Compile Data Set for Download or QSAR
Found 192 with Last Name = 'limatola' and Initial = 'a'
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples"Federico II"

Curated by ChEMBL
LigandPNGBDBM50048691(CHEMBL3315139)copy SMILES
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples"Federico II"

Curated by ChEMBL
LigandPNGBDBM50320463(CHEMBL218994 | D[CFWKYC]V | H-Asp-Cys-Phe-Trp-Lys-...)copy SMILEScopy InChI
Affinity DataKi:  0.251nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples"Federico II"

Curated by ChEMBL
LigandPNGBDBM50048696(CHEMBL3315142)copy SMILES
Affinity DataKi:  0.398nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples"Federico II"

Curated by ChEMBL
LigandPNGBDBM50048695(CHEMBL3315141)copy SMILES
Affinity DataKi:  0.724nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples"Federico II"

Curated by ChEMBL
LigandPNGBDBM50048701(CHEMBL3315148)copy SMILES
Affinity DataKi:  0.776nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples"Federico II"

Curated by ChEMBL
LigandPNGBDBM50413784(UROTENSIN-II)copy SMILEScopy InChI
Affinity DataKi:  0.794nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universit£ di Chieti-Pescara"G. d'Annunzio"

Curated by ChEMBL
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain membranes by liquid scintillation counting based competition binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9JS5PubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples"Federico II"

Curated by ChEMBL
LigandPNGBDBM50048700(CHEMBL3315147)copy SMILES
Affinity DataKi:  1nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples"Federico II"

Curated by ChEMBL
LigandPNGBDBM50048699(CHEMBL3315146)copy SMILES
Affinity DataKi:  1.20nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples"Federico II"

Curated by ChEMBL
LigandPNGBDBM50048697(CHEMBL3315144)copy SMILES
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Universit£ di Chieti-Pescara"G. d'Annunzio"

Curated by ChEMBL
LigandPNGBDBM50026764(CHEMBL3331509)copy SMILEScopy InChI
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]Ile5,6deltorphin II from delta opioid receptor in Wistar rat brain membranes by liquid scintillation counting based competition b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9JS5PubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples"Federico II"

Curated by ChEMBL
LigandPNGBDBM50048705(CHEMBL3315152)copy SMILES
Affinity DataKi:  1.80nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples"Federico II"

Curated by ChEMBL
LigandPNGBDBM50048703(CHEMBL3315150)copy SMILES
Affinity DataKi:  1.80nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universit£ di Chieti-Pescara"G. d'Annunzio"

Curated by ChEMBL
LigandPNGBDBM50026762(CHEMBL3331510)copy SMILEScopy InChI
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain membranes by liquid scintillation counting based competition binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9JS5PubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples"Federico II"

Curated by ChEMBL
LigandPNGBDBM50048692(CHEMBL3315140)copy SMILES
Affinity DataKi:  2nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples"Federico II"

Curated by ChEMBL
LigandPNGBDBM50048702(CHEMBL3315149)copy SMILES
Affinity DataKi:  2.20nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universit£ di Chieti-Pescara"G. d'Annunzio"

Curated by ChEMBL
LigandPNGBDBM21014((2S)-2-amino-N-[(1R)-1-[({[(1S)-1-{N'-[(2S)-2-{2-[...)copy SMILEScopy InChI
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Wistar rat brain membranes by liquid scintillation counting based competition binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9JS5PubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples"Federico II"

Curated by ChEMBL
LigandPNGBDBM50411333(URANTIDE)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Universit£ di Chieti-Pescara"G. d'Annunzio"

Curated by ChEMBL
LigandPNGBDBM50026762(CHEMBL3331510)copy SMILEScopy InChI
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]Ile5,6deltorphin II from delta opioid receptor in Wistar rat brain membranes by liquid scintillation counting based competition b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9JS5PubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Universit£ di Chieti-Pescara"G. d'Annunzio"

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)copy SMILEScopy InChI
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in Wistar rat brain membranes by liquid scintillation counting based competition binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9JS5PubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples"Federico II"

Curated by ChEMBL
LigandPNGBDBM50048690(CHEMBL3315143)copy SMILES
Affinity DataKi:  6.5nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples"Federico II"

Curated by ChEMBL
LigandPNGBDBM50048704(CHEMBL3315151)copy SMILES
Affinity DataKi:  12nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples"Federico II"

Curated by ChEMBL
LigandPNGBDBM50048698(CHEMBL3315145)copy SMILES
Affinity DataKi:  13nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Universit£ di Chieti-Pescara"G. d'Annunzio"

Curated by ChEMBL
LigandPNGBDBM21014((2S)-2-amino-N-[(1R)-1-[({[(1S)-1-{N'-[(2S)-2-{2-[...)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:Displacement of [3H]Ile5,6deltorphin II from delta opioid receptor in Wistar rat brain membranes by liquid scintillation counting based competition b...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9JS5PubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University of Naples"Federico II"

Curated by ChEMBL
LigandPNGBDBM50048706(CHEMBL3315153)copy SMILES
Affinity DataKi:  17nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC91NBPubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50229787((4S,5R)-Nutlin-3 | (rac)-(4,5-bis(4-chlorophenyl)-...)copy SMILEScopy InChI
Affinity DataKi:  43nMAssay Description:Binding affinity to 6xHis-taged MDM2 (unknown origin) expressed in Escherichia coli Gold (DE3) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Universit£ di Chieti-Pescara"G. d'Annunzio"

Curated by ChEMBL
LigandPNGBDBM50026762(CHEMBL3331510)copy SMILEScopy InChI
Affinity DataKi:  258nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in Wistar rat brain membranes by liquid scintillation counting based competition binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9JS5PubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Universit£ di Chieti-Pescara"G. d'Annunzio"

Curated by ChEMBL
LigandPNGBDBM21014((2S)-2-amino-N-[(1R)-1-[({[(1S)-1-{N'-[(2S)-2-{2-[...)copy SMILEScopy InChI
Affinity DataKi:  283nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in Wistar rat brain membranes by liquid scintillation counting based competition binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9JS5PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)copy SMILES
Affinity DataIC50: 1.10nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC4R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6FF7PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50453125(CHEMBL4214826)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6FF7PubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)copy SMILES
Affinity DataIC50: 1.20nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC1R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6FF7PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)copy SMILES
Affinity DataIC50: 1.20nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6FF7PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50453133(CHEMBL4211275)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6FF7PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50453126(CHEMBL4208874)copy SMILEScopy InChI
Affinity DataIC50: 3.90nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6FF7PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50453137(CHEMBL4217528)copy SMILEScopy InChI
Affinity DataIC50: 4.40nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6FF7PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50453138(CHEMBL4212209)copy SMILEScopy InChI
Affinity DataIC50: 5.10nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6FF7PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50453132(CHEMBL4207725)copy SMILEScopy InChI
Affinity DataIC50: 5.20nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC4R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6FF7PubMed
TargetDelta-type opioid receptor(MOUSE)
Universit£ di Chieti-Pescara"G. d'Annunzio"

Curated by ChEMBL
LigandPNGBDBM50026762(CHEMBL3331510)copy SMILEScopy InChI
Affinity DataIC50: 7.20nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-induced smooth muscle contractionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9JS5PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)copy SMILES
Affinity DataIC50: 7.5nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC5R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6FF7PubMed
TargetMu-type opioid receptor(GUINEA PIG)
Universit£ di Chieti-Pescara"G. d'Annunzio"

Curated by ChEMBL
LigandPNGBDBM21014((2S)-2-amino-N-[(1R)-1-[({[(1S)-1-{N'-[(2S)-2-{2-[...)copy SMILEScopy InChI
Affinity DataIC50: 8.80nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig ileum longitudinal muscle myenteric plexus assessed as inhibition of electrically-induce...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9JS5PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50453135(CHEMBL4204975)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6FF7PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50453130(CHEMBL4206406)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6FF7PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50453128(CHEMBL4207858)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC5R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6FF7PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50453131(CHEMBL4212629)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6FF7PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50453134(CHEMBL4216654)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6FF7PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50453137(CHEMBL4217528)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC5R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6FF7PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50453132(CHEMBL4207725)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6FF7PubMed
TargetMu-type opioid receptor(GUINEA PIG)
Universit£ di Chieti-Pescara"G. d'Annunzio"

Curated by ChEMBL
LigandPNGBDBM50026762(CHEMBL3331510)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig ileum longitudinal muscle myenteric plexus assessed as inhibition of electrically-induce...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9JS5PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
University of Naples "Federico II"

Curated by ChEMBL
LigandPNGBDBM50453133(CHEMBL4211275)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC5R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22J6FF7PubMed
TargetDelta-type opioid receptor(MOUSE)
Universit£ di Chieti-Pescara"G. d'Annunzio"

Curated by ChEMBL
LigandPNGBDBM21014((2S)-2-amino-N-[(1R)-1-[({[(1S)-1-{N'-[(2S)-2-{2-[...)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-induced smooth muscle contractionMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23T9JS5PubMed
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