Compile Data Set for Download or QSAR
Found 29 with Last Name = 'maruyama' and Initial = 'a'
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50403994(CHEMBL2114287)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:The compound was tested for the inhibitory activity against alpha-L-Fucosidase in bovine kidneyMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CF9PDKPubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50403995(CHEMBL2115269)copy SMILEScopy InChI
Affinity DataKi:  200nMAssay Description:The compound was tested for the inhibitory activity against alpha-L-Fucosidase in bovine kidneyMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CF9PDKPubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50403995(CHEMBL2115269)copy SMILEScopy InChI
Affinity DataKi:  200nMAssay Description:The compound was tested for the inhibitory activity against alpha-L-Fucosidase in bovine kidneyMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CF9PDKPubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50110400(1-Aminomethyl-5-methyl-cyclohexane-1,2,3,4-tetraol...)copy SMILEScopy InChI
Affinity DataKi:  2.80E+3nMAssay Description:The compound was tested for the inhibitory activity against alpha-L-Fucosidase in bovine kidneyMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CF9PDKPubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50110400(1-Aminomethyl-5-methyl-cyclohexane-1,2,3,4-tetraol...)copy SMILEScopy InChI
Affinity DataKi:  3.00E+3nMAssay Description:The compound was tested for the inhibitory activity against alpha-L-Fucosidase in bovine kidneyMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CF9PDKPubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50110399(6-Amino-4-methyl-cyclohex-4-ene-1,2,3-triol | CHEM...)copy SMILEScopy InChI
Affinity DataKi:  4.50E+4nMAssay Description:The compound was tested for the inhibitory activity against alpha-L-Fucosidase in bovine kidneyMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CF9PDKPubMed
TargetTissue alpha-L-fucosidase(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50110399(6-Amino-4-methyl-cyclohex-4-ene-1,2,3-triol | CHEM...)copy SMILEScopy InChI
Affinity DataKi:  4.50E+4nMAssay Description:The compound was tested for the inhibitory activity against alpha-L-Fucosidase in bovine kidneyMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CF9PDKPubMed
TargetGlucocorticoid receptor(RAT)
Mitsubishi Kasei Corporation

Curated by ChEMBL
LigandPNGBDBM39347(CLOBETASOL PROPIONATE | MLS000028708 | SMR00005874...)copy SMILEScopy InChI
Affinity DataIC50: 3.20nMAssay Description:Competitive displacement of [3H]dexamethasone from glucocorticoid receptor of rat liver cytosolMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W096H9PubMed
TargetGlucocorticoid receptor(RAT)
Mitsubishi Kasei Corporation

Curated by ChEMBL
LigandPNGBDBM50009401(CHEMBL315931 | Succinic acid 17-(2-chloro-acetyl)-...)copy SMILEScopy InChI
Affinity DataIC50: 5.20nMAssay Description:Competitive displacement of [3H]dexamethasone from glucocorticoid receptor of rat liver cytosolMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W096H9PubMed
TargetGlucocorticoid receptor(RAT)
Mitsubishi Kasei Corporation

Curated by ChEMBL
LigandPNGBDBM50421892(Alphatrex | BETAMETHASONE DIPROPIONATE | Diprolene...)copy SMILEScopy InChI
Affinity DataIC50: 5.30nMAssay Description:Competitive displacement of [3H]dexamethasone from glucocorticoid receptor of rat liver cytosolMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W096H9PubMed
TargetGlucocorticoid receptor(RAT)
Mitsubishi Kasei Corporation

Curated by ChEMBL
LigandPNGBDBM50009403(CHEMBL81387 | Pentanedioic acid 17-(2-chloro-acety...)copy SMILEScopy InChI
Affinity DataIC50: 9.70nMAssay Description:Competitive displacement of [3H]dexamethasone from glucocorticoid receptor of rat liver cytosolMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W096H9PubMed
TargetGlucocorticoid receptor(RAT)
Mitsubishi Kasei Corporation

Curated by ChEMBL
LigandPNGBDBM50009402(CHEMBL83845 | Succinic acid tert-butyl ester 17-(2...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Competitive displacement of [3H]dexamethasone from glucocorticoid receptor of rat liver cytosolMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W096H9PubMed
TargetGlucocorticoid receptor(RAT)
Mitsubishi Kasei Corporation

Curated by ChEMBL
LigandPNGBDBM50009406(CHEMBL311802 | Succinic acid 17-(2-chloro-acetyl)-...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Competitive displacement of [3H]dexamethasone from glucocorticoid receptor of rat liver cytosolMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W096H9PubMed
TargetGlucocorticoid receptor(RAT)
Mitsubishi Kasei Corporation

Curated by ChEMBL
LigandPNGBDBM50009405(CHEMBL311457 | Succinic acid mono-[17-(2-chloro-ac...)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Competitive displacement of [3H]dexamethasone from glucocorticoid receptor of rat liver cytosolMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2W096H9PubMed
TargetThromboxane-A synthase(Rattus norvegicus)
Chugai Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50017896((E)-3-(4-Imidazol-1-ylmethyl-phenyl)-acrylic acid ...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in rat whole bloodMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QJ7GBKPubMed
TargetThromboxane-A synthase(Rattus norvegicus)
Chugai Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50017896((E)-3-(4-Imidazol-1-ylmethyl-phenyl)-acrylic acid ...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in rat plateletMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QJ7GBKPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Chugai Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50017896((E)-3-(4-Imidazol-1-ylmethyl-phenyl)-acrylic acid ...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in human plateletMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QJ7GBKPubMed
TargetThromboxane-A synthase(Rattus norvegicus)
Chugai Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50043282(2-Methyl-4-thiazol-5-yl-2H-phthalazin-1-one | CHEM...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in rat plateletMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QJ7GBKPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Chugai Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50017896((E)-3-(4-Imidazol-1-ylmethyl-phenyl)-acrylic acid ...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in human plateletMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QJ7GBKPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Chugai Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50043282(2-Methyl-4-thiazol-5-yl-2H-phthalazin-1-one | CHEM...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in human plateletMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QJ7GBKPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Chugai Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50017896((E)-3-(4-Imidazol-1-ylmethyl-phenyl)-acrylic acid ...)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QJ7GBKPubMed
TargetThromboxane-A synthase(Rattus norvegicus)
Chugai Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50043283(2-Ethyl-4-pyridin-3-yl-2H-phthalazin-1-one | CHEMB...)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in rat plateletMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QJ7GBKPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Chugai Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50043283(2-Ethyl-4-pyridin-3-yl-2H-phthalazin-1-one | CHEMB...)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in human microsomeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QJ7GBKPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Chugai Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50043283(2-Ethyl-4-pyridin-3-yl-2H-phthalazin-1-one | CHEMB...)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in human microsomeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QJ7GBKPubMed
TargetThromboxane-A synthase(Rattus norvegicus)
Chugai Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50043283(2-Ethyl-4-pyridin-3-yl-2H-phthalazin-1-one | CHEMB...)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in rat whole bloodMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QJ7GBKPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Chugai Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50043283(2-Ethyl-4-pyridin-3-yl-2H-phthalazin-1-one | CHEMB...)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+3nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QJ7GBKPubMed
TargetThromboxane-A synthase(Rattus norvegicus)
Chugai Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50043282(2-Methyl-4-thiazol-5-yl-2H-phthalazin-1-one | CHEM...)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+3nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in rat whole bloodMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QJ7GBKPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Chugai Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50043282(2-Methyl-4-thiazol-5-yl-2H-phthalazin-1-one | CHEM...)copy SMILEScopy InChI
Affinity DataIC50: 3.90E+3nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in human microsomeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QJ7GBKPubMed
TargetThromboxane-A synthase(Homo sapiens (Human))
Chugai Pharmaceutical Company, Ltd.

Curated by ChEMBL
LigandPNGBDBM50043282(2-Methyl-4-thiazol-5-yl-2H-phthalazin-1-one | CHEM...)copy SMILEScopy InChI
Affinity DataIC50: 8.70E+3nMAssay Description:Tested in vitro against TXA2 synthetase inhibitory activity in human whole bloodMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QJ7GBKPubMed