KPubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173168(4-[(S)-2-(4-Fluoro-phenyl)-5-(4-methoxy-benzyloxym...)copy SMILEScopy InChI
Affinity DataIC50: 61.2nMAssay Description:Inhibitory activity against c-Jun N-terminal kinase 3 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8K8KPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415788(CHEMBL1093772)copy SMILEScopy InChI
Affinity DataIC50: 63.1nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415789(CHEMBL1093773)copy SMILEScopy InChI
Affinity DataIC50: 63.1nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415790(CHEMBL1093774 | GSK-1564023A | US10272074, Example...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173172(4-[(R)-2-(4-Fluoro-phenyl)-5-(4-methoxy-benzyloxym...)copy SMILEScopy InChI
Affinity DataIC50: 116nMAssay Description:Inhibitory activity against p38 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8K8KPubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173171(CHEMBL199247 | N-(3-(4-(4-fluorophenyl)-5-(pyridin...)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibitory concentration against c-Jun N-terminal kinase 3 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8K8KPubMed
TargetFibroblast growth factor 2(Homo sapiens (Human))
University College Dublin

Curated by ChEMBL
LigandPNGBDBM50000128(CHEMBL113091)copy SMILEScopy InChI
Affinity DataIC50: 149nMAssay Description:23% inhibition of FGF-2 binding to heparin-albumin by ELISAMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZP45G2PubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415791(CHEMBL1089404)copy SMILEScopy InChI
Affinity DataIC50: 158nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415794(CHEMBL1093602 | GSK-325971A)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415793(CHEMBL1089744)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415792(CHEMBL1089743)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173170(CHEMBL198261 | {4-[(R)-2-(4-Fluoro-phenyl)-5-(4-me...)copy SMILEScopy InChI
Affinity DataIC50: 217nMAssay Description:Inhibitory activity against p38 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8K8KPubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173170(CHEMBL198261 | {4-[(R)-2-(4-Fluoro-phenyl)-5-(4-me...)copy SMILEScopy InChI
Affinity DataIC50: 233nMAssay Description:Inhibitory activity against c-Jun N-terminal kinase 3 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8K8KPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415808(CHEMBL1091054)copy SMILEScopy InChI
Affinity DataIC50: 251nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415806(CHEMBL1094035)copy SMILEScopy InChI
Affinity DataIC50: 251nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415807(CHEMBL1090973)copy SMILEScopy InChI
Affinity DataIC50: 251nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415796(CHEMBL1089350)copy SMILEScopy InChI
Affinity DataIC50: 251nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415795(CHEMBL1089745)copy SMILEScopy InChI
Affinity DataIC50: 251nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173172(4-[(R)-2-(4-Fluoro-phenyl)-5-(4-methoxy-benzyloxym...)copy SMILEScopy InChI
Affinity DataIC50: 270nMAssay Description:Inhibitory activity against c-Jun N-terminal kinase 3 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8K8KPubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173168(4-[(S)-2-(4-Fluoro-phenyl)-5-(4-methoxy-benzyloxym...)copy SMILEScopy InChI
Affinity DataIC50: 295nMAssay Description:Inhibitory activity against p38 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28G8K8KPubMed
TargetFibroblast growth factor 2(Homo sapiens (Human))
University College Dublin

Curated by ChEMBL
LigandPNGBDBM50421574(CHEMBL2303729)copy SMILEScopy InChI
Affinity DataIC50: 313nMAssay Description:25% inhibition of FGF-2 binding to heparin-albumin by ELISAMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZP45G2PubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415809(CHEMBL1091439)copy SMILEScopy InChI
Affinity DataIC50: 316nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415810(CHEMBL1091440 | US10272074, Example 30)copy SMILEScopy InChI
Affinity DataIC50: 316nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetFibroblast growth factor 2(Homo sapiens (Human))
University College Dublin

Curated by ChEMBL
LigandPNGBDBM50421574(CHEMBL2303729)copy SMILEScopy InChI
Affinity DataIC50: 340nMAssay Description:25% inhibition of FGF-2 binding to heparin-albumin by ELISAMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2ZP45G2PubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415798(CHEMBL1089600)copy SMILEScopy InChI
Affinity DataIC50: 398nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415797(CHEMBL1089692)copy SMILEScopy InChI
Affinity DataIC50: 398nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415811(CHEMBL1093055)copy SMILEScopy InChI
Affinity DataIC50: 501nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415812(CHEMBL1091066)copy SMILEScopy InChI
Affinity DataIC50: 794nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415799(CHEMBL1093352)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetProgesterone receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415794(CHEMBL1093602 | GSK-325971A)copy SMILEScopy InChI
Affinity DataIC50: 1.26E+3nMAssay Description:Antagonist activity at human progesterone receptor B expressed in african green monkey CV1 cells assessed as inhibition of progesterone-induced effec...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415790(CHEMBL1093774 | GSK-1564023A | US10272074, Example...)copy SMILEScopy InChI
Affinity DataIC50: 2.51E+3nMAssay Description:Inhibition of human PDE4B by ATP-luciferace luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetProgesterone receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415790(CHEMBL1093774 | GSK-1564023A | US10272074, Example...)copy SMILEScopy InChI
Affinity DataIC50: 3.16E+3nMAssay Description:Antagonist activity at human progesterone receptor B expressed in african green monkey CV1 cells assessed as inhibition of progesterone-induced effec...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415794(CHEMBL1093602 | GSK-325971A)copy SMILEScopy InChI
Affinity DataIC50: 3.98E+3nMAssay Description:Inhibition of human PDE4B by ATP-luciferace luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetProgesterone receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415792(CHEMBL1089743)copy SMILEScopy InChI
Affinity DataIC50: 5.01E+3nMAssay Description:Antagonist activity at human progesterone receptor B expressed in african green monkey CV1 cells assessed as inhibition of progesterone-induced effec...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415814(CHEMBL1094032)copy SMILEScopy InChI
Affinity DataIC50: 6.31E+3nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415800(CHEMBL1093353)copy SMILEScopy InChI
Affinity DataIC50: 6.31E+3nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415801(CHEMBL1093354)copy SMILEScopy InChI
Affinity DataIC50: 6.31E+3nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415802(CHEMBL1089707)copy SMILEScopy InChI
Affinity DataIC50: 6.31E+3nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415803(CHEMBL1094031)copy SMILEScopy InChI
Affinity DataIC50: 6.31E+3nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415804(CHEMBL1094033)copy SMILEScopy InChI
Affinity DataIC50: 6.31E+3nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415805(CHEMBL1094034)copy SMILEScopy InChI
Affinity DataIC50: 6.31E+3nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Medicines Research Centre

Curated by ChEMBL
LigandPNGBDBM50415813(CHEMBL1091320)copy SMILEScopy InChI
Affinity DataIC50: 6.31E+3nMAssay Description:Antagonist activity at glucocorticoid receptor expressed in human A549 cells assessed as inhibition of cortisol-induced renilla luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2XDJPubMed
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