Compile Data Set for Download or QSAR
Found 251 with Last Name = 'fedolak' and Initial = 'a'
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50049750((S)-3-(azetidin-2-ylmethoxy)pyridine | 3-((S)-1-Az...)copy SMILEScopy InChI
Affinity DataKi:  0.0400nMAssay Description:Binding affinity to alpha4beta2 nAChR in human brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CJ8FM1PubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-2(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50210335(CHEMBL3898434)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-2(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50210334(CHEMBL3948977)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-2(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50216347((1R,4R)-2-(3-pyridinyl)-2,5-diazabicyclo[2.2.1]hep...)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50166908(5,8,14-triazatetracyclo[10.3.1.02,11.04,9]hexadeca...)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Binding affinity to alpha4beta2 nAChRMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50210335(CHEMBL3898434)copy SMILEScopy InChI
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50210334(CHEMBL3948977)copy SMILEScopy InChI
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50210337(CHEMBL3970672)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-2(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50210337(CHEMBL3970672)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50216347((1R,4R)-2-(3-pyridinyl)-2,5-diazabicyclo[2.2.1]hep...)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-2(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50088438(1-(pyridin-3-yl)-1,4-diazepane | 1-Pyridin-3-yl-[1...)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50216347((1R,4R)-2-(3-pyridinyl)-2,5-diazabicyclo[2.2.1]hep...)copy SMILEScopy InChI
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-2(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50210338(CHEMBL3926480)copy SMILEScopy InChI
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50088438(1-(pyridin-3-yl)-1,4-diazepane | 1-Pyridin-3-yl-[1...)copy SMILEScopy InChI
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)copy SMILEScopy InChI
Affinity DataKi:  4.90nMAssay Description:Binding affinity to alpha4beta2 nAChR by PDSP assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50088438(1-(pyridin-3-yl)-1,4-diazepane | 1-Pyridin-3-yl-[1...)copy SMILEScopy InChI
Affinity DataKi:  5.10nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)copy SMILEScopy InChI
Affinity DataKi:  5.5nMAssay Description:Binding affinity to alpha2beta2 nAChR by PDSP assayMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50210338(CHEMBL3926480)copy SMILEScopy InChI
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50216347((1R,4R)-2-(3-pyridinyl)-2,5-diazabicyclo[2.2.1]hep...)copy SMILEScopy InChI
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta4 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetAcetylcholine-binding protein(Great pond snail)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50382466(CHEMBL2024087)copy SMILEScopy InChI
Affinity DataKi:  12.8nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis AChBPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62BWPubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-4(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50216347((1R,4R)-2-(3-pyridinyl)-2,5-diazabicyclo[2.2.1]hep...)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta4 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50210335(CHEMBL3898434)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50210334(CHEMBL3948977)copy SMILEScopy InChI
Affinity DataKi:  17nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-2(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50210332(CHEMBL3889475)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetAcetylcholine-binding protein(Great pond snail)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50382467(CHEMBL2024089)copy SMILEScopy InChI
Affinity DataKi:  22nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis AChBPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62BWPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50210332(CHEMBL3889475)copy SMILEScopy InChI
Affinity DataKi:  25nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50210336(CHEMBL3899499)copy SMILEScopy InChI
Affinity DataKi:  36nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50210337(CHEMBL3970672)copy SMILEScopy InChI
Affinity DataKi:  42nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-2(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50210336(CHEMBL3899499)copy SMILEScopy InChI
Affinity DataKi:  43nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-2(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50210333(CHEMBL3908556)copy SMILEScopy InChI
Affinity DataKi:  46nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50210333(CHEMBL3908556)copy SMILEScopy InChI
Affinity DataKi:  51nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-4(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50088438(1-(pyridin-3-yl)-1,4-diazepane | 1-Pyridin-3-yl-[1...)copy SMILEScopy InChI
Affinity DataKi:  62nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta4 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50216347((1R,4R)-2-(3-pyridinyl)-2,5-diazabicyclo[2.2.1]hep...)copy SMILEScopy InChI
Affinity DataKi:  65nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50210337(CHEMBL3970672)copy SMILEScopy InChI
Affinity DataKi:  68nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta4 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50088438(1-(pyridin-3-yl)-1,4-diazepane | 1-Pyridin-3-yl-[1...)copy SMILEScopy InChI
Affinity DataKi:  72nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta4 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50166908(5,8,14-triazatetracyclo[10.3.1.02,11.04,9]hexadeca...)copy SMILEScopy InChI
Affinity DataKi:  125nMAssay Description:Binding affinity to rat alpha7 nACHR at 10 uMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7JS7PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50210338(CHEMBL3926480)copy SMILEScopy InChI
Affinity DataKi:  141nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50049750((S)-3-(azetidin-2-ylmethoxy)pyridine | 3-((S)-1-Az...)copy SMILEScopy InChI
Affinity DataKi:  148nMAssay Description:Binding affinity to human alpha7 nAChR in human brainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CJ8FM1PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50210334(CHEMBL3948977)copy SMILEScopy InChI
Affinity DataKi:  151nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta4 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-4(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50210335(CHEMBL3898434)copy SMILEScopy InChI
Affinity DataKi:  168nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta4 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-4(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50210335(CHEMBL3898434)copy SMILEScopy InChI
Affinity DataKi:  256nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta4 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-4(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50210337(CHEMBL3970672)copy SMILEScopy InChI
Affinity DataKi:  331nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta4 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50088438(1-(pyridin-3-yl)-1,4-diazepane | 1-Pyridin-3-yl-[1...)copy SMILEScopy InChI
Affinity DataKi:  366nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-2/beta-4(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50210334(CHEMBL3948977)copy SMILEScopy InChI
Affinity DataKi:  460nMAssay Description:Displacement of [3H]epibatidine from rat alpha2beta4 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetAcetylcholine-binding protein(Great pond snail)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)copy SMILEScopy InChI
Affinity DataKi:  496nMAssay Description:Displacement of [3H]epibatidine from Lymnaea stagnalis AChBPMore data for this Ligand-Target Pair
TargetSoluble acetylcholine receptor(California sea hare)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)copy SMILEScopy InChI
Affinity DataKi:  598nMAssay Description:Displacement of [3H]epibatidine from Aplysia californica AChBPMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50210336(CHEMBL3899499)copy SMILEScopy InChI
Affinity DataKi:  617nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50210332(CHEMBL3889475)copy SMILEScopy InChI
Affinity DataKi:  681nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
TargetSoluble acetylcholine receptor(California sea hare)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50382466(CHEMBL2024087)copy SMILEScopy InChI
Affinity DataKi:  979nMAssay Description:Displacement of [3H]epibatidine from Aplysia californica AChBPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC62BWPubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-2(Rat)
University of Illinois at Chicago

Curated by ChEMBL
LigandPNGBDBM50210333(CHEMBL3908556)copy SMILEScopy InChI
Affinity DataKi:  1.04E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta2 nAChR by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41TDBPubMed
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