Affinity DataKi: 0.300nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
TargetD(3) dopamine receptor(Homo sapiens (Human))
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 14.7nMAssay Description:Inhibition constant against human intestinal carboxylesterase (hiCE) expressed in Sf21 cells using 3 mM o-NPAMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
TargetLiver carboxylesterase 1(Homo sapiens (Human))
St. Jude Children's Research Hospital
Curated by ChEMBL
St. Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition constant against human liver carboxylesterase (hCE1) expressed in Sf21 cells using 3 mM o-NPAMore data for this Ligand-Target Pair
TargetLiver carboxylesterase 1(Homo sapiens (Human))
St. Jude Children's Research Hospital
Curated by ChEMBL
St. Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition constant against human liver carboxylesterase (hCE1) expressed in Sf21 cells using 3 mM o-NPAMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 40nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
TargetLiver carboxylesterase 1(Homo sapiens (Human))
St. Jude Children's Research Hospital
Curated by ChEMBL
St. Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataKi: 45.1nMAssay Description:Inhibition constant against human liver carboxylesterase (hCE1) expressed in Sf21 cells using 3 mM o-NPAMore data for this Ligand-Target Pair
TargetLiver carboxylesterase 1(Homo sapiens (Human))
St. Jude Children's Research Hospital
Curated by ChEMBL
St. Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataKi: 45.1nMAssay Description:Inhibition constant against human liver carboxylesterase (hCE1) expressed in Sf21 cells using 3 mM o-NPAMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 75nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 85nMAssay Description:Inhibition constant against human intestinal carboxylesterase (hiCE) expressed in Sf21 cells using 3 mM o-NPAMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
TargetLiver carboxylesterase 1(Homo sapiens (Human))
St. Jude Children's Research Hospital
Curated by ChEMBL
St. Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataKi: 126nMAssay Description:Inhibition constant against human liver carboxylesterase (hCE1) expressed in Sf21 cells using 3 mM o-NPAMore data for this Ligand-Target Pair
TargetLiver carboxylesterase 1(Homo sapiens (Human))
St. Jude Children's Research Hospital
Curated by ChEMBL
St. Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataKi: 126nMAssay Description:Inhibition constant against human liver carboxylesterase (hCE1) expressed in Sf21 cells using 3 mM o-NPAMore data for this Ligand-Target Pair
Affinity DataKi: 146nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 152nMAssay Description:Inhibition constant against human intestinal carboxylesterase (hiCE) expressed in Sf21 cells using 3 mM o-NPAMore data for this Ligand-Target Pair
TargetLiver carboxylesterase 1(Homo sapiens (Human))
St. Jude Children's Research Hospital
Curated by ChEMBL
St. Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataKi: 210nMAssay Description:Inhibition constant against human liver carboxylesterase (hCE1) expressed in Sf21 cells using 3 mM o-NPAMore data for this Ligand-Target Pair
TargetLiver carboxylesterase 1(Homo sapiens (Human))
St. Jude Children's Research Hospital
Curated by ChEMBL
St. Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataKi: 210nMAssay Description:Inhibition constant against human liver carboxylesterase (hCE1) expressed in Sf21 cells using 3 mM o-NPAMore data for this Ligand-Target Pair
TargetLiver carboxylesterase 1(Homo sapiens (Human))
St. Jude Children's Research Hospital
Curated by ChEMBL
St. Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataKi: 212nMAssay Description:Inhibition constant against human liver carboxylesterase (hCE1) expressed in Sf21 cells using 3 mM o-NPAMore data for this Ligand-Target Pair
TargetLiver carboxylesterase 1(Homo sapiens (Human))
St. Jude Children's Research Hospital
Curated by ChEMBL
St. Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataKi: 212nMAssay Description:Inhibition constant against human liver carboxylesterase (hCE1) expressed in Sf21 cells using 3 mM o-NPAMore data for this Ligand-Target Pair
Affinity DataKi: 237nMAssay Description:Inhibition constant against human intestinal carboxylesterase (hiCE) expressed in Sf21 cells using 3 mM o-NPAMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 4(PIGLET)
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
TargetLiver carboxylesterase 1(Homo sapiens (Human))
St. Jude Children's Research Hospital
Curated by ChEMBL
St. Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataKi: 255nMAssay Description:Inhibition constant against human liver carboxylesterase (hCE1) expressed in Sf21 cells using 3 mM o-NPAMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1F(Homo sapiens (Human))
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
TargetLiver carboxylesterase 1(Homo sapiens (Human))
St. Jude Children's Research Hospital
Curated by ChEMBL
St. Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataKi: 365nMAssay Description:Inhibition constant against human liver carboxylesterase (hCE1) expressed in Sf21 cells using 3 mM o-NPAMore data for this Ligand-Target Pair
TargetLiver carboxylesterase 1(Homo sapiens (Human))
St. Jude Children's Research Hospital
Curated by ChEMBL
St. Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataKi: 365nMAssay Description:Inhibition constant against human liver carboxylesterase (hCE1) expressed in Sf21 cells using 3 mM o-NPAMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 430nMAssay Description:Displacement of [3H]nisoxetine from recombinant human Dopamine transporter after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 573nMAssay Description:Inhibition constant against human intestinal carboxylesterase (hiCE) expressed in Sf21 cells using 3 mM o-NPAMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
Affinity DataKi: 1.04E+3nMAssay Description:Inhibition constant against human intestinal carboxylesterase (hiCE) expressed in Sf21 cells using 3 mM o-NPAMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
TargetLiver carboxylesterase 1(Homo sapiens (Human))
St. Jude Children's Research Hospital
Curated by ChEMBL
St. Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataKi: 1.17E+3nMAssay Description:Inhibition constant against human liver carboxylesterase (hCE1) expressed in Sf21 cells using 3 mM o-NPAMore data for this Ligand-Target Pair
TargetLiver carboxylesterase 1(Homo sapiens (Human))
St. Jude Children's Research Hospital
Curated by ChEMBL
St. Jude Children's Research Hospital
Curated by ChEMBL
Affinity DataKi: 1.17E+3nMAssay Description:Inhibition constant against human liver carboxylesterase (hCE1) expressed in Sf21 cells using 3 mM o-NPAMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database
SmithKline Beecham Pharmaceuticals
Curated by PDSP Ki Database