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Found 93 with Last Name = 'martinez gil' and Initial = 'a'
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS

US Patent
LigandPNGBDBM350906(3-Phenyl-2-(2-naphthylmethylthio)-4-oxo-3,4-dihydr...)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Measurement of PDE7 inhibition was carried out using a commercial phosphodiesterase activity measurement kit.Some of the compounds of the present inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MDCUS Patent
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS

US Patent
LigandPNGBDBM350888(3-Phenyl-2-neopentylthio-4-oxo-3,4-dihydroquinazol...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Measurement of PDE7 inhibition was carried out using a commercial phosphodiesterase activity measurement kit.Some of the compounds of the present inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MDCUS Patent
LigandPNGBDBM50526882(CHEMBL4527232 | US11912678, Compound 2)copy SMILEScopy InChI
Affinity DataIC50: 108nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS

US Patent
LigandPNGBDBM350903(3-(2-Methylphenyl)-2-(3-pyridylmethylthio)-4-oxo-3...)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Measurement of PDE7 inhibition was carried out using a commercial phosphodiesterase activity measurement kit.Some of the compounds of the present inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MDCUS Patent
LigandPNGBDBM50526883(CHEMBL4455001 | US11912678, Compound 7)copy SMILEScopy InChI
Affinity DataIC50: 158nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50526881(CHEMBL4473326 | US11912678, Compound 6)copy SMILEScopy InChI
Affinity DataIC50: 190nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS

US Patent
LigandPNGBDBM350886(2-Cyclohexylmethylthio-3-phenyl-4-oxo-3,4-dihydroq...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Measurement of PDE7 inhibition was carried out using a commercial phosphodiesterase activity measurement kit.Some of the compounds of the present inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MDCUS Patent
LigandPNGBDBM50526878(CHEMBL4450247 | US11912678, Compound 3)copy SMILEScopy InChI
Affinity DataIC50: 293nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50526883(CHEMBL4455001 | US11912678, Compound 7)copy SMILEScopy InChI
Affinity DataIC50: 308nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50526887(CHEMBL4445322 | US11912678, Compound 4)copy SMILEScopy InChI
Affinity DataIC50: 332nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50526879(CHEMBL4565316 | US11912678, Compound 1)copy SMILEScopy InChI
Affinity DataIC50: 360nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50526882(CHEMBL4527232 | US11912678, Compound 2)copy SMILEScopy InChI
Affinity DataIC50: 368nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50526881(CHEMBL4473326 | US11912678, Compound 6)copy SMILEScopy InChI
Affinity DataIC50: 426nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50526889(CHEMBL4452771 | US11912678, Compound 8)copy SMILEScopy InChI
Affinity DataIC50: 474nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50526887(CHEMBL4445322 | US11912678, Compound 4)copy SMILEScopy InChI
Affinity DataIC50: 523nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS

US Patent
LigandPNGBDBM350902(8-Chloro-2-(3-pyridylmethylthio)-4-oxo-3,4-dihydro...)copy SMILEScopy InChI
Affinity DataIC50: 540nMAssay Description:Measurement of PDE7 inhibition was carried out using a commercial phosphodiesterase activity measurement kit.Some of the compounds of the present inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MDCUS Patent
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS

US Patent
LigandPNGBDBM350899(2-Benzylthio-3-phenyl-4-oxo-3,4-dihydroquinazoline...)copy SMILEScopy InChI
Affinity DataIC50: 600nMAssay Description:Measurement of PDE7 inhibition was carried out using a commercial phosphodiesterase activity measurement kit.Some of the compounds of the present inv...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MDCUS Patent
LigandPNGBDBM50526879(CHEMBL4565316 | US11912678, Compound 1)copy SMILEScopy InChI
Affinity DataIC50: 696nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS

US Patent
LigandPNGBDBM350901(3-Phenyl-2-(3-pyridylmethylthio)-4-oxo-3,4-dihydro...)copy SMILEScopy InChI
Affinity DataIC50: 700nMAssay Description:Measurement of PDE7 inhibition was carried out using a commercial phosphodiesterase activity measurement kit.Some of the compounds of the present inv...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MDCUS Patent
LigandPNGBDBM50526890(CHEMBL4437566 | US11912678, Compound 5)copy SMILEScopy InChI
Affinity DataIC50: 777nMMore data for this Ligand-Target Pair
In DepthDetails
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS

US Patent
LigandPNGBDBM350900(3-Phenyl-2-(2-pyridylmethylthio)-4-oxo-3,4-dihydro...)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Measurement of PDE7 inhibition was carried out using a commercial phosphodiesterase activity measurement kit.Some of the compounds of the present inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MDCUS Patent
LigandPNGBDBM50526878(CHEMBL4450247 | US11912678, Compound 3)copy SMILEScopy InChI
Affinity DataIC50: 1.06E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM653909(N-(6-isopropylbenzothiazole-2-yl)-4-morpholinobenz...)copy SMILES
Affinity DataIC50: 1.17E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50526888(CHEMBL4543902 | US11912678, Compound 9)copy SMILEScopy InChI
Affinity DataIC50: 1.19E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS

US Patent
LigandPNGBDBM350890(8-Chloro-3-phenyl-2-neopentylthio-4-oxo-3,4-dihydr...)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Measurement of PDE7 inhibition was carried out using a commercial phosphodiesterase activity measurement kit.Some of the compounds of the present inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MDCUS Patent
LigandPNGBDBM50526889(CHEMBL4452771 | US11912678, Compound 8)copy SMILEScopy InChI
Affinity DataIC50: 1.38E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS

US Patent
LigandPNGBDBM350891(3-(2-Methylphenyl)-2-neopentylthio-4-oxo-3,4-dihyd...)copy SMILEScopy InChI
Affinity DataIC50: 1.85E+3nMAssay Description:Measurement of PDE7 inhibition was carried out using a commercial phosphodiesterase activity measurement kit.Some of the compounds of the present inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MDCUS Patent
LigandPNGBDBM653909(N-(6-isopropylbenzothiazole-2-yl)-4-morpholinobenz...)copy SMILES
Affinity DataIC50: 1.95E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294083(6-Bromo-N′-dodecanoyl-1-ethyl-4-hydroxy-2-ox...)copy SMILEScopy InChI
Affinity DataIC50: 2.01E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1FQRUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294083(6-Bromo-N′-dodecanoyl-1-ethyl-4-hydroxy-2-ox...)copy SMILEScopy InChI
Affinity DataIC50: 2.01E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3H5ZUS Patent
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS

US Patent
LigandPNGBDBM350887(3-(2-Bromophenyl)-2-cyclohexylmethylthio-4-oxo-3,4...)copy SMILEScopy InChI
Affinity DataIC50: 2.11E+3nMAssay Description:Measurement of PDE7 inhibition was carried out using a commercial phosphodiesterase activity measurement kit.Some of the compounds of the present inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MDCUS Patent
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS

US Patent
LigandPNGBDBM350898(8-Chloro-2-ethylthio-3-(2,6-difluorophenyl)-4-oxo-...)copy SMILEScopy InChI
Affinity DataIC50: 2.44E+3nMAssay Description:Measurement of PDE7 inhibition was carried out using a commercial phosphodiesterase activity measurement kit.Some of the compounds of the present inv...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MDCUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294091(7-Chloro-N′-dodecanoyl-1-ethyl-4-hydroxy-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 2.48E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1FQRUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294091(7-Chloro-N′-dodecanoyl-1-ethyl-4-hydroxy-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 2.48E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3H5ZUS Patent
TargetHigh affinity cAMP-specific 3',5'-cyclic phosphodiesterase 7A(Homo sapiens (Human))
CONSEJO SUPERIOR DE INVESTIGACIONES CIENTIFICAS

US Patent
LigandPNGBDBM350904(3-Phenyl-2-(4-pyridylmethylthio)-4-oxo-3,4-dihydro...)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+3nMAssay Description:Measurement of PDE7 inhibition was carried out using a commercial phosphodiesterase activity measurement kit.Some of the compounds of the present inv...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MDCUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM50384798(CHEMBL2037482 | US9585879, 6 | US9757369, 6)copy SMILEScopy InChI
Affinity DataIC50: 2.85E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3H5ZUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM50384798(CHEMBL2037482 | US9585879, 6 | US9757369, 6)copy SMILEScopy InChI
Affinity DataIC50: 2.85E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1FQRUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294072(7-Chloro-N′-dodecanoyl-4-hydroxy-2-oxo-2-hyd...)copy SMILEScopy InChI
Affinity DataIC50: 3.12E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1FQRUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM339879(7-Chloro-N′-dodecanoyl-4-hydroxy-2-oxo-2-hyd...)copy SMILEScopy InChI
Affinity DataIC50: 3.12E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3H5ZUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294087(6-Chloro-N′-dodecanoyl-1-ethyl-4-hydroxy-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 3.18E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1FQRUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294087(6-Chloro-N′-dodecanoyl-1-ethyl-4-hydroxy-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 3.18E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3H5ZUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM339885(6-Bromo-N′-dodecanoyl-4-hydroxy-2-oxo-2-hydr...)copy SMILEScopy InChI
Affinity DataIC50: 3.54E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3H5ZUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294078(6-Bromo-N′-dodecanoyl-4-hydroxy-2-oxo-2-hydr...)copy SMILES
Affinity DataIC50: 3.54E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1FQRUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM339886(6-Chloro-N′-dodecanoyl-4-hydroxy-2-oxo-2-hyd...)copy SMILEScopy InChI
Affinity DataIC50: 3.81E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3H5ZUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294079(6-Chloro-N′-dodecanoyl-4-hydroxy-2-oxo-2-hyd...)copy SMILES
Affinity DataIC50: 3.81E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1FQRUS Patent
LigandPNGBDBM50526888(CHEMBL4543902 | US11912678, Compound 9)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294089(7-Chloro-N′-dodecanoyl-4-hydroxy-1-methyl-2-...)copy SMILEScopy InChI
Affinity DataIC50: 4.03E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1FQRUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294089(7-Chloro-N′-dodecanoyl-4-hydroxy-1-methyl-2-...)copy SMILEScopy InChI
Affinity DataIC50: 4.03E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3H5ZUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294081(6-Bromo-N′-dodecanoyl-4-hydroxy-1-methyl-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 4.28E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NK3H5ZUS Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294081(6-Bromo-N′-dodecanoyl-4-hydroxy-1-methyl-2-o...)copy SMILEScopy InChI
Affinity DataIC50: 4.28E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1FQRUS Patent
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