Compile Data Set for Download or QSAR
Found 135 with Last Name = 'massaro' and Initial = 'a'
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"

Curated by ChEMBL
LigandPNGBDBM81395(APO-866)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Noncompetitive inhibition of NAMPT (unknown origin)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50001775((ritanserin)6-(2-{4-[Bis-(4-fluoro-phenyl)-methyle...)copy SMILEScopy InChI
Affinity DataKi:  0.450nMAssay Description:Binding affinity to 5HT2A receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01B01PubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50001775((ritanserin)6-(2-{4-[Bis-(4-fluoro-phenyl)-methyle...)copy SMILEScopy InChI
Affinity DataKi:  0.450nMAssay Description:Binding affinity to 5HT2A receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01B01PubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50001775((ritanserin)6-(2-{4-[Bis-(4-fluoro-phenyl)-methyle...)copy SMILEScopy InChI
Affinity DataKi:  0.710nMAssay Description:Binding affinity to 5HT2C receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01B01PubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50001775((ritanserin)6-(2-{4-[Bis-(4-fluoro-phenyl)-methyle...)copy SMILEScopy InChI
Affinity DataKi:  0.710nMAssay Description:Binding affinity to 5HT2C receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01B01PubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Florence

Curated by ChEMBL
LigandPNGBDBM50434226(CHEMBL2385483)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B859HTPubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Florence

Curated by ChEMBL
LigandPNGBDBM50294120(2-(biphenyl-4-ylsulfonamido)-N-hydroxyacetamide | ...)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Florence

Curated by ChEMBL
LigandPNGBDBM50434222(CHEMBL2385487)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B859HTPubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Florence

Curated by ChEMBL
LigandPNGBDBM50434224(CHEMBL2385485)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B859HTPubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Florence

Curated by ChEMBL
LigandPNGBDBM50434213(CHEMBL2385489)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B859HTPubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Florence

Curated by ChEMBL
LigandPNGBDBM50434221(CHEMBL2385490)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B859HTPubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Florence

Curated by ChEMBL
LigandPNGBDBM50434223(CHEMBL2385486)copy SMILEScopy InChI
Affinity DataKi:  7nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B859HTPubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Florence

Curated by ChEMBL
LigandPNGBDBM50434219(CHEMBL2385492)copy SMILEScopy InChI
Affinity DataKi:  9nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B859HTPubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Florence

Curated by ChEMBL
LigandPNGBDBM50434227(CHEMBL2385482)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Florence

Curated by ChEMBL
LigandPNGBDBM50434225(CHEMBL2385484)copy SMILEScopy InChI
Affinity DataKi:  10nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B859HTPubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Florence

Curated by ChEMBL
LigandPNGBDBM50434214(CHEMBL2385488)copy SMILEScopy InChI
Affinity DataKi:  15nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B859HTPubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Florence

Curated by ChEMBL
LigandPNGBDBM50434215(CHEMBL2385481)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Florence

Curated by ChEMBL
LigandPNGBDBM11328(CHEMBL83508 | Hydroxamate 9 | N-hydroxy-2-[(4-meth...)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Florence

Curated by ChEMBL
LigandPNGBDBM50434216(CHEMBL2385480)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Florence

Curated by ChEMBL
LigandPNGBDBM50434217(CHEMBL2385479)copy SMILEScopy InChI
Affinity DataKi:  62nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B859HTPubMedMMDB
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Florence

Curated by ChEMBL
LigandPNGBDBM50434220(CHEMBL2385491)copy SMILEScopy InChI
Affinity DataKi:  272nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B859HTPubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Florence

Curated by ChEMBL
LigandPNGBDBM50434218(CHEMBL2385493)copy SMILEScopy InChI
Affinity DataKi:  672nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B859HTPubMed
TargetDiacylglycerol kinase alpha(Homo sapiens)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50529935(COCHLIOQUINONE A)copy SMILEScopy InChI
Affinity DataKi:  2.26E+3nMAssay Description:Inhibition of DGKalpha in human erythrocytes using OAG as substrate preincubated for 1 min followed by OAG addition and measured after 8 mins in pres...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01B01PubMed
TargetDiacylglycerol kinase alpha(Homo sapiens)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50529935(COCHLIOQUINONE A)copy SMILEScopy InChI
Affinity DataKi:  2.26E+3nMAssay Description:Inhibition of DGKalpha in human erythrocytes using OAG as substrate preincubated for 1 min followed by OAG addition and measured after 8 mins in pres...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01B01PubMed
TargetDiacylglycerol kinase alpha(Homo sapiens)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50529932(STEMPHONE)copy SMILEScopy InChI
Affinity DataKi:  3.32E+3nMAssay Description:Inhibition of DGKalpha in human erythrocytes using OAG as substrate preincubated for 1 min followed by OAG addition and measured after 8 mins in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01B01PubMed
TargetDiacylglycerol kinase alpha(Homo sapiens)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50529932(STEMPHONE)copy SMILEScopy InChI
Affinity DataKi:  3.32E+3nMAssay Description:Inhibition of DGKalpha in human erythrocytes using OAG as substrate preincubated for 1 min followed by OAG addition and measured after 8 mins in pres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01B01PubMed
TargetMatrilysin(Homo sapiens (Human))
University of Florence

Curated by ChEMBL
LigandPNGBDBM50434217(CHEMBL2385479)copy SMILEScopy InChI
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of MMP7 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B859HTPubMed
TargetMatrilysin(Homo sapiens (Human))
University of Florence

Curated by ChEMBL
LigandPNGBDBM11328(CHEMBL83508 | Hydroxamate 9 | N-hydroxy-2-[(4-meth...)copy SMILEScopy InChI
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of MMP7 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B859HTPubMed
TargetMatrilysin(Homo sapiens (Human))
University of Florence

Curated by ChEMBL
LigandPNGBDBM50294120(2-(biphenyl-4-ylsulfonamido)-N-hydroxyacetamide | ...)copy SMILEScopy InChI
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of MMP7 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B859HTPubMed
TargetMatrilysin(Homo sapiens (Human))
University of Florence

Curated by ChEMBL
LigandPNGBDBM50434213(CHEMBL2385489)copy SMILEScopy InChI
Affinity DataKi:  6.00E+3nMAssay Description:Inhibition of MMP7 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B859HTPubMed
TargetMatrilysin(Homo sapiens (Human))
University of Florence

Curated by ChEMBL
LigandPNGBDBM50434215(CHEMBL2385481)copy SMILEScopy InChI
Affinity DataKi:  7.00E+3nMAssay Description:Inhibition of MMP7 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B859HTPubMed
TargetMatrilysin(Homo sapiens (Human))
University of Florence

Curated by ChEMBL
LigandPNGBDBM50434216(CHEMBL2385480)copy SMILEScopy InChI
Affinity DataKi:  1.07E+4nMAssay Description:Inhibition of MMP7 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B859HTPubMed
TargetMacrophage metalloelastase(Homo sapiens (Human))
University of Florence

Curated by ChEMBL
LigandPNGBDBM50400562(CHEMBL1335679)copy SMILEScopy InChI
Affinity DataKi:  1.80E+4nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B859HTPubMed
TargetMatrilysin(Homo sapiens (Human))
University of Florence

Curated by ChEMBL
LigandPNGBDBM50434214(CHEMBL2385488)copy SMILEScopy InChI
Affinity DataKi:  1.85E+4nMAssay Description:Inhibition of MMP7 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B859HTPubMed
TargetDiacylglycerol kinase alpha(Homo sapiens)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50529934(ETHYLENE GLYCOL DIOCTANOATE)copy SMILEScopy InChI
Affinity DataKi:  5.80E+4nMAssay Description:Inhibition of DGKalpha in human erythrocytes using OAG as substrate preincubated for 1 min followed by OAG addition and measured after 8 mins in pres...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01B01PubMed
TargetDiacylglycerol kinase alpha(Homo sapiens)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50529934(ETHYLENE GLYCOL DIOCTANOATE)copy SMILEScopy InChI
Affinity DataKi:  5.80E+4nMAssay Description:Inhibition of DGKalpha in human erythrocytes using OAG as substrate preincubated for 1 min followed by OAG addition and measured after 8 mins in pres...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01B01PubMed
TargetDiacylglycerol kinase alpha(Homo sapiens)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50529937(CHEBI:75342 | Glyceryl monooleate)copy SMILEScopy InChI
Affinity DataKi:  9.10E+4nMAssay Description:Inhibition of DGKalpha in human erythrocytes using OAG as substrate preincubated for 1 min followed by OAG addition and measured after 8 mins in pres...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01B01PubMed
TargetDiacylglycerol kinase alpha(Homo sapiens)
University of Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50529937(CHEBI:75342 | Glyceryl monooleate)copy SMILEScopy InChI
Affinity DataKi:  9.10E+4nMAssay Description:Inhibition of DGKalpha in human erythrocytes using OAG as substrate preincubated for 1 min followed by OAG addition and measured after 8 mins in pres...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N01B01PubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"

Curated by ChEMBL
LigandPNGBDBM50439676(CHEMBL2417796)copy SMILEScopy InChI
Affinity DataIC50: 0.230nMAssay Description:Inhibition of NAMPT (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4XJ8PubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"

Curated by ChEMBL
LigandPNGBDBM50347432(CHEMBL1801863)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Inhibition of NAMPT (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4XJ8PubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"

Curated by ChEMBL
LigandPNGBDBM50347433(CHEMBL1801864)copy SMILEScopy InChI
Affinity DataIC50: 0.450nMAssay Description:Inhibition of NAMPT (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4XJ8PubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"

Curated by ChEMBL
LigandPNGBDBM50439675(CHEMBL2417788 | US11279687, Compound 196)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of NAMPT (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4XJ8PubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"

Curated by ChEMBL
LigandPNGBDBM50439678(CHEMBL2417789)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:Inhibition of recombinant his-tagged NAMPT (unknown origin) expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4XJ8PubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"

Curated by ChEMBL
LigandPNGBDBM50439677(CHEMBL2417790 | US9169209, Table 3, Compound 55)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of recombinant his-tagged NAMPT (unknown origin) expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4XJ8PubMed
TargetNicotinamide phosphoribosyltransferase(Mus musculus)
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"

Curated by ChEMBL
LigandPNGBDBM50236217(CHEMBL4061448)copy SMILEScopy InChI
Affinity DataIC50: 3.10nMAssay Description:Inhibition of recombinant mouse NAMPT expressed in bacterial expression system using nicotinamide as substrate after 1 hr by fluorescence based NMNAT...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ63TKPubMed
TargetNicotinamide phosphoribosyltransferase(Mus musculus)
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"

Curated by ChEMBL
LigandPNGBDBM50236220(CHEMBL4074848)copy SMILEScopy InChI
Affinity DataIC50: 3.80nMAssay Description:Inhibition of recombinant mouse NAMPT expressed in bacterial expression system using nicotinamide as substrate after 1 hr by fluorescence based NMNAT...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ63TKPubMed
TargetNicotinamide phosphoribosyltransferase(Mus musculus)
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"

Curated by ChEMBL
LigandPNGBDBM81395(APO-866)copy SMILEScopy InChI
Affinity DataIC50: 4.90nMAssay Description:Inhibition of recombinant mouse NAMPT expressed in bacterial expression system using nicotinamide as substrate after 1 hr by fluorescence based NMNAT...More data for this Ligand-Target Pair
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"

Curated by ChEMBL
LigandPNGBDBM50236217(CHEMBL4061448)copy SMILEScopy InChI
Affinity DataIC50: 4.90nMAssay Description:Inhibition of NAMPT in human Jurkat T cells assessed as reduction in NAD levelsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TQ63TKPubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"

Curated by ChEMBL
LigandPNGBDBM50439680(CHEMBL2417798)copy SMILEScopy InChI
Affinity DataIC50: 5.40nMAssay Description:Inhibition of recombinant his-tagged NAMPT (unknown origin) expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4XJ8PubMed
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"

Curated by ChEMBL
LigandPNGBDBM50439679(CHEMBL2417799)copy SMILEScopy InChI
Affinity DataIC50: 6.30nMAssay Description:Inhibition of recombinant his-tagged NAMPT (unknown origin) expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25Q4XJ8PubMed
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