Found 115 with Last Name = 'mizusawa' and Initial = 'a' TargetProteasome subunit beta type-5(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
3D Structure (crystal)TargetProteasome subunit beta type-1(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of PGPH activity of human 26S proteasome using Z-LLE-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Boc-LRR-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 280nMAssay Description:Inhibition of PGPH activity of human 20S proteasome using Z-LLE-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 350nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Boc-LRR-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 370nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of PGPH activity of human 20S proteasome using Z-LLE-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 720nMAssay Description:Inhibition of PGPH activity of human 20S proteasome using Z-LLE-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 890nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 890nMAssay Description:Inhibition of PGPH activity of human 20S proteasome using Z-LLE-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 890nMAssay Description:Inhibition of PGPH activity of human 20S proteasome using Z-LLE-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 890nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 990nMAssay Description:Inhibition of PGPH activity of human 20S proteasome using Z-LLE-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Boc-LRR-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 1.93E+3nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Boc-LRR-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome in human KMS11 cells using Suc-LLVY-MCA as substrate after 24 to 48 hrs by luminescence-ba...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome in human RPMI8226 cells using Suc-LLVY-MCA as substrate after 24 to 48 hrs by luminescence...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 26S proteasome using Suc-LLVY-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 26S proteasome using Z-LLE-MCA as substrate measured for 1 hr in presence of ATPgammaS by fluoresce...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of PGPH-like activity of 26S proteasome in human KMS11 cells using Z-LLE-MCA as substrate after 24 to 48 hrs by luminescence-based assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of PGPH-like activity of 26S proteasome in human RPMI8226 cells using Z-LLE-MCA as substrate after 24 to 48 hrs by luminescence-based assa...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Boc-LRR-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 3.25E+3nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Boc-LRR-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of PGPH activity of human 20S proteasome using Z-LLE-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Boc-LRR-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Boc-LRR-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Boc-LRR-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of trypsin-like activity of 26S proteasome in human KMS11 cells using Boc-LRR-MCA as substrate after 24 to 48 hrs by luminescence-based as...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 4.28E+3nMAssay Description:Inhibition of PGPH activity of human 20S proteasome using Z-LLE-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of PGPH activity of human 20S proteasome using Z-LLE-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 4.58E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of PGPH-like activity of 26S proteasome in human KMS11 cells using Z-LLE-MCA as substrate after 24 to 48 hrs by luminescence-based assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Boc-LRR-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 4.96E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 26S proteasome using Suc-LLVY-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 26S proteasome using Suc-LLVY-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 26S proteasome using Suc-LLVY-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome in human RPMI8226 cells using Suc-LLVY-MCA as substrate after 24 to 48 hrs by luminescence...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 26S proteasome using Z-LLE-MCA as substrate measured for 1 hr in presence of ATPgammaS by fluoresce...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome in human KMS11 cells using Suc-LLVY-MCA as substrate after 24 to 48 hrs by luminescence-ba...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of PGPH-like activity of 26S proteasome in human RPMI8226 cells using Z-LLE-MCA as substrate after 24 to 48 hrs by luminescence-based assa...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Boc-LRR-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of PGPH activity of human 20S proteasome using Z-LLE-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of PGPH activity of human 20S proteasome using Z-LLE-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of PGPH activity of human 20S proteasome using Z-LLE-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Nagahama Institute of Bio-Science and Technology
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Boc-LRR-MCA as substrate measured for 1 hr by fluorescence assayMore data for this Ligand-Target Pair
