Compile Data Set for Download or QSAR
Found 928 with Last Name = 'hammed' and Initial = 'a'
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50138119(CHEMBL3753475)copy SMILEScopy InChI
Affinity DataKi:  0.0300nMAssay Description:Binding affinity to recombinant human H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F191KFPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Suven Life Sciences Ltd.

Curated by ChEMBL
LigandPNGBDBM221048(US9284322, varenicline | US9303017, Varenicline)copy SMILEScopy InChI
Affinity DataKi:  0.0400nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50138124(CHEMBL3753901)copy SMILEScopy InChI
Affinity DataKi:  0.100nMAssay Description:Binding affinity to recombinant human H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F191KFPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Suven Life Sciences Ltd.

Curated by ChEMBL
LigandPNGBDBM50538045(CHEMBL4636163)copy SMILEScopy InChI
Affinity DataKi:  0.140nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29027BJPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Suven Life Sciences Ltd.

Curated by ChEMBL
LigandPNGBDBM50538008(CHEMBL4638732)copy SMILEScopy InChI
Affinity DataKi:  0.190nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29027BJPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Suven Life Sciences Ltd.

Curated by ChEMBL
LigandPNGBDBM50538046(CHEMBL4647198)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29027BJPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Suven Life Sciences Ltd.

Curated by ChEMBL
LigandPNGBDBM50538047(CHEMBL4647019)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29027BJPubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50318633(3-benzenesulfonyl-8-piperazin-1-ylquinoline | CHEM...)copy SMILEScopy InChI
Affinity DataKi:  0.230nMAssay Description:Inhibitory concentration against Herpes simplex virus type 1 thymidine kinase(HSV-1 TK)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7R1XPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50483134(CHEBI:64156 | Imetit)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of [3]-RAMH from recombinant human histamine H3 receptor expressed in CHO-K1 cell membranes after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD152GPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Suven Life Sciences Ltd.

Curated by ChEMBL
LigandPNGBDBM50538027(CHEMBL4644169)copy SMILEScopy InChI
Affinity DataKi:  0.370nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29027BJPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50138119(CHEMBL3753475)copy SMILEScopy InChI
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F191KFPubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50019754(IDALOPIRDINE | LU-AE58054)copy SMILEScopy InChI
Affinity DataKi:  0.830nMAssay Description:Antagonist activity at 5-HT6 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7R1XPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50138120(CHEMBL3753093)copy SMILEScopy InChI
Affinity DataKi:  0.900nMAssay Description:Binding affinity to recombinant human H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F191KFPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50517508(CHEMBL4594107)copy SMILEScopy InChI
Affinity DataKi:  0.960nMAssay Description:Displacement of [3]-RAMH from recombinant human histamine H3 receptor expressed in CHO-K1 cell membranes after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD152GPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50138122(CHEMBL3752655)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Binding affinity to recombinant human H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F191KFPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50138123(CHEMBL3753703)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F191KFPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Suven Life Sciences Ltd.

Curated by ChEMBL
LigandPNGBDBM50538033(CHEMBL4648557)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29027BJPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50517531(CHEMBL4445638)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Displacement of [3]-RAMH from recombinant human histamine H3 receptor expressed in CHO-K1 cell membranes after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD152GPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Suven Life Sciences Ltd.

Curated by ChEMBL
LigandPNGBDBM50538030(CHEMBL4638919)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29027BJPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50517534(CHEMBL4476066)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Displacement of [3]-RAMH from recombinant human histamine H3 receptor expressed in CHO-K1 cell membranes after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD152GPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50138123(CHEMBL3753703)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Binding affinity to recombinant human H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F191KFPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50138117(CHEMBL3753315)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F191KFPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Suven Life Sciences Ltd.

Curated by ChEMBL
LigandPNGBDBM50538038(CHEMBL4648098)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29027BJPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50517529(CHEMBL4587541)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Displacement of [3]-RAMH from recombinant human histamine H3 receptor expressed in CHO-K1 cell membranes after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD152GPubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50236846(CHEMBL4080401)copy SMILEScopy InChI
Affinity DataKi:  1.30nMAssay Description:Inhibition of recombinant mammalian Geranylgeranyl transferase type I expressed in baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7R1XPubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50044616(Cerlapirdine | PF-05212365 | SAM-531 | WAY-262531)copy SMILEScopy InChI
Affinity DataKi:  1.30nMAssay Description:Effective concentration required for agonistic activity at Metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7R1XPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Suven Life Sciences Ltd.

Curated by ChEMBL
LigandPNGBDBM50538036(CHEMBL4634253)copy SMILEScopy InChI
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29027BJPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Suven Life Sciences Ltd.

Curated by ChEMBL
LigandPNGBDBM50538063(CHEMBL4642118)copy SMILEScopy InChI
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29027BJPubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50236844(CHEMBL4100484)copy SMILEScopy InChI
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7R1XPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50517507(CHEMBL4456037)copy SMILEScopy InChI
Affinity DataKi:  1.60nMAssay Description:Displacement of [3]-RAMH from recombinant human histamine H3 receptor expressed in CHO-K1 cell membranes after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD152GPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50138106(CHEMBL3753814)copy SMILEScopy InChI
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F191KFPubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50236780(CHEMBL4068232)copy SMILEScopy InChI
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7R1XPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50138118(CHEMBL3754200)copy SMILEScopy InChI
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F191KFPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50517523(CHEMBL4518550)copy SMILEScopy InChI
Affinity DataKi:  1.90nMAssay Description:Displacement of [3]-RAMH from recombinant human histamine H3 receptor expressed in CHO-K1 cell membranes after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD152GPubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50236754(CHEMBL4082473)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Effective concentration required for partial agonistic activity at Metabotropic glutamate receptor 2; Partial agonistMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7R1XPubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50236756(CHEMBL4101284)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7R1XPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50138124(CHEMBL3753901)copy SMILEScopy InChI
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F191KFPubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50236773(CHEMBL4065437)copy SMILEScopy InChI
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7R1XPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Suven Life Sciences Ltd.

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)copy SMILEScopy InChI
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50517505(CHEMBL4521909)copy SMILEScopy InChI
Affinity DataKi:  2.40nMAssay Description:Displacement of [3]-RAMH from recombinant human histamine H3 receptor expressed in CHO-K1 cell membranes after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD152GPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50517521(CHEMBL4574463)copy SMILEScopy InChI
Affinity DataKi:  2.40nMAssay Description:Displacement of [3]-RAMH from recombinant human histamine H3 receptor expressed in CHO-K1 cell membranes after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD152GPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50138104(CHEMBL3754209)copy SMILEScopy InChI
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]R-alpha-methyl histamine from recombinant human H3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F191KFPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50517522(CHEMBL4534815)copy SMILEScopy InChI
Affinity DataKi:  2.60nMAssay Description:Displacement of [3]-RAMH from recombinant human histamine H3 receptor expressed in CHO-K1 cell membranes after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD152GPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50517502(CHEMBL4439392)copy SMILEScopy InChI
Affinity DataKi:  2.60nMAssay Description:Displacement of [3]-RAMH from recombinant human histamine H3 receptor expressed in CHO-K1 cell membranes after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD152GPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Suven Life Sciences Ltd.

Curated by ChEMBL
LigandPNGBDBM50538014(CHEMBL4637076)copy SMILEScopy InChI
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29027BJPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50517540(CHEMBL4452215)copy SMILEScopy InChI
Affinity DataKi:  2.80nMAssay Description:Displacement of [3]-RAMH from recombinant human histamine H3 receptor expressed in CHO-K1 cell membranes after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD152GPubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50517527(CHEMBL4576724)copy SMILEScopy InChI
Affinity DataKi:  2.90nMAssay Description:Displacement of [3]-RAMH from recombinant human histamine H3 receptor expressed in CHO-K1 cell membranes after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD152GPubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
Suven Life Sciences Ltd.

Curated by ChEMBL
LigandPNGBDBM50538035(CHEMBL4634110)copy SMILEScopy InChI
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in CHOK1 cell membrane by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29027BJPubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University of Heidelberg

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)copy SMILEScopy InChI
Affinity DataKi:  2.95nMAssay Description:Binding affinity was measured on Sigma receptor type 1 with guinea pig membranes and [3H]- pentazocine as ligand.More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Suven Life Sciences Ltd

Curated by ChEMBL
LigandPNGBDBM50517491(CHEMBL4468778)copy SMILEScopy InChI
Affinity DataKi:  3.20nMAssay Description:Displacement of [3]-RAMH from recombinant human histamine H3 receptor expressed in CHO-K1 cell membranes after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD152GPubMed
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