TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"
Curated by ChEMBL
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Noncompetitive inhibition of NAMPT (unknown origin)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University of Piemonte Orientale
Curated by ChEMBL
University of Piemonte Orientale
Curated by ChEMBL
Affinity DataKi: 0.450nMAssay Description:Binding affinity to 5HT2A receptor (unknown origin)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University of Piemonte Orientale
Curated by ChEMBL
University of Piemonte Orientale
Curated by ChEMBL
Affinity DataKi: 0.450nMAssay Description:Binding affinity to 5HT2A receptor (unknown origin)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University of Piemonte Orientale
Curated by ChEMBL
University of Piemonte Orientale
Curated by ChEMBL
Affinity DataKi: 0.710nMAssay Description:Binding affinity to 5HT2C receptor (unknown origin)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University of Piemonte Orientale
Curated by ChEMBL
University of Piemonte Orientale
Curated by ChEMBL
Affinity DataKi: 0.710nMAssay Description:Binding affinity to 5HT2C receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 62nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 272nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 672nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.26E+3nMAssay Description:Inhibition of DGKalpha in human erythrocytes using OAG as substrate preincubated for 1 min followed by OAG addition and measured after 8 mins in pres...More data for this Ligand-Target Pair
Affinity DataKi: 2.26E+3nMAssay Description:Inhibition of DGKalpha in human erythrocytes using OAG as substrate preincubated for 1 min followed by OAG addition and measured after 8 mins in pres...More data for this Ligand-Target Pair
Affinity DataKi: 3.32E+3nMAssay Description:Inhibition of DGKalpha in human erythrocytes using OAG as substrate preincubated for 1 min followed by OAG addition and measured after 8 mins in pres...More data for this Ligand-Target Pair
Affinity DataKi: 3.32E+3nMAssay Description:Inhibition of DGKalpha in human erythrocytes using OAG as substrate preincubated for 1 min followed by OAG addition and measured after 8 mins in pres...More data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nMAssay Description:Inhibition of MMP7 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nMAssay Description:Inhibition of MMP7 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.00E+3nMAssay Description:Inhibition of MMP7 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.00E+3nMAssay Description:Inhibition of MMP7 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.00E+3nMAssay Description:Inhibition of MMP7 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.07E+4nMAssay Description:Inhibition of MMP7 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.80E+4nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.85E+4nMAssay Description:Inhibition of MMP7 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.80E+4nMAssay Description:Inhibition of DGKalpha in human erythrocytes using OAG as substrate preincubated for 1 min followed by OAG addition and measured after 8 mins in pres...More data for this Ligand-Target Pair
Affinity DataKi: 5.80E+4nMAssay Description:Inhibition of DGKalpha in human erythrocytes using OAG as substrate preincubated for 1 min followed by OAG addition and measured after 8 mins in pres...More data for this Ligand-Target Pair
Affinity DataKi: 9.10E+4nMAssay Description:Inhibition of DGKalpha in human erythrocytes using OAG as substrate preincubated for 1 min followed by OAG addition and measured after 8 mins in pres...More data for this Ligand-Target Pair
Affinity DataKi: 9.10E+4nMAssay Description:Inhibition of DGKalpha in human erythrocytes using OAG as substrate preincubated for 1 min followed by OAG addition and measured after 8 mins in pres...More data for this Ligand-Target Pair
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"
Curated by ChEMBL
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"
Curated by ChEMBL
Affinity DataIC50: 0.230nMAssay Description:Inhibition of NAMPT (unknown origin)More data for this Ligand-Target Pair
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"
Curated by ChEMBL
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of NAMPT (unknown origin)More data for this Ligand-Target Pair
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"
Curated by ChEMBL
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"
Curated by ChEMBL
Affinity DataIC50: 0.450nMAssay Description:Inhibition of NAMPT (unknown origin)More data for this Ligand-Target Pair
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"
Curated by ChEMBL
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Inhibition of NAMPT (unknown origin)More data for this Ligand-Target Pair
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"
Curated by ChEMBL
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"
Curated by ChEMBL
Affinity DataIC50: 2.60nMAssay Description:Inhibition of recombinant his-tagged NAMPT (unknown origin) expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"
Curated by ChEMBL
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of recombinant his-tagged NAMPT (unknown origin) expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetNicotinamide phosphoribosyltransferase(Mus musculus)
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"
Curated by ChEMBL
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"
Curated by ChEMBL
Affinity DataIC50: 3.10nMAssay Description:Inhibition of recombinant mouse NAMPT expressed in bacterial expression system using nicotinamide as substrate after 1 hr by fluorescence based NMNAT...More data for this Ligand-Target Pair
TargetNicotinamide phosphoribosyltransferase(Mus musculus)
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"
Curated by ChEMBL
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"
Curated by ChEMBL
Affinity DataIC50: 3.80nMAssay Description:Inhibition of recombinant mouse NAMPT expressed in bacterial expression system using nicotinamide as substrate after 1 hr by fluorescence based NMNAT...More data for this Ligand-Target Pair
TargetNicotinamide phosphoribosyltransferase(Mus musculus)
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"
Curated by ChEMBL
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"
Curated by ChEMBL
Affinity DataIC50: 4.90nMAssay Description:Inhibition of recombinant mouse NAMPT expressed in bacterial expression system using nicotinamide as substrate after 1 hr by fluorescence based NMNAT...More data for this Ligand-Target Pair
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"
Curated by ChEMBL
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"
Curated by ChEMBL
Affinity DataIC50: 4.90nMAssay Description:Inhibition of NAMPT in human Jurkat T cells assessed as reduction in NAD levelsMore data for this Ligand-Target Pair
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"
Curated by ChEMBL
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"
Curated by ChEMBL
Affinity DataIC50: 5.40nMAssay Description:Inhibition of recombinant his-tagged NAMPT (unknown origin) expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
TargetNicotinamide phosphoribosyltransferase(Homo sapiens (Human))
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"
Curated by ChEMBL
Universit£ degli Studi del Piemonte Orientale"A. Avogadro"
Curated by ChEMBL
Affinity DataIC50: 6.30nMAssay Description:Inhibition of recombinant his-tagged NAMPT (unknown origin) expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair